MCHR1 antagonist 1

Name: MCHR1 antagonist 1
Brand: TargetMol
SKU: T10173
Rating: 4.5 (1 reviews)

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Catalog No. T10173Cas No. 391610-37-0

MCHR1 antagonist 1 is a selective antagonist of the melanin-concentrating hormone-1 (MCH1) receptor with a Kb of 1 nM and a Ki of 4 nM at the human MCH1 receptor.

MCHR1 antagonist 1

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Catalog No. T10173Cas No. 391610-37-0

MCHR1 antagonist 1 is a selective antagonist of the melanin-concentrating hormone-1 (MCH1) receptor with a Kb of 1 nM and a Ki of 4 nM at the human MCH1 receptor.

Pack Size	Price	Availability
25 mg	$1,520	6-8 weeks
50 mg	$1,980	6-8 weeks
100 mg	$2,500	6-8 weeks

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Product Introduction

Bioactivity

Description	MCHR1 antagonist 1 is a selective antagonist of the melanin-concentrating hormone-1 (MCH1) receptor with a Kb of 1 nM and a Ki of 4 nM at the human MCH1 receptor.
Targets&IC50	MCH1 (human): ki： 4 nM , MCH1 (human): 1 nM (Kb)
In vitro	MCHR1 antagonist 1 exhibits potent activities against melanin-concentrating hormone-1 receptor, but less potent against human GALR1, GALR2, GALR3, MCH1, NPY1, NPY5, and rat 5HT2C receptors (Kis >50000 nM).

Chemical Properties

Molecular Weight	557.59
Formula	C₂₈H₃₃F₂N₅O₅
Cas No.	391610-37-0
Relative Density.	no data available

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Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

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