Powder: -20°C for 3 years | In solvent: -80°C for 1 year
BChE-IN-17 (compound 6n) is a potent, selective inhibitor of butyrylcholinesterase (BChE), demonstrating inhibitory half-maximal inhibitory concentrations (IC50s) of 10.5 nM for equine BChE (eqBChE) and 32.5 nM for human BChE (hBChE). It exhibits over 1000-fold greater selectivity for BChE compared to acetylcholinesterase (AChE), while also presenting low neurotoxicity and moderate neuroprotective effects [1].
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
25 mg | 6-8 weeks | $ 1,520.00 | |
50 mg | 6-8 weeks | $ 1,980.00 | |
100 mg | 6-8 weeks | $ 2,500.00 |
Description | BChE-IN-17 (compound 6n) is a potent, selective inhibitor of butyrylcholinesterase (BChE), demonstrating inhibitory half-maximal inhibitory concentrations (IC50s) of 10.5 nM for equine BChE (eqBChE) and 32.5 nM for human BChE (hBChE). It exhibits over 1000-fold greater selectivity for BChE compared to acetylcholinesterase (AChE), while also presenting low neurotoxicity and moderate neuroprotective effects [1]. |
Targets&IC50 | AChE:686.4 μM, eqBCHE:10.5 nM, BCHE (human):32.5 nM |
Molecular Weight | 535.47 |
Formula | C23H23BrN2O4S2 |
CAS No. | 2425632-57-9 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
You can also refer to dose conversion for different animals. More
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BChE-IN-17 2425632-57-9 inhibitor inhibit