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L 888607 Racemate

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Catalog No. T15829Cas No. 1030017-51-6

L 888607 Racemate is a selective antagonist of the prostaglandin D2 receptor subtype 1 (DP1) with Ki values of 132 nM and 17 nM for DP1 and the thromboxane A2 receptor (TP), respectively.

L 888607 Racemate
Other Forms of L 888607 Racemate:
L 888607T15828860033-06-3
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L 888607 Racemate

😃Good
Catalog No. T15829Cas No. 1030017-51-6
L 888607 Racemate is a selective antagonist of the prostaglandin D2 receptor subtype 1 (DP1) with Ki values of 132 nM and 17 nM for DP1 and the thromboxane A2 receptor (TP), respectively.
Pack SizePriceUSA WarehouseGlobal WarehouseQuantity
25 mg$1,0806-8 weeks6-8 weeks
50 mg$1,4106-8 weeks6-8 weeks
100 mg$1,9906-8 weeks6-8 weeks
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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]
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Product Introduction

Bioactivity
Description
L 888607 Racemate is a selective antagonist of the prostaglandin D2 receptor subtype 1 (DP1) with Ki values of 132 nM and 17 nM for DP1 and the thromboxane A2 receptor (TP), respectively.
Targets&IC50
DP/DP1:132 nM (ki), TP Receptor:17 nM (ki)
In vitro
L 888607 Racemate is actually 8-fold more effective on the TP receptor (Ki = 17 nM). L 888607 Racemate maintains a modest binding affinity for the DP1 receptor (Ki = 132 nM) .
Chemical Properties
Molecular Weight375.84
FormulaC19H15ClFNO2S
Cas No.1030017-51-6
Relative Density.1.46 g/cm3 (Predicted)
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
Solubility Information
DMSO: 6 mg/mL (15.96 mM), Sonication is recommended.
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM2.6607 mL13.3035 mL26.6071 mL133.0353 mL
5 mM0.5321 mL2.6607 mL5.3214 mL26.6071 mL
10 mM0.2661 mL1.3304 mL2.6607 mL13.3035 mL

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Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
TargetMol | Animal experimentsFor example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH2O. So your working solution concentration is 2 mg/mL。
Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH2OTargetMol | reagent mix well and clarify
For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.
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Keywords

TPL 888607 RacemateDP/DP1AuroraKinaseAurora Kinase
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