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Droxicainide

Name: Droxicainide
Brand: TargetMol
SKU: T11099
Price: 91 USD
Availability: InStock
Rating: 5 (10 reviews)

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Catalog No. T11099Cas No. 78289-26-6

Droxicainide is an antiarrhythmic agent, [used] to treat irregular heartbeats.

Droxicainide

😃Good

Purity: 99.86%

Catalog No. T11099Cas No. 78289-26-6

Droxicainide is an antiarrhythmic agent, [used] to treat irregular heartbeats.

Pack Size	Price	USA Warehouse	Global Warehouse
1 mg	$91	In Stock	In Stock
5 mg	$179	In Stock	In Stock
10 mg	$261	In Stock	In Stock
25 mg	$407	In Stock	In Stock
50 mg	$547	In Stock	In Stock
100 mg	$708	In Stock	In Stock
200 mg	$958	-	In Stock
1 mL x 10 mM (in DMSO)	$179	In Stock	In Stock

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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]

This molecule is a custom-made product. TargetMol has an excellent synthesis team with the experience and capability to provide you with cost-effective products. If you have any questions, please feel free to contact us. We are committed to serving you wholeheartedly.

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Batch Information

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Purity:99.86%

Appearance:Solid

Color:White

Resource Download

COA HNMR LCMS

Product Introduction

Bioactivity

Description	Droxicainide is an antiarrhythmic agent, [used] to treat irregular heartbeats.
In vivo	In coronary artery occlusion studies, Droxicainide reduced the progression of hypoperfusion to necrosis and reduced the infarct size in dogs[1].Droxicainide reduces ansa node, atrioventricular excitability and contractility, and increases intractable studies on spontaneous beating atrium, electrical stimulation atrium and isolated papillary muscles in rats[2].

Chemical Properties

Molecular Weight	276.37
Formula	C₁₆H₂₄N₂O₂
Cas No.	78289-26-6
Smiles	C(NC1=C(C)C=CC=C1C)(=O)C2N(CCO)CCCC2
Relative Density.	1.133g/cm3

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 50 mg/mL (180.92 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	3.6183 mL	18.0917 mL	36.1834 mL	180.9169 mL
5 mM	0.7237 mL	3.6183 mL	7.2367 mL	36.1834 mL
10 mM	0.3618 mL	1.8092 mL	3.6183 mL	18.0917 mL
20 mM	0.1809 mL	0.9046 mL	1.8092 mL	9.0458 mL
50 mM	0.0724 mL	0.3618 mL	0.7237 mL	3.6183 mL
100 mM	0.0362 mL	0.1809 mL	0.3618 mL	1.8092 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the stock solution preparation method and in vivo formula preparation method:

For example, if the intended dosage is 10 mg/kg for animals weighing 20 g , with a dosing volume of 100 μL per animal, TargetMol | Animal experiments

and a total of 10 animals are to be administered, using a formulation of TargetMol | reagent

10% DMSO+ 40% PEG300+ 5% Tween 80+ 45% Saline/PBS/ddH₂O , the resulting working solution concentration would be 2 mg/mL.

Stock Solution Preparation:

Dissolve 2 mg of the compound in 100 μL DMSO TargetMol | reagent to obtain a stock solution at a concentration of 20 mg/mL . If the required concentration exceeds the compound's known solubility, please contact us for technical support before proceeding.

Preparation of the In Vivo Formulation:

1) Add 100 μL of the DMSO TargetMol | reagent stock solution to 400 μL PEG300 and mix thoroughly until the solution becomes clear.

2) Add 50 μL Tween 80 and mix well until fully clarified.

3) Add 450 μL Saline,PBS or ddH₂O TargetMol | reagent and mix thoroughly until a homogeneous solution is obtained.

This example is provided solely to demonstrate the use of the In Vivo Formulation Calculator and does not constitute a recommended formulation for any specific compound. Please select an appropriate dissolution and formulation strategy based on your experimental model and route of administration.

All co-solvents required for this protocol, includingDMSO, PEG300/PEG400, Tween 80, SBE-β-CD, and Corn oil, are available for purchase on the TargetMol website.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc