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BI-167107

Name: BI-167107
Brand: TargetMol
SKU: T14556
Rating: 4.5 (1 reviews)

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Catalog No. T14556Cas No. 1202235-68-4

BI-167107 is a high-affinity, full agonist that binds to the β2 adrenergic receptor (β2AR) with a Kd of 84 pM.

BI-167107

😃Good

Catalog No. T14556Cas No. 1202235-68-4

BI-167107 is a high-affinity, full agonist that binds to the β2 adrenergic receptor (β2AR) with a Kd of 84 pM.

Pack Size	Price	Availability
5 mg	$297	8-10 weeks
25 mg	$987	8-10 weeks
50 mg	$1,360	8-10 weeks
100 mg	$1,860	8-10 weeks
1 mL x 10 mM (in DMSO)	$318	8-10 weeks

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Product Introduction

Bioactivity

Description	BI-167107 is a high-affinity, full agonist that binds to the β2 adrenergic receptor (β2AR) with a Kd of 84 pM.
Targets&IC50	β2-adrenoceptor:（kd）84 pM
In vitro	Compared to other βAR ligands, BI-167107 exhibits nanomolar affinities and slow off-rates[1], demonstrating its high affinity and prolonged interaction with its targets.

Chemical Properties

Molecular Weight	370.44
Formula	C₂₁H₂₆N₂O₄
Cas No.	1202235-68-4
Relative Density.	1.229 g/cm3 (Predicted)

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 75 mg/mL (202.46 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.6995 mL	13.4975 mL	26.9949 mL	134.9746 mL
5 mM	0.5399 mL	2.6995 mL	5.3990 mL	26.9949 mL
10 mM	0.2699 mL	1.3497 mL	2.6995 mL	13.4975 mL
20 mM	0.1350 mL	0.6749 mL	1.3497 mL	6.7487 mL
50 mM	0.0540 mL	0.2699 mL	0.5399 mL	2.6995 mL
100 mM	0.0270 mL	0.1350 mL	0.2699 mL	1.3497 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc