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Pilsicainide
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Catalog No. T60482Cas No. 88069-67-4
Pilsicainide (SUN 1165 free acid) is a potent class Ic antiarrhythmic agent and a sodium channel blocker[1][2].
Pilsicainide
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Catalog No. T60482Cas No. 88069-67-4
Pilsicainide (SUN 1165 free acid) is a potent class Ic antiarrhythmic agent and a sodium channel blocker[1][2].
| Pack Size | Price | USA Warehouse | Global Warehouse | Quantity |
|---|---|---|---|---|
| 25 mg | $1,520 | 1-2 weeks | 1-2 weeks | |
| 50 mg | $1,980 | 1-2 weeks | 1-2 weeks | |
| 100 mg | $2,500 | 1-2 weeks | 1-2 weeks |
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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]
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Product Introduction
Bioactivity
Chemical Properties
| Description | Pilsicainide (SUN 1165 free acid) is a potent class Ic antiarrhythmic agent and a sodium channel blocker[1][2]. |
| In vitro | Pilsicainide (SUN 1165 free acid; 10-200 μg/mL) dose-dependently reduces the peak amplitude of the net inward current, with an IC50 of 29.2 μg/mL in levo-thyroxine (T4)-treated rat atrial cells [1]. |
| In vivo | Pilsicainide (SUN 1165 free acid; 2 mg/kg; i.v.; once) significantly reduces conduction velocity in the atrium of T4-treated male Sprague-Dawley rats (weighing 200-220 g) by decreasing Max dV/dt and net inward current, and altering electrocardiographic parameters. Administered as a bolus into the right external carotid vein over two minutes, pilsicainide extends the QT interval at 15 and 60 minutes post-administration, decreases the durations of P wave and QRS complex, reduces action potential amplitudes (APA) and Max dV/dt, and lengthens action potential duration. |
| Molecular Weight | 272.39 |
| Formula | C17H24N2O |
| Cas No. | 88069-67-4 |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature. |
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Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . A total of 10 animals were administered, and the formula you used is 5% 
DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH2O. So your working solution concentration is 2 mg/mL。Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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