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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T15721 | Latrunculin A | LAT-A | Others |
Latrunculin A is a toxin isolated from the red sea sponge Latrunculia magnifica. Latrunculin A binds to actin monomers and it also inhibits polymerization of actin (Kds: 0.1, 0.4, 4.7 μM, and 0.19 μM for ATP-actin, ADP-P... | |||
T20636 | Latrunculin B | LAT-B,LATB,NSC 339663,NSC339663,NSC-339663,LAT B,INS115644 | Antifungal |
Latrunculin B, an alkaloid from the Red Sea sponge, is an actin polymerization inhibitor with antifungal and antiprotozoal activity.Latrunculin B modulates the electrophysiological characteristics of the pulmonary veins ... | |||
T15411 | GPNA hydrochloride | Apoptosis , Others | |
GPNA hydrochloride is specific glutamine (Gln) transporter ASCT2(SLC1A5) inhibitor. GPNA reversibly induces apoptosis in A549 cells. GPNA hydrochloride is a well-known substrate of the enzyme γ-glutamyltransferase (GGT).... | |||
T11820 | LAT1-IN-1 | BCH | Apoptosis , Others |
LAT1-IN-1 (BCH) (BCH) significantly inhibit cellular uptake of amino acids and mTOR phosphorylation, which induces the suppression of cancer growth and apoptosis. is a selective and competitive inhibitor of large neutral... | |||
T20351 | Ethyl phenylglyoxylate | AI3-10033,AI3 10033,AI310033 | Lipid |
Ethyl phenylglyoxylate (AI3 10033) is a simultaneous inhibitor and substrate of chicken liver carboxylesterase. | |||
T4875 | Palatinose hydrate | 6-O-α-D-Glucopyranosyl-D-fructose, Isoma | Others , Endogenous Metabolite |
Palatinose hydrate (6-O-α-D-Glucopyranosyl-D-fructose, Isoma) is a disaccharide having an α(1→6) linkage between D-glucose and D-fructose and is similar to sucrose in its physicochemical properties. It is produced from s... | |||
T21983L | PKI 14-22 amide, myristoylated Acetate | PKI 14-22 amide, myristoylated Acetate(201422-03-9 Free base) | PKA |
PKI 14-22 amide, myristoylated Acetate inhibit cAMP-dependent protein kinase (PKA) and blocks hyperalgesia produced by spinal administration of 8-bromo-cAMP. | |||
T7598 | Calcium N5-methyltetrahydrofolate | NSC173328 | Others , Antifolate |
Calcium N5-methyltetrahydrofolate (NSC-173328) is the calcium salt of levomefolic acid, which has been proposed for treatment of cardiovascular disease and advanced cancers such as breast and colorectal cancers | |||
TN6745 | PALATINOSE | TNP-470,Isomaltulose | Others |
PALATINOSE (TNP-470) is a natural occurring disaccharide composed of alpha-1,6-linked glucose and fructose。 PALATINOSE has a beneficial effect on liver metabolic functions and might therefore be a good substitute for suc... | |||
TN6710 | Methyl acetylsalicylate | ACETYLSALICYLIC ACID METHYL ESTER | Others |
Methyl acetylsalicylate (ACETYLSALICYLIC ACID METHYL ESTER) is a natural product isolated from Pisum sativum. Inhibition of collagen-induced human platelet rich plasma aggregation | |||
T77478 | Milatuzumab | hLL1,MEDI-115 | Others |
Milatuzumab (MEDI-115) is a humanized monoclonal antibody against CD74. Milatuzumab promotes the production of free radical oxygen and the loss of mitochondrial membrane potential, reduces CD20/CD74 aggregates and cell a... | |||
T14552 | Dactolisib Tosylate | BEZ235 Tosylate,NVP-BEZ 235 Tosylate | PI3K , mTOR |
Dactolisib Tosylate (BEZ235 Tosylate) is a dual kinase inhibitor that targets PI3K and mTOR. dactolisib Tosylate exhibits IC50 values of 4, 75, 7, and 5 nM for PI3Kα, β, γ, and δ, respectively. dactolisib Tosylate inhibi... | |||
T10759 | CEP-28122 mesylate salt (1022958-60-6 free base) | CEP-28122 mesylate salt | ALK |
CEP-28122 mesylate salt (1022958-60-6 free base) is a highly selective orally active ALK inhibitor (IC50: 1.9 nM in an enzyme-based TRF assay). | |||
T7175 | Alflutinib mesylate | AST2818 mesylate | EGFR |
Alflutinib mesylate (AST2818 mesylate) ,is an irreversible tyrosine kinase inhibitor that selectively inhibits EGFR mutations, especially T790M. | |||
T8216 | T-1101 tosylate | TAI-95 tosylate | Apoptosis , Microtubule Associated |
T-1101 tosylate (TAI-95 tosylate) is an inhibitor of Hec1/Nek2, with antitumor activity. | |||
TN2349 | Taurodeoxycholate sodium salt | Sodium taurodeoxylate | Endogenous Metabolite |
Taurodeoxycholate sodium salt (Sodium taurodeoxylate) is a bile salt-related anionic detergent used for isolation of membrane proteins including inner mitochondrial membrane proteins. and it inhibits various inflammatory... | |||
TP1658L | Type A Allatostatin I acetate | Type A Allatostatin I acetate(123209-95-0 free base) | Others |
Type A Allatostatin I acetate is a tridecapeptide. Allatostatins are pleiotropic neuropeptides for inhibition of juvenile hormone synthesis in insects. | |||
T72528 | NSC243928 mesylate | HuR | |
NSC243928 mesylate binds to human lymphocyte antigen 6 (LY6), a cell growth inhibitor with anticancer activity, and induces cell death in triple-negative breast cancer cells in a LY6K-dependent manner. | |||
TP1907L1 | Dynamin inhibitory peptide, myristoylated acetate | Dynamin inhibitory peptide, myristoylated acetate(251634-22-7 free base) | Dynamin |
Dynamin inhibitory peptide, myristoylated acetate is a DynaMin inhibitor to interfere with the binding of amphiphysin with dynamin. DynaMin inhibitory peptide, myristoylated TFA is a membrane-permeant form of the peptide... | |||
T61483 | GLP-1R modulator C5 | Glucagon Receptor | |
GLP-1R modulator C5 is a small molecule GLP-1R orthosteric modulator that enhances GLP-1 binding to GLP-1R via transmembrane sites and can be used in the study of type II diabetes. |