Powder: -20°C for 3 years | In solvent: -80°C for 1 year
GABAA receptor agent 6 (compound 2027) is a potent γ-GABAAR antagonist with low cellular membrane permeability (Ki = 0.56 μM) [1].
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
25 mg | 6-8 weeks | $ 1,520.00 | |
50 mg | 6-8 weeks | $ 1,980.00 | |
100 mg | 6-8 weeks | $ 2,500.00 |
Description | GABAA receptor agent 6 (compound 2027) is a potent γ-GABAAR antagonist with low cellular membrane permeability (Ki = 0.56 μM) [1]. |
In vitro | Compound 2027, a GABAA receptor agent, exhibits antagonist activity, with IC50 values of 6.68 μM for α1β2δ, 1.03 μM for α4β1δ, 0.36 μM for α4β2δ, 4.13 μM for α6β2δ, 4.96 μM for α1β2γ2, 2.96 μM for α2β2γ2, 0.29 μM for α3β2γ2, and 0.59 μM for α5β2γ2 subtypes, respectively [1]. |
Molecular Weight | 315.41 |
Formula | C18H25N3O2 |
CAS No. | 1808463-81-1 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
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GABAA receptor agent 6 1808463-81-1 inhibitor inhibit