keep away from moisture
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
[Orn8]-Urotensin II acetate is a Urotensin receptor ligand and a partial agonist at Urotensin receptors.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 195.00 | |
5 mg | In stock | $ 437.00 | |
10 mg | In stock | $ 646.00 | |
25 mg | In stock | $ 987.00 | |
50 mg | In stock | $ 1,380.00 | |
100 mg | In stock | $ 1,860.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 928.00 |
Description | [Orn8]-Urotensin II acetate is a Urotensin receptor ligand and a partial agonist at Urotensin receptors. |
Targets&IC50 | UT receptor/GPR14:8 (pEC50) |
In vivo | [Orn8]-Urotensin II acetate behaves as a full agonist (pEC50 approximately equal 8) at both human and rat UT receptors in the FlipR calcium assay eliciting similar maximal effects as the natural ligand U-II. On the contrary, in the rat aorta bioassay, [Orn8]-Urotensin II acetate behaves as a competitive and selective antagonist (pA2 = 6.56) showing however a small but consistent residual agonist activity[2]. |
Molecular Weight | 1434.59 |
Formula | C65H87N13O20S2 |
keep away from moisture
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 14.35 mg/mL (10 mM)
You can also refer to dose conversion for different animals. More
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[Orn8]-Urotensin II acetate Endocrinology/Hormones GPCR/G Protein GPR [Orn8]Urotensin II acetate [Orn8]-Urotensin II Acetate [Orn8] Urotensin II acetate [Orn-8]-Urotensin II acetate(479065-85-5 Free base) inhibitor inhibit