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Veldoreotide TFA

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Catalog No. T84719Cas No. 2126831-23-8
Alias PTR-3173 TFA, DG3173 TFA

Veldoreotide (DG3173) TFA, a somatostatin analogue, effectively binds to and activates somatostatin receptors (SSTR) 2, 4, and 5. This compound demonstrates a higher efficacy in inhibiting growth hormone (GH) secretion in adenomas than Octreotide, showcasing its potential as a pain modulating agent [1].

Veldoreotide TFA
Other Forms of Veldoreotide TFA:
VeldoreotideTP2420252845-37-7
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Veldoreotide TFA

😃Good
Catalog No. T84719Alias PTR-3173 TFA, DG3173 TFACas No. 2126831-23-8
Veldoreotide (DG3173) TFA, a somatostatin analogue, effectively binds to and activates somatostatin receptors (SSTR) 2, 4, and 5. This compound demonstrates a higher efficacy in inhibiting growth hormone (GH) secretion in adenomas than Octreotide, showcasing its potential as a pain modulating agent [1].
Pack SizePriceUSA WarehouseGlobal WarehouseQuantity
10 mgInquiry8-10 weeks8-10 weeks
50 mgInquiry8-10 weeks8-10 weeks
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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]
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Product Introduction

Bioactivity
Description
Veldoreotide (DG3173) TFA, a somatostatin analogue, effectively binds to and activates somatostatin receptors (SSTR) 2, 4, and 5. This compound demonstrates a higher efficacy in inhibiting growth hormone (GH) secretion in adenomas than Octreotide, showcasing its potential as a pain modulating agent [1].
Targets&IC50
sst2 receptor:37.6 nM (EC50), SST4 receptor:10.5 nM (EC50), SST3 receptor:31.3 nM (EC50)
SynonymsPTR-3173 TFA, DG3173 TFA
Chemical Properties
Molecular Weight1237.33
FormulaC62H75F3N12O12
Cas No.2126831-23-8
SmilesC(C(O)=O)(F)(F)F.C(C=1C=2C(NC1)=CC=CC2)[C@H]3C(=O)N[C@H](CC=4C=5C(NC4)=CC=CC5)C(=O)N[C@@H](CCCCN)C(=O)N[C@@]([C@@H](C)O)(C(=O)N[C@@H](CC6=CC=CC=C6)C(=O)N(CC(N)=O)CCCC(=O)NCCCC(=O)N[C@@H](CC7=CC=CC=C7)C(=O)N3)[H]
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

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Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH2OTargetMol | reagent mix well and clarify
For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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