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A1899 is a effective and selective TASK-1 and TASK-3 antagonist.

| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 5 mg | $395 | 35 days | |
| 25 mg | $1,560 | 35 days |
| Description | A1899 is a effective and selective TASK-1 and TASK-3 antagonist. |
| Targets&IC50 | Kv1.1:2.7 μM, TASK-2:12 μM, TASK3:0.318 pg/mL, TRAAK:>20 μM, THIK-1:2.2 μM, TASK1:0.035 μM, TASK-4:8.1 μM, TRESK:0.9 μM, TREK2:8.4 μM, TREK1:23.8 μM (pIC50) |
| Synonyms | S-20951, S20951, S 20951, A-1899, A 1899 |
| Molecular Weight | 500.54 |
| Formula | C30H26F2N2O3 |
| Cas No. | 498577-46-1 |
| Relative Density. | 1.238 g/cm3 (Predicted) |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature. |

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