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Search Results for "kinase"

Targets

Libraries

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Compounds

Cat No. Product Name
T6335 Tie2 kinase inhibitor 1 Tie2 kinase inhibitor Tie-2
Tie2 kinase inhibitor 1 是Tie2激酶选择性抑制剂9IC50:250 nM),具有抗癌作用。
T5524 Aurora kinase inhibitor-3 Aurora Kinase Inhibitor III Aurora Kinase
Aurora kinase inhibitor-3 是一种有效的,选择性 Aurora A 激酶抑制剂,IC50为 42 nM。
T4191 Multi-kinase inhibitor 1 Multi-kinase inhibitor I Others , PDGFR , Bcr-Abl , c-Kit
Multi-kinase inhibitor 1 是多激酶抑制剂。它有用于导致与酪氨酸激酶活性异常或失控有关的疾病或失调的潜力,特别是与c-Kit,PDGF-R,Bcr-abl 活性相关的疾病。
T9040 Aurora kinase inhibitor-2 Aurora Kinase Inhibitor II,IUN-70219 Aurora Kinase
Aurora kinase inhibitor-2 是一种可渗透细胞的苯胺喹唑啉,可抑制极光激酶的活性,对Aurora A 和Aurora B 的IC50分别为 390 nM 和 240 nM。
T11184 EML4-ALK kinase inhibitor 1 EML4 ALK kinase inhibitor 1 ALK
EML4-ALK kinase inhibitor 1 是有效的、具有口服活性的类棘皮细胞微管相关蛋白4-间变性淋巴瘤激酶 (EML4-ALK) 的抑制剂,其 IC50 值为 1 nM。
TP1053L Protein Kinase C 19-31 acetate Protein Kinase C 19-31 acetate(121545-65-1 free base),PKC (19-31) acetate PKC
Protein Kinase C 19-31 acetate(121545-65-1 free base) 是一种蛋白激酶 C (PKC) 的肽抑制剂,源自 PKCa 的假底物调节结构域(残基 19-31),在 25 位用丝氨酸取代野生型丙...
T60108 PDGFR Tyrosine Kinase Inhibitor III PDGF Receptor Tyrosine Kinase Inhibitor III PDGFR
PDGFR Tyrosine Kinase Inhibitor III (PDGF Receptor Tyrosine Kinase Inhibitor III)是一种多激酶抑制剂,可抑制 PDGFR、EGFR、FGFR、PKA 和 PKC...
T4692 Protein kinase inhibitors 1 hydrochlorid Protein kinase inhibitors 1 hydrochlorid (1365986-44-2(free base)) Others
Protein kinase inhibitors 1 hydrochlorid 是一种新型 HIPK2 抑制剂,IC50 为 74 nM,Kd 为 9.5 nM。
TP1271L Calmodulin-Dependent Protein Kinase II 290-309 acetate Calmodulin-Dependent Protein Kinase II 290-309 acetate (115044-69-4 Free base) CaMK
Calmodulin-Dependent Protein Kinase II 290-309 acetate 是 Ca2+/calmodulin-dependent protein kinase II 的有效拮抗剂(IC50 = 52 nM...
TP1051L Protein Kinase C Peptide Substrate acetate Protein Kinase C Peptide Substrate acetate(120253-69-2 free base) Others
Protein Kinase C Peptide Substrate acetate(120253-69-2 free base) 以依赖于第二信使和特定衔接蛋白的方式靶向特定细胞间隔物,以响应激活 g 蛋白偶联受体、酪氨酸激酶受体或酪氨酸...
T8864 Thymidylate Kinase Inhibitor, YMU1 Others
YMU1 是一种选择性抑制剂,特异性作用于人胸苷酸激酶 (IC50: 610 nM) 。
T16987 TAO Kinase inhibitor 1 Others , MAPK
TAO Kinase inhibitor 1 是一种ATP 竞争性的thousand-and-one amino acid kinases (TAOK)选择性抑制剂,对于 TAOK1 和 TAOK2 的IC50s 分别为 11 nM 和 1...
T12721 Rho-Kinase-IN-1 ROCK
Rho-Kinase-IN-1 是一种 ROCK 抑制剂,对 ROCK1 和 ROCK2 的 Kis 分别为 30.5 nM 和 3.9 nM。 Rho-Kinase-IN-1 可用于细胞过度增殖、重塑、水肿和炎症疾病的研究。
T5466 Tyrosine kinase-IN-1 PDGFR , FGFR , VEGFR , FLT
Tyrosine kinase-IN-1是一种多靶点酪氨酸激酶抑制剂,能够抑制KDR (IC50:4 nM),Flt-1 (IC50:20 nM),FGFR1 (IC50:4 nM) 和 PDGFRα (IC50:2 nM)。
T4026 SU5408 VEGFR2 Kinase Inhibitor I VEGFR
VEGFR2 Kinase Inhibitor I 是一种可渗透细胞的VEGFR2激酶抑制剂,其IC50=70 nM。
T10687 Casein Kinase II Inhibitor IV Casein Kinase
Casein Kinase II Inhibitor IV 是一种小分子诱导剂,可诱导表皮角质形成细胞分化。
T9564 IRE1α kinase-IN-1 IRE1
IRE1α kinase-IN-1 是IRE1α 的选择性抑制剂(IC50为 77 nM),对 IRE1α 的选择性高于 IRE1β 亚型 100 倍。它抑制内质网诱导的 IRE1α 寡聚和自磷酸化,并抑制 IRE1α RNase 活性 (...
T12728 RIP2 Kinase Inhibitor 3 RIP kinase , Others
RIP2 Kinase Inhibitor 3 是一种有效的选择性 受体相互作用蛋白2 激酶抑制剂,IC50 为 1 nM。
T9631 IRAK-4 protein kinase inhibitor 2 IRAK
IRAK-4 protein kinase inhibitor 2 是有效的白介素 1 受体相关激酶 4 抑制剂,IC50为 4 μM。它在与炎症和免疫相关的疾病领域有研究价值。
T77500 Casein kinase 1δ-IN-6 Casein Kinase
Casein kinase 1δ-IN-6 是一种有效且具有选择性的蛋白激酶 CK-1δ 抑制剂,其 IC50 为 23 nM。Casein kinase 1δ-IN-6 在体外和体内实验中均显示出神经保护和抗炎活性。Casein kina...
Tie2 kinase inhibitor 1
T6335
synonym: Tie2 kinase inhibitor
Target:
Aurora kinase inhibitor-3
T5524
synonym: Aurora Kinase Inhibitor III
Target:
Multi-kinase inhibitor 1
T4191
synonym: Multi-kinase inhibitor I
Target:
Aurora kinase inhibitor-2
T9040
synonym: Aurora Kinase Inhibitor II,IUN-70219
Target:
EML4-ALK kinase inhibitor 1
T11184
synonym: EML4 ALK kinase inhibitor 1
Target:
Protein Kinase C 19-31 acetate
TP1053L
synonym: Protein Kinase C 19-31 acetate(121545-65-1 free base),PKC (19-31) acetate
Target:
PDGFR Tyrosine Kinase Inhibitor III
T60108
synonym: PDGF Receptor Tyrosine Kinase Inhibitor III
Target:
Protein kinase inhibitors 1 hydrochlorid
T4692
synonym: Protein kinase inhibitors 1 hydrochlorid (1365986-44-2(free base))
Target:
Calmodulin-Dependent Protein Kinase II 290-309 acetate
TP1271L
synonym: Calmodulin-Dependent Protein Kinase II 290-309 acetate (115044-69-4 Free base)
Target:
Protein Kinase C Peptide Substrate acetate
TP1051L
synonym: Protein Kinase C Peptide Substrate acetate(120253-69-2 free base)
Target:
Thymidylate Kinase Inhibitor, YMU1
T8864
synonym:
Target:
TAO Kinase inhibitor 1
T16987
synonym:
Target:
Rho-Kinase-IN-1
T12721
synonym:
Target:
Tyrosine kinase-IN-1
T5466
synonym:
Target:
SU5408
T4026
synonym: VEGFR2 Kinase Inhibitor I
Target:
Casein Kinase II Inhibitor IV
T10687
synonym:
Target:
IRE1α kinase-IN-1
T9564
synonym:
Target:
RIP2 Kinase Inhibitor 3
T12728
synonym:
Target:
IRAK-4 protein kinase inhibitor 2
T9631
synonym:
Target:
Casein kinase 1δ-IN-6
T77500
synonym:
Target:
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