rn — TargetMol Chemicals

Cat No.	Product Name	Synonyms	Targets
T16763	RN-1747		TRP/TRPV Channel
	RN-1747 is a selective transient receptor potential cation channel subfamily V member 4 agonists (EC50: 0.77 μM, 4.0 μM, and 4.1 μM for hTRPV4, mTRPV4, and rTRPV4 respectively). RN-1747 also antagonizes TRPM8 (IC50: 4 μM...		TRP/TRPV Channel
T16764	RN-18		HIV Protease
	RN-18 is an inhibitor of HIV-1 viral infectivity factor (IC50: 6 μM in nonpermissive H9 cells).		HIV Protease
T77723	RN-1665		TRP/TRPV Channel
	RN-1665 is a potent and selective TRPV4 receptor antagonist.		TRP/TRPV Channel
T21652	RN-1 dihydrochloride		Histone Demethylase , MAO
	RN-1 dihydrochloride is an effective and selective irreversible inhibitor of lysine-specific demethylase 1 (LSD1, IC50 = 70 nM).		Histone Demethylase , MAO
T7572	RN-1734		TRP/TRPV Channel
	RN-1734 is selective TRPV4 channel antagonist(IC50 of 2.3 μM,5.9 μM,3.2 μM for hTRPV4, mTRPV4 and rTRPV4,respectively)		TRP/TRPV Channel
T28548	RN9893	RN9893 Hydrochloride,RN 9893 HCl,RN-9893 HCl,RN-9893,RN-9893 Hydrochloride,RN 9893 Hydrochloride	TRP/TRPV Channel
	RN9893 is a selective and potent TRPV4 receptor antagonist with IC50 values of 320, 420 and 660 nM for TRPV4 receptors in mouse, human and rat, respectively.		TRP/TRPV Channel
T12711	Retro-2 cycl	RN 1-001	Virus Protease
	Retro-2 cycl is a dihydroquinazolinone (DHQZ) retrograde trafficking inhibitor. Retro-2 cycl (RN 1-001) inhibits JCPyV and HPV16 pseudovirus(IC50s of 54 μM and 160 μM, respectively),with antiviral agent.		Virus Protease
T37321	RN-9893 (hydrochloride)
	RN-9893 is an antagonist of transient receptor potential vanilloid 4 (TRPV4; IC50s = 0.42 and 0.66 μM, respectively, for the human and rat receptors).1 It is selective for TRPV4 over TRPV1, TRPV3, and TRPM8 (IC50s = 10, ...
T1844	KPT330,(E)-	(E)-RN,KPT-330,KPT330,KPT 330	Others , CRM1
	(E)-RN (KPT 330) is a CRM1-selective inhibitor of nuclear export. It inhibits protein trafficking from the nucleus and induces cell cycle arrest and apoptosis in mesothelioma cells.		Others , CRM1
T34337	RN983	RN 983,RN-983
	RN983 is a potent and selective BTK inhibitor.
T1976	RN486		BTK
	RN486 is an effective and specific BTK inhibitor (IC50: 4 nM).		BTK
T76739	Bococizumab	RN316,PF-04950615	Others
	Bococizumab(PF-04950615) is a humanized mAb against PCSK9 and an inhibitor of the synthesis of PCSK9 in the liver that reduces the amount of low-density lipoprotein cholesterol (LDL-C) in the blood.Bococizumab is used to...		Others
T78282	Tanezumab	RN-624,PF 4383119
	Tanezumab (RN-624) is a high-affinity, specific humanized anti-NGF monoclonal antibody (mAb) that inhibits nerve growth factor (NGF) from binding to its p75 and TrkA receptors in the peripheral nervous system. It is util...
T32371	Kebuzone	Chepirol,RN 0308507,Chebutan,Chetazolidin,Chetil
	Kebuzone is a non-steroidal anti-inflammatory drug, known to have analgesic, antipyretic, and platelet inhibitory activities.
T28547	RN941
	RN941 is a highly potent Bruton's tyrosine kinase (BTK) inhibitor.
TN4919	Rosthornin A		Others
	Rosthornin A is a kind of natural product derived from the herbs of Rabdosia rosthornii.		Others
T8028	Farnesyl acetate	Farnesyl Acetate (mixture of isomers)	Others
	Farnesyl acetate (Farnesyl Acetate (mixture of isomers)) is a flavouring compound identified in foods such as blueberries.		Others
TP1928L1	[Orn5]-URP acetate	[Orn5]-URP acetate(782485-03-4 free base)	GPR
	[Orn5]-URP acetate is an effective and selective Urotensin-II receptor (UT) antagonist (pEC50 = 7.24). [Orn5]-URP exhibits no agonist activity.		GPR
T2785	4-Methylherniarin	7-Methoxy-4-methylcoumarin	Others , Antibacterial
	4-Methylherniarin (7-Methoxy-4-methylcoumarin) is a coumarin derivative and fluorescent label, it displays good activity against B. subtilis.		Others , Antibacterial
T6475	(±)-Carnitine chloride	Monocamin,DL-Carnitine HCl,Bicarnesine,DL-Carnitine chloride	Reactive Oxygen Species
	(±)-Carnitine chloride (Monocamin) is a quaternary ammonium compound biosynthesized from the amino acids lysine and methionine.		Reactive Oxygen Species