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J-104129 fumarate

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Catalog No. T69576Cas No. 257603-40-0

J-104129 fumarate is a potent M3 muscarinic receptor antagonist.

J-104129 fumarate
Other Forms of J-104129 fumarate:
J 104129 fumarateT22876244277-89-2
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J-104129 fumarate

😃Good
Catalog No. T69576Cas No. 257603-40-0
J-104129 fumarate is a potent M3 muscarinic receptor antagonist.
Pack SizePriceUSA WarehouseGlobal WarehouseQuantity
10 mg$97535 days35 days
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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]
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Product Introduction

Bioactivity
Description
J-104129 fumarate is a potent M3 muscarinic receptor antagonist.
Targets&IC50
M3 mAChR:4.2 nM (Ki), M2 mAChR:490 nM (Ki)
Chemical Properties
Molecular Weight500.63
FormulaC28H40N2O6
Cas No.257603-40-0
SmilesC(=C/C(O)=O)\C(O)=O.[C@@](C(NC1CCN(CCC=C(C)C)CC1)=O)(O)(C2CCCC2)C3=CC=CC=C3
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
TargetMol | Animal experimentsFor example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH2O. So your working solution concentration is 2 mg/mL。
Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH2OTargetMol | reagent mix well and clarify
For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.
1 Enter information below:
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2 Enter the in vivo formulation:
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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc

Keywords

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