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TRV120056 acetate

Name: TRV120056 acetate
Brand: TargetMol
SKU: T40508L
Price: 36 USD
Availability: InStock
Rating: 5 (10 reviews)

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Catalog No. T40508L

Alias TRV120056 acetate (40678-47-5 Free base)

TRV120056 acetate is a Gq-biased agonist with 10-fold greater molecular efficiency on AT1R-Gq fusion proteins than AT1R-βarr2 fusion proteins.

TRV120056 acetate

🥰Excellent

Purity: 99.16%

Catalog No. T40508LAlias TRV120056 acetate (40678-47-5 Free base)

TRV120056 acetate is a Gq-biased agonist with 10-fold greater molecular efficiency on AT1R-Gq fusion proteins than AT1R-βarr2 fusion proteins.

Pack Size	Price	Availability
5 mg	$36	In Stock
10 mg	$57	In Stock
25 mg	$103	In Stock
50 mg	$155	In Stock
100 mg	$233	In Stock
200 mg	$335	In Stock

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Batch Information

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Purity:99.16%

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COA HPLC MS

Product Introduction

Bioactivity

Description	TRV120056 acetate is a Gq-biased agonist with 10-fold greater molecular efficiency on AT1R-Gq fusion proteins than AT1R-βarr2 fusion proteins.
Synonyms	TRV120056 acetate (40678-47-5 Free base)

Chemical Properties

Molecular Weight	1016.11
Formula	C₄₅H₆₉N₁₃O₁₄
Smiles	O=C(N(CCC1)[C@@H]1C(NCC(O)=O)=O)[C@@H](NC([C@@]([C@H](C)CC)([H])NC([C@@H](NC([C@@H](C(C)C)NC([C@@H](CCCNC(N)=N)NC([C@@H](N)CC(O)=O)=O)=O)=O)CC2=CC=C(O)C=C2)=O)=O)CC3=CNC=N3.CC(O)=O
Sequence	Asp-Arg-Val-Tyr-Ile-His-Pro-Gly
Sequence Short	DRVYIHPG

Storage & Solubility Information

Storage

keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 10.16 mg/mL (10 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	0.9841 mL	4.9207 mL	9.8415 mL	49.2073 mL
5 mM	0.1968 mL	0.9841 mL	1.9683 mL	9.8415 mL
10 mM	0.0984 mL	0.4921 mL	0.9841 mL	4.9207 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc