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Search Results for " esi "

Targets

194

Compounds

122

Natural Products

11

Recombinant Proteins

3

Libraries

Cat No. Product Name Synonyms Targets
T11234 ESI-08 cAMP
ESI-08 is an effective antagonist of EPAC2 with an IC50 of 8.4 μM. ESI-08 selectively blocks cAMP-induced EPAC activation but not cAMP-mediated PKA activation.
T2244 ESI-09 cAMP , Virus Protease
ESI-09 is a new-typel noncyclic nucleotide EPAC antagonist.The IC50 values of ESI-09 for EPAC1 and EPAC2 is 3.2 and 1.4 μM, respectively.
T15247 ESI-05 NSC 116966 cAMP
ESI-05 (NSC-116966) is a specific EPAC2 (exchange protein directly activated by cAMP 2) antagonist (IC50: 0.4 μM). ESI-05 inhibits cAMP-mediated activation of EPAC2, as well as EAPC2, mediated Rap1 activation.
T19389 L-Ascorbic acid 2-phosphate magnesium 2-Phospho-L-ascorbic acid magnesium Phosphatase , Phosphorylase
L-Ascorbic acid 2-phosphate magnesium (2-Phospho-L-ascorbic acid magnesium) acts as an antioxidant and a stimulator of hepatocyte growth factor (HGF) production.It is a long-acting vitamin C derivative that can stimulate...
T76831 Tesidolumab LFG316 Complement System
Tesidolumab (LFG316) is a fully human IgG1/λ anti-C5 monoclonal antibody. Tesidolumab (LFG316) has an inhibitory effect on crovalimab and C5, blocking the cutting of C5 and preventing the subsequent formation of membrane...
T36395 Trotabresib CC-90010 Epigenetic Reader Domain
Trotabresib (CC-90010) is an orally active inhibitor of BET and can be used in studies about advanced solid tumors.
T12834 Saroglitazar Magnesium Others
Saroglitazar Magnesium is a novel peroxissome proliferator-activated receptor (PPAR) agonist with significant activation activity against PPARα (EC50 0.65pM) and moderate activation against PPARγ (EC50 3 nM).
T15337 Forodesine BCX-1777,Immucillin-H Others
Forodesine is a potent human lymphocyte proliferation inhibitor. Forodesine is an orally active inhibitor of purine nucleoside phosphorylase (IC50s: 0.48 to 1.57 nM for human, mouse, rat, monkey, and dog PNP). It could i...
T10491 Galidesivir BCX4430,Immucillin-A Others
Galidesivir (BCX4430) is a broad-spectrum antiviral compound, an adenosine analog that inhibits viral RNA-dependent RNA polymerase (RdRp) activity.Galidesivir inhibits a wide range of RNA viral pathogens in vitro, and re...
T26778L Besipirdine hydrochloride HP 749 hydrochloride,Besipirdine hydrochloride(119257-34-0 Free base) Adrenergic Receptor
Besipirdine hydrochloride is a non-receptor-dependent cholinomimetic compound with alpha-adrenergic and cardiovascular activities.Besipirdine hydrochloride inhibits voltage-dependent sodium-potassium channels and inhibit...
T12399 Peldesine BCX 34 Nucleoside Antimetabolite/Analog , HIV Protease
Peldesine (BCX 34) is an effective, competitive, reversible, and orally active inhibitor of purine nucleoside phosphorylase. Peldesine inhibits T-cell proliferation with an IC50 of 800 nM. Peldesine can be used in resear...
T6032 Birabresib OTX-015,OTX015 (MK 8628/Birabresib),MK-8628 Epigenetic Reader Domain
Birabresib (MK-8628) is a synthetic, small molecule inhibitor of the BET (Bromodomain and Extra-Terminal) family of bromodomain-containing proteins 2, 3 and 4 with potential antineoplastic activity.
T39994 Sovilnesib AMG650 Microtubule Associated
Sovilnesib is a kinesin-like protein KIF18A inhibitor. Sovilnesib can be used for the cancer research.
T3258 Ponesimod ACT-128800 S1P Receptor , LPL Receptor
Ponesimod (ACT-128800) is an orally available sphingosine-1-phosphate receptor 1 (S1PR1, S1P1) agonist with potential immunomodulating activity.
T6405 Bepotastine Besilate Talion,TAU 284,Bepreve,Bepotastine Beslilate Histamine Receptor
Bepotastine Besilate (TAU 284) is a non-sedating and selective H1 receptor antagonist (pIC50: 5.7).
T4512 Magnesium glycinate magnesium 2-aminoacetate,Magnesium diglycinate Others
Magnesium glycinate (magnesium 2-aminoacetate) is a supplement that boost magnesium levels in people with a deficiency of the mineral. Magnesium is a vital nutrient for regulating many body processes, including muscle an...
T26778 Besipirdine HP 749 free base,P-867493,P867493,HP 749,HP749,P 867493 Sodium Channel , Adrenergic Receptor
Besipirdine (HP 749 free base) is a non-receptor-dependent cholinomimetic compound with alpha-adrenergic and cardiovascular activities.Besipirdine inhibits voltage-dependent sodium-potassium channels and inhibits biogeni...
T8391 Cesium chloride CsCl Potassium Channel
Cesium chloride (CsCl) is considered to be the most toxic of the alkali chlorides, inhibiting fungal growth.
T6964 Resiquimod R848,S28463 HCV Protease , TLR
Resiquimod (R848) is an imidazoquinoline amine and Toll-like receptor (TLR) agonist with potential immune response modifying activity. Resiquimod exerts its effect through the TLR signaling pathway by binding to and acti...
T5832 Besifovir HBV
Besifovir, a parent drug converted by LB80380, further metabolizes to its active form, LB80317. LB80380 is potent antiviral agent against hepatitis B virus (HBV).
T67822L Ulodesine BCX4208 Endogenous Metabolite
Ulodesine (BCX4208) is a purine nucleoside phosphorylase (PNP) inhibitor that inhibits PNP with an IC50 value of 2.293 nM/L. Ulodesine may be used to study hyperuricaemia.
T3712 Mivebresib ABBV-075 Apoptosis , Epigenetic Reader Domain
Mivebresib (ABBV-075), also known as ABBV-075, is a potent BET inhibitor (bromodomain (BRD)-containing protein) with potential antineoplastic activity. Upon administration, the bromodomain inhibitor ABBV-075 binds to the...
TP1153L Fibronectin Adhesion-promoting Peptide acetate Fibronectin Adhesion-promoting Peptide acetate(125720-21-0 free base),Heparin Binding Peptide acetate Others
Fibronectin Adhesion-promoting Peptide acetate (Heparin Binding Peptide acetate) is one of the heparin-binding amino acid sequences found in the carboxy-terminal heparin-binding domain of fibronectin.
T67817 Besifovir PM LB80331 PM HBV
Besifovir PM (LB80331 PM) is an analogue of Besifovir, a novel orally available acyclic nucleotide phosphonate for the treatment of chronic hepatitis B infection.
T7882 Indomethacin farnesil Infree Others , COX , Autophagy
Indomethacin farnesil (Infree) is a prodrug of indomethacin. It acts as a nonsteroidal anti-inflammatory drug (NSAID) and disease-modifying anti-rheumatic drug (DMARD).
T8772 Sumaresinolic Acid Others
Sumaresinolic Acid is a natural lignan found in a variety of plants such as flaxseed, sesame and wheat bran and is a secondary metabolite of plants. It has been widely studied for its potential health benefits, including...
TP2219L Alytesin acetate Others
Alytesin acetate is an amphibian bombesin-like peptide.
TP1916L1 [D-Phe12,Leu14]-Bombesin acetate [D-Phe12,Leu14]-Bombesin acetate(108437-88-3 Free base) Bombesin Receptor
[D-Phe12,Leu14]-Bombesin acetate inhibits bombesin-stimulated secretion.
T6875 Lesinurad RDEA594 OAT
Lesinurad (RDEA594) is a selective inhibitor of uric acid reabsorption which is used in combination with other agents in the therapy of gout. Lesinurad has had a limited clinical use but has not been associated with seru...
T7780 Blarcamesine AE-37,AVex-73 AChR
Blarcamesine (AVex-73) is a muscarinic M1 agonist potentially for the treatment of Alzheimer's disease.
T4507 Chlorphenesin Adermykon,Chlorophenesin,Gecophen Antibacterial , Antifungal , Histamine Receptor
Chlorphenesin (Chlorophenesin) is an antigen-associated immunosuppressant that inhibits IgE-mediated histamine release. It is also used as an antimycotic agent.
T7766 Remdesivir GS-5734 SARS-CoV , DNA/RNA Synthesis
Remdesivir (GS-5734) is a nucleoside analog, a broad-spectrum antiviral compound that exerts its activity by inhibiting the RNA-dependent RNA polymerase of viruses. Remdesivir is active against Ebola, SARS, and MERS viru...
T8386 Esomeprazole Magnesium trihydrate (S)-Omeprazole magnesium trihydrate Proton pump
Esomeprazole Magnesium trihydrate ((S)-Omeprazole magnesium trihydrate) is a proton pump inhibitor indicated for the short-term treatment of gastroesophageal reflux disease in patients with a history of erosive esophagit...
T40864 Magnesium sulfate Others
Magnesium sulfate is the preferred anticonvulsant for preventing and controlling eclamptic seizures. Additionally, it is extensively utilized as a tocolytic agent.
TQ0318 Filanesib ARRY-520,ARRY 520 KSP
Filanesib (ARRY 520) is a selective inhibitor of kinesin spindle protein (KSP, IC50 = 6 nM) with potent anti-proliferative activity.
T9379 L-Threonic acid magnesium salt Others
L-Threonic acid magnesium salt (L-TAMS) increases synapse density and memory ability in both aged rats and late stage Alzheimer’s disease (AD) model mice.
T9978 Glutathione synthesis-IN-1 Others
Glutathione synthesis-IN-1 (DC-1) is a inhibitor of glutathione synthesis[1].
TP1281L1 Bombesin acetate(31362-50-2 free base) Bombesin Receptor
Bombesin acetate is a 14-amino acid peptide originally isolated from the skin of the European fire-bellied toad (Bombina bombina). It has two known homologs in mammals called neuromedin B and gastrin-releasing peptide.
T5939 Calcium dobesilate Apoptosis , Others
Calcium dobesilate(CaD) has angioprotective properties and protects endothelial cells partly by ameliorating HG induced inflammation.
T1906 Molibresib GSK 525762A,GSK525762,I-BET 762 Epigenetic Reader Domain
Molibresib (GSK525762) is an inhibitor of BET proteins (IC50: about 35 nM).
T8495 Alobresib Vorolanib,GS-5829 Epigenetic Reader Domain
Alobresib (Vorolanib) is an inhibitor of BET bromodomain,is an antineoplastic drug candidate.
T3272 Metamizole magnesium Metamizolemagnesiumsalt Antibiotic
Metamizole magnesium (Metamizolemagnesiumsalt) is a pain reliever, which can antispasmodic.
TP2239L [D-Phe12]-Bombesin acetate [D-Phe12]-Bombesin acetate(108437-87-2 free base) Bombesin Receptor
[D-Phe12]-Bombesin acetate inhibits bombesin-stimulated secretion.
T2686 Esomeprazole Magnesium (S)-Omeprazole magnesium,NEXIUM,(-)-Omeprazole magnesium ATPase , Proton pump
Esomeprazole Magnesium (NEXIUM) is the S-isomer of omeprazole, can reduce gastric acid secretion with selective and irreversible proton pump inhibitor activity.Esomeprazole magnesium acts as an exosome inhibitor by block...
T4111 Blarcamesine hydrochloride Anavex 2-73,AVex-73 hydrochloride,AE-37 hydrochloride Sigma receptor
Blarcamesine hydrochloride (AVex-73 hydrochloride) is a Sigma-1 Receptor agonist (IC50: 860 nM).
T3597 Cutamesine dihydrochloride AGY94806 dihydrochloride,SA4503 (dihydrochloride),SA4503 dihydrochloride Sigma receptor
Cutamesine dihydrochloride (SA4503 dihydrochloride) is a selective σ1 receptor agonist (IC50: 17.4 nM). It shows selectivity for σ1 over σ2 receptors, and inhibits angiotensin II-induced cardiomyocyte hypertrophy in vitr...
T1885 Siramesine hydrochloride Lu 28-179 hydrochloride Ferroptosis , Sigma receptor , lysosomal autophagy
Siramesine hydrochloride (Lu 28-179 hydrochloride) is a selective sigma-2 receptor agonist, which has been shown to trigger cell death of Y cells and to exhibit a potent anticancer activity in vivo.
T6406 Besifloxacin Hydrochloride BOL-303224-A,Besivance hydrochloride,Besifloxacin HCl Antibacterial , Antibiotic
Besifloxacin Hydrochloride (BOL-303224-A) is a fourth-generation fluoroquinolone antibiotic.
T65281 Magnesium acetate tetrahydrate Endogenous Metabolite , Antibacterial
Magnesium acetate tetrahydrate is the hydrated form of the anhydrous magnesium acetate salt.Magnesium acetate tetrahydrate is commonly used to synthesize other compounds, cocoa as an electrolyte supplement or as a reagen...
T0991 Desipramine hydrochloride NSC-114901,Desmethylimipramine,JB-8181,EX-4355,Norimipramine,G-35020 Dopamine Receptor , 5-HT Receptor , Serotonin Transporter , Adrenergic Receptor
Desipramine hydrochloride (Norimipramine) ,a secondary amine tricyclic antidepressant (TCA), is the hydrochloride salt form of desipramine. In the central nervous system (CNS), Desipramine hydrochloride blocks the re-upt...

Compounds

ESI-08
T11234
Synonym:
Target: cAMP
ESI-09
T2244
Synonym:
Target: cAMP, Virus Protease
ESI-05
T15247
Synonym: NSC 116966
Target: cAMP
L-Ascorbic acid 2-phosphate magnesium
T19389
Synonym: 2-Phospho-L-ascorbic acid magnesium
Target: Phosphatase, Phosphorylase
Tesidolumab
T76831
Synonym: LFG316
Target: Complement System
Trotabresib
T36395
Synonym: CC-90010
Target: Epigenetic Reader Domain
Saroglitazar Magnesium
T12834
Synonym:
Target: Others
Forodesine
T15337
Synonym: BCX-1777,Immucillin-H
Target: Others
Galidesivir
T10491
Synonym: BCX4430,Immucillin-A
Target: Others
Besipirdine hydrochloride
T26778L
Synonym: HP 749 hydrochloride,Besipirdine hydrochloride(119257-34-0 Free base)
Target: Adrenergic Receptor
Peldesine
T12399
Synonym: BCX 34
Target: Nucleoside Antimetabolite/Analog, HIV Protease
Birabresib
T6032
Synonym: OTX-015,OTX015 (MK 8628/Birabresib),MK-8628
Target: Epigenetic Reader Domain
Sovilnesib
T39994
Synonym: AMG650
Target: Microtubule Associated
Ponesimod
T3258
Synonym: ACT-128800
Target: S1P Receptor, LPL Receptor
Bepotastine Besilate
T6405
Synonym: Talion,TAU 284,Bepreve,Bepotastine Beslilate
Target: Histamine Receptor
Magnesium glycinate
T4512
Synonym: magnesium 2-aminoacetate,Magnesium diglycinate
Target: Others
Besipirdine
T26778
Synonym: HP 749 free base,P-867493,P867493,HP 749,HP749,P 867493
Target: Sodium Channel, Adrenergic Receptor
Cesium chloride
T8391
Synonym: CsCl
Target: Potassium Channel
Resiquimod
T6964
Synonym: R848,S28463
Target: HCV Protease, TLR
Besifovir
T5832
Synonym:
Target: HBV
Ulodesine
T67822L
Synonym: BCX4208
Target: Endogenous Metabolite
Mivebresib
T3712
Synonym: ABBV-075
Target: Apoptosis, Epigenetic Reader Domain
Fibronectin Adhesion-promoting Peptide acetate
TP1153L
Synonym: Fibronectin Adhesion-promoting Peptide acetate(125720-21-0 free base),Heparin Binding Peptide acetate
Target: Others
Besifovir PM
T67817
Synonym: LB80331 PM
Target: HBV
Indomethacin farnesil
T7882
Synonym: Infree
Target: Others, COX, Autophagy
Sumaresinolic Acid
T8772
Synonym:
Target: Others
Alytesin acetate
TP2219L
Synonym:
Target: Others
[D-Phe12,Leu14]-Bombesin acetate
TP1916L1
Synonym: [D-Phe12,Leu14]-Bombesin acetate(108437-88-3 Free base)
Target: Bombesin Receptor
Lesinurad
T6875
Synonym: RDEA594
Target: OAT
Blarcamesine
T7780
Synonym: AE-37,AVex-73
Target: AChR
Chlorphenesin
T4507
Synonym: Adermykon,Chlorophenesin,Gecophen
Target: Antibacterial, Antifungal, Histamine Receptor
Remdesivir
T7766
Synonym: GS-5734
Target: SARS-CoV, DNA/RNA Synthesis
Esomeprazole Magnesium trihydrate
T8386
Synonym: (S)-Omeprazole magnesium trihydrate
Target: Proton pump
Magnesium sulfate
T40864
Synonym:
Target: Others
Filanesib
TQ0318
Synonym: ARRY-520,ARRY 520
Target: KSP
L-Threonic acid magnesium salt
T9379
Synonym:
Target: Others
Glutathione synthesis-IN-1
T9978
Synonym:
Target: Others
Bombesin acetate(31362-50-2 free base)
TP1281L1
Synonym:
Target: Bombesin Receptor
Calcium dobesilate
T5939
Synonym:
Target: Apoptosis, Others
Molibresib
T1906
Synonym: GSK 525762A,GSK525762,I-BET 762
Target: Epigenetic Reader Domain
Alobresib
T8495
Synonym: Vorolanib,GS-5829
Target: Epigenetic Reader Domain
Metamizole magnesium
T3272
Synonym: Metamizolemagnesiumsalt
Target: Antibiotic
[D-Phe12]-Bombesin acetate
TP2239L
Synonym: [D-Phe12]-Bombesin acetate(108437-87-2 free base)
Target: Bombesin Receptor
Esomeprazole Magnesium
T2686
Synonym: (S)-Omeprazole magnesium,NEXIUM,(-)-Omeprazole magnesium
Target: ATPase, Proton pump
Blarcamesine hydrochloride
T4111
Synonym: Anavex 2-73,AVex-73 hydrochloride,AE-37 hydrochloride
Target: Sigma receptor
Cutamesine dihydrochloride
T3597
Synonym: AGY94806 dihydrochloride,SA4503 (dihydrochloride),SA4503 dihydrochloride
Target: Sigma receptor
Siramesine hydrochloride
T1885
Synonym: Lu 28-179 hydrochloride
Target: Ferroptosis, Sigma receptor, lysosomal autophagy
Besifloxacin Hydrochloride
T6406
Synonym: BOL-303224-A,Besivance hydrochloride,Besifloxacin HCl
Target: Antibacterial, Antibiotic
Magnesium acetate tetrahydrate
T65281
Synonym:
Target: Endogenous Metabolite, Antibacterial
Desipramine hydrochloride
T0991
Synonym: NSC-114901,Desmethylimipramine,JB-8181,EX-4355,Norimipramine,G-35020
Target: Dopamine Receptor, 5-HT Receptor, Serotonin Transporter, Adrenergic Receptor
1 2 3 4
Cat No. Product Name Synonyms Targets
T13739 Isopropylidenylacetyl-marmesin (±)-Prantschimgin,Prantschimgin Others
Isopropylidenylacetyl-marmesin (Prantschimgin) is a natural product derived from the roots of Notopterygium incisum and Ferulago bracteata.
T5755 Aloesin Tyrosinase
Aloesin is a C-glycosylated chromone compound found in aloe (Liliaceae) that inhibits tyrosinase (IC50 = 0.9 mM), an enzyme responsible for catalyzing the first step of the conversion of tyrosine to melanin.
T3S0488 Syringaresinol diglucoside Syringaresinol-di-O-glucoside Others
Syringaresinol diglucoside (Syringaresinol-di-O-glucoside) protects the animals from the stress-induced decreases in sex behaviours and in rectal temperature, the stress-induced failure of retrieval of memory, and the st...
T9425 Epipinoresinol-4'-O-β-D-glucoside Others
Epipinoresinol-4'-O-β-D-glucoside (Simplocosin) is a glucoside compound[1].
TN1594 DL-Syringaresinol (±)-Syringaresinol Antioxidant , Antifungal
DL-Syringaresinol ( (±)-Syringaresinol) is a lignan from ginseng berries with anti-inflammatory, antioxidant, analgesic and weak anti-mycobacterial activities.DL-Syringaresinol can delay oxidative stress-induced skin agi...
T2S0531 Pinoresinol dimethyl ether (+)-Eudesmin Others , PKC
Pinoresinol dimethyl ether, a non-phenolic furan lignan isolated from the bark of Magnolia kobus, exhibits neuroactivity. It stimulates upstream MAPK, PKC, and PKA pathways, inducing neurite outgrowth in PC12 cells.
T4S0792 Pinoresinol 4-O-β-D-glucopyranoside (+)-pinor,(+)-pinoresinol-β-D-glucoside; (+)-pinor,(+)-pinoresinol-β-D-glucoside Others
(+)-Pinoresinol-β-D-glucoside, also known as (+)-pinor, is a major active lignan furanoid found in Forsythia. It exhibits antioxidative, antihypertensive activities, and acts as an inhibitor of cyclic adenosine monophosp...
TN2079 (-)-Pinoresinol Others , TNF , NF-κB , COX
(-)-Pinoresinol is isolated from the whole plant of Serissa japonica (Thunb.) Thunb.
TN1853 Lariciresinol VEGFR , Antifection
Lariciresinol is an enterolignan precursor, it possesses fungicidal activities by disrupting the fungal plasma membrane and therapeutic potential as a novel antifungal agent for the treatment of fungal infectious disease...
T22455 Vindesine sulfate DVA,Desacetylvinblastine amide,DAVA,Desacetyl Vinblastine amide,VDS Others
Vindesine sulfate (Desacetyl Vinblastine amide) is a vinca alkaloid which is a synthetic derivative of vinblastine, binds to the microtubular proteins of the mitotic spindle, leading to crystallization of the microtubule...
T4A2458 Resibufogenin Bufogenin,Recibufogenin Others
1. Resibufogenin (Bufogenin) is a cytotoxic steroid isolated from the Chinese drug ChanSu. 2. Resibufogenin can inhibit rectifier potassium current ( I K ) and transient potassium current ( I A ), it has pathological eff...
T5759 S-(+)-Marmesin (+)-Marmesin,(S)-Marmesin,marmesin Lipoxygenase , COX
S-(+)-Marmesin (marmesin) is a coumarin originally isolated from the mature bark of A. marmelos,exhibiting COX-2/5-LOX dual inhibitory activity.
TN2080 Pinoresinol (+)-Pinoresinol Apoptosis , NF-κB , CDK , p53
Pinoresinol ((+)-Pinoresinol) has antiinflammatory, hepatoprotective, and fungicidal activities, it can protect pial microcirculation from I-reperfusion injury, to increase nitric oxide release and to reduce oxidative st...
T8179 Aloeresin D Beta-Secretase , BACE
Aloeresin D, a natural chromone glycoside, inhibits β-Secretase (BACE1) activity (IC50: 39 μM).
TN1782 (+)-Isolariciresinol (+)-Cyclolariciresinol,Isolariciresinol Immunology/Inflammation related
(+)-Isolariciresinol ((+)-Cyclolariciresinol) is extracted from Radix Isatidis and shows antioxidant and anti-inflammatory activities and can be used in studies about rheumatism.
TMS0484 Episyringaresinol 4'-O-β-D-glncopyranoside (-)-Syringaresinol 4-O-β-D-glucopyranosi Others
Episyringaresinol 4'-O-β-D-glncopyranoside ((-)-Syringaresinol 4-O-β-D-glucopyranosi) inhibits the proliferation of human promyelocytic HL-6 cells through G(1) arrest and induction of apoptosis, may be a potential chemot...
T19281L Dihydroxyacetone phosphate hemimagnesium salt hydrate Dihydroxyacetone phosphate hemimagnesium salt hydrate(57-04-5 free base) Others
Dihydroxyacetone phosphate hemimagnesium salt hydrate is also known as dihydroxyacetone phosphate or 3-hydroxy-2-oxopropyl phosphate. Dihydroxyacetone phosphate hemimagnesium salt hydrate is found in all organisms from b...
T3S1265 Liriopesides B Nolinospiroside F Others
Liriopesides B (Nolinospiroside F) exhibited potential anticancer activity against human ovarian cancer A2780 cells.
T0739 Guaifenesin Glycerol guaiacolate,Guaiacol glyceryl ether,Guaiphenesin Others
Guaifenesin (Guaiphenesin) is an expectorant that also has some muscle relaxing action. It is used in many cough preparations.
T5S2178 Fargesin (+/-)-Fargesin Adrenergic Receptor
1. Fargesin ((+/-)-Fargesin) as a potential β1AR antagonist through cAMP/PKA pathway could protect against myocardial ischemia/reperfusion injury in rats. 2. Fargesin improves dyslipidemia and hyperglycemia by activating...
T21820 Resistomycin Geliomycin,Heliomycin Antibiotic
Resistomycin (Geliomycin), a pentacyclic polyketide antibiotic, exhibits potent anticancer properties by triggering apoptosis.
T34295 Resiniferatoxin RTX,[3H]resiniferatoxin IL Receptor
Resiniferatoxin ([3H]resiniferatoxin) inhibits the production of Th1 cytokines, contributing to the defense against T. spiralis infection, and can be used in studies about the modulator of the immune response.
TJS0487 (-)-Syringaresinol DL-Syringaresinol,Lirioresinol b Others
(-)-Syringaresinol (DL-Syringaresinol) is derived from the stems of Annona Montana. (-)-Syringaresinol inhibits the proliferation of human promyelocytic HL-60 cells through G1 arrest and induction of apoptosis and posses...
TN4510 (+)-Medioresinol Di-O-β-D-glucopyranoside (+)-Mediresinol Di-O-beta-D-glucopyranoside,(+)-Medioresinol Di-O-β-D-glucopyranoside PDE
(+)-Medioresinol Di-O-β-D-glucopyranoside has strong inhibitory activity of cyclic AMP phosphodiesterase.
T6S0535 Pinoresinol diglucoside Pinoresinol Diglucopyranoside Glucosidase
1. Pinoresinol diglucoside (Pinoresinol Diglucopyranoside) is a putative α-glucosidase inhibiting compound. 2. Pinoresinol diglucoside is a important antihypertensive compound.
T20793 Magnesium Lithospermate B Monomethyl lithospermate B,Lithospermate B Others
Magnesium Lithospermate B is a natural product activates eNOS and ameliorates endothelial dysfunction in diabetes by enhancing vasodilation in addition to reducing oxidative stress, it can protecte cardiomyocytes from is...
T3415 Secoisolariciresinol diglucoside LGM2605 ROS
Secoisolariciresinol diglucoside (LGM2605) was cytoprotective in an in vitro model of iron overload-induced redox-inflammatory damage. Secoisolariciresinol diglucoside (25 mg/kg b.w.) exerts the antihyperglycemic effect ...
TN2197 Secoisolariciresinol TNF
Secoisolariciresinol is an enterolignan precursor, it has antioxidant, and estrogen-like activities, it can significantly suppress triglyceride (TG) accumulation in 3T3-L1 adipocytes.
TN1916 Matairesinol ATPase , p38 MAPK , ROS
Matairesinol has radical and superoxide scavenging activities,; it also has anti-angiogenic activity by suppressing mROS signaling , can decrease hypoxia-inducible factor-1α± in hypoxic HeLa cells.
TP2223 Beesioside Q Others
Beesioside Q is a natural product extracted from the rhizome of Beesia calthaefolia (Maxim.) Ulbr.
TN5015 Siaresinolic acid 28-O-β-D-glucopyranosyl ester Siaresinolic acid 28-O-beta-D-glucopyranosyl ester Others
Siaresinolic acid 28-O-β-D-glucopyranosyl ester is a natural product for research related to life sciences. The catalog number is TN5015 and the CAS number is 155653-86-4.
TN5402 (-)-Pinoresinol 4-O-glucoside
(-)-Pinoresinol 4-O-glucoside is a natural product from Lonicera japonica THUNB.
TN3127 5'-Methoxylariciresinol Others
5'-Methoxylariciresinol is a natural product from Stellera chamaejasme.
TN3077 5,5'-Dimethoxylariciresinol 4-O-glucoside Others
5,5'-Dimethoxylariciresinol-4'-O-beta-D-glucoside is shown to effectively enhance chemosensitivity of resistant cells, which makes it may be a suitable candidate for potential multidrug resistance (MDR)-reversing agents.
TN5083 Syringaresinol diacetate Others
Syringaresinol diacetate is a natural product for research related to life sciences. The catalog number is TN5083 and the CAS number is 1990-77-8.
TMA0627 Taxiresinol TNF
Taxiresinol shows anticancer, antinociceptive, and antiallergic activities, it shows inhibitory activity on induced histamine release from the human basophilic cell line, KU812. Taxiresinol can protect the hepatocytes fr...
TN3355 Agatharesinol acetonide Antifection
Agatharesinol acetonide shows anticancer activity towards the A549 non-small-cell lung-cancer cell line (IC50 = 27.1 microM).
TN4305 (+)-Isolariciresinol 9'-O-glucoside
(+)-Isolariciresinol 9'-O-glucoside is a lignan glycoside that can be isolated from several plant species.
T8518 Erigeside I Others
Erigeside I is a radical scavenger.
TN4333 Isotaxiresinol 9,9'-acetonide Others
Isotaxiresinol 9,9'-acetonide is a natural product for research related to life sciences. The catalog number is TN4333 and the CAS number is 252333-72-5.
T79961 Aloeresin G
Aloeresin G, a chromone glycoside isolated from Aloe, exhibits a moderate inhibitory effect on TNFα-induced NF-κB transcriptional activity, evidenced by an IC50 of 40.02 μM [1].
TN3334 Abiesinol F Others
Abiesinol F is a natural product for research related to life sciences. The catalog number is TN3334 and the CAS number is 1190070-91-7.
TN3310 9,9'-Di-O-(E)-feruloylsecoisolariciresinol mTOR
1,4-O-Diferuloylsecoisolariciresinol(9,9'-Di-O-(E)-feruloylsecoisolariciresinol),and pierreione B, two novel inhibitors of mTOR signaling, have strong anticancer activity. (+)-9,9'-O-Diferuloylsecoisolariciresinol has si...
TN1392 Anhydrosecoisolariciresinol Others
Anhydrosecoisolariciresinol can significantly decrease the growth of human breast cancer MCF-7 and MDA-MB-231 cell lines at 50 and 100 microM.
TN5418 Secoisolariciresinol diglucoside (S,S)-Secoisolariciresinol diglucoside,(S,S)-SDG
Secoisolariciresinol diglucoside is a natural product for research related to life sciences. The catalog number is TN5418 and the CAS number is 257930-74-8.
TN6160 Pleionesin C
Pleionesin C is a natural product for research related to life sciences. The catalog number is TN6160 and the CAS number is 1222077-25-9.
TN2299 Vindesine Others
Vindesine is a microtubule inhibitor and widely used to treat malignancies. Vindesine neuropathy seems to be the cause of the patient's neurological symptoms.
TN4507 Matairesinoside Others
Matairesinoside is a natural product from Styrax japonica.
TN2545 1-Hydroxypinoresinol 1-O-glucoside ROS
(+)-1-Hydroxypinoresinol 1-O-beta-D-glucoside exhibits peroxynitrite, total ROS and DPPH radical scavenging activities with IC50 values of 3.23 +/- 0.04, 2.26 +/- 0.07 and 32.3 +/- 0.13 microM, respectively.
TN4927 Rupesin E Antifection
Rupesin E shows significant antibacterial activities against Escherichia coli.
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Natural Products

Isopropylidenylacetyl-marmesin
T13739
Synonym: (±)-Prantschimgin,Prantschimgin
Target: Others
Aloesin
T5755
Synonym:
Target: Tyrosinase
Syringaresinol diglucoside
T3S0488
Synonym: Syringaresinol-di-O-glucoside
Target: Others
Epipinoresinol-4'-O-β-D-glucoside
T9425
Synonym:
Target: Others
DL-Syringaresinol
TN1594
Synonym: (±)-Syringaresinol
Target: Antioxidant, Antifungal
Pinoresinol dimethyl ether
T2S0531
Synonym: (+)-Eudesmin
Target: Others, PKC
Pinoresinol 4-O-β-D-glucopyranoside
T4S0792
Synonym: (+)-pinor,(+)-pinoresinol-β-D-glucoside; (+)-pinor,(+)-pinoresinol-β-D-glucoside
Target: Others
(-)-Pinoresinol
TN2079
Synonym:
Target: Others, TNF, NF-κB, COX
Lariciresinol
TN1853
Synonym:
Target: VEGFR, Antifection
Vindesine sulfate
T22455
Synonym: DVA,Desacetylvinblastine amide,DAVA,Desacetyl Vinblastine amide,VDS
Target: Others
Resibufogenin
T4A2458
Synonym: Bufogenin,Recibufogenin
Target: Others
S-(+)-Marmesin
T5759
Synonym: (+)-Marmesin,(S)-Marmesin,marmesin
Target: Lipoxygenase, COX
Pinoresinol
TN2080
Synonym: (+)-Pinoresinol
Target: Apoptosis, NF-κB, CDK, p53
Aloeresin D
T8179
Synonym:
Target: Beta-Secretase, BACE
(+)-Isolariciresinol
TN1782
Synonym: (+)-Cyclolariciresinol,Isolariciresinol
Target: Immunology/Inflammation related
Episyringaresinol 4'-O-β-D-glncopyranoside
TMS0484
Synonym: (-)-Syringaresinol 4-O-β-D-glucopyranosi
Target: Others
Dihydroxyacetone phosphate hemimagnesium salt hydrate
T19281L
Synonym: Dihydroxyacetone phosphate hemimagnesium salt hydrate(57-04-5 free base)
Target: Others
Liriopesides B
T3S1265
Synonym: Nolinospiroside F
Target: Others
Guaifenesin
T0739
Synonym: Glycerol guaiacolate,Guaiacol glyceryl ether,Guaiphenesin
Target: Others
Fargesin
T5S2178
Synonym: (+/-)-Fargesin
Target: Adrenergic Receptor
Resistomycin
T21820
Synonym: Geliomycin,Heliomycin
Target: Antibiotic
Resiniferatoxin
T34295
Synonym: RTX,[3H]resiniferatoxin
Target: IL Receptor
(-)-Syringaresinol
TJS0487
Synonym: DL-Syringaresinol,Lirioresinol b
Target: Others
(+)-Medioresinol Di-O-β-D-glucopyranoside
TN4510
Synonym: (+)-Mediresinol Di-O-beta-D-glucopyranoside,(+)-Medioresinol Di-O-β-D-glucopyranoside
Target: PDE
Pinoresinol diglucoside
T6S0535
Synonym: Pinoresinol Diglucopyranoside
Target: Glucosidase
Magnesium Lithospermate B
T20793
Synonym: Monomethyl lithospermate B,Lithospermate B
Target: Others
Secoisolariciresinol diglucoside
T3415
Synonym: LGM2605
Target: ROS
Secoisolariciresinol
TN2197
Synonym:
Target: TNF
Matairesinol
TN1916
Synonym:
Target: ATPase, p38 MAPK, ROS
Beesioside Q
TP2223
Synonym:
Target: Others
Siaresinolic acid 28-O-β-D-glucopyranosyl ester
TN5015
Synonym: Siaresinolic acid 28-O-beta-D-glucopyranosyl ester
Target: Others
(-)-Pinoresinol 4-O-glucoside
TN5402
Synonym:
Target:
5'-Methoxylariciresinol
TN3127
Synonym:
Target: Others
5,5'-Dimethoxylariciresinol 4-O-glucoside
TN3077
Synonym:
Target: Others
Syringaresinol diacetate
TN5083
Synonym:
Target: Others
Taxiresinol
TMA0627
Synonym:
Target: TNF
Agatharesinol acetonide
TN3355
Synonym:
Target: Antifection
(+)-Isolariciresinol 9'-O-glucoside
TN4305
Synonym:
Target:
Erigeside I
T8518
Synonym:
Target: Others
Isotaxiresinol 9,9'-acetonide
TN4333
Synonym:
Target: Others
Aloeresin G
T79961
Synonym:
Target:
Abiesinol F
TN3334
Synonym:
Target: Others
9,9'-Di-O-(E)-feruloylsecoisolariciresinol
TN3310
Synonym:
Target: mTOR
Anhydrosecoisolariciresinol
TN1392
Synonym:
Target: Others
Secoisolariciresinol diglucoside
TN5418
Synonym: (S,S)-Secoisolariciresinol diglucoside,(S,S)-SDG
Target:
Pleionesin C
TN6160
Synonym:
Target:
Vindesine
TN2299
Synonym:
Target: Others
Matairesinoside
TN4507
Synonym:
Target: Others
1-Hydroxypinoresinol 1-O-glucoside
TN2545
Synonym:
Target: ROS
Rupesin E
TN4927
Synonym:
Target: Antifection

Recombinant Proteins

Cat No. Product Name Species Expression System
TMPY-01909 Elafin Protein, Human, Recombinant (His) Human HEK293 Cells
Elafin, also known as Elastase-specific inhibitor, Peptidase inhibitor 3, Protease inhibitor WAP3, Skin-derived antileukoproteinase, WAP four-disulfide core domain protein 14, PI3, WAP3 and WFDC14, is a secreted protein ...
TMPH-03031 P30 adhesin Protein, Mycoplasma pneumoniae, Recombinant (GST & His) Mycoplasma pneumoniae E. coli
Adhesin necessary for successful cytadherence and virulence. P30 adhesin Protein, Mycoplasma pneumoniae, Recombinant (GST & His) is expressed in E. coli expression system with N-6xHis-GST tag. The predicted molecular wei...
TMPH-03144 SEY1 Protein, Plasmodium knowlesi, Recombinant (His) Plasmodium knowlesi E. coli
Probable GTP-binding protein that may be involved in cell development. SEY1 Protein, Plasmodium knowlesi, Recombinant (His) is expressed in E. coli expression system with N-10xHis tag. The predicted molecular weight is 1...
TMPY-02660 Resistin Protein, Mouse, Recombinant (hFc) Mouse HEK293 Cells
Resistin is an adipocytokine, which has been studied for its role in insulin resistance and recently in inflammation. The RETN and CAP1 polymorphisms and gene expression may be potential biomarkers for breast cancer risk...
TMPJ-00014 Resistin Protein, Human, Recombinant (His) Human E. coli
Resistin known as adipose tissue-specific secretory factor (ADSF) or C/EBP-epsilon-regulated myeloid-specific secreted cysteine-rich protein (XCP1) that seems to suppress insulin ability to stimulate glucose uptake into ...
TMPH-00298 Resistin Protein, Bovine, Recombinant (His) Bovine E. coli
Hormone that seems to suppress insulin ability to stimulate glucose uptake into adipose cells. Potentially links obesity to diabetes. Resistin Protein, Bovine, Recombinant (His) is expressed in E. coli expression system ...
TMPY-01127 Influenza A H5N1 (A/Indonesia/5/2005) Hemagglutinin/HA Protein (His) H5N1 HEK293 Cells
Influenza A H5N1 (A/Indonesia/5/2005) Hemagglutinin/HA Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 59 kDa and the accession number is A8HWY8.
TMPY-04305 Influenza A H5N1 (A/Indonesia/5/2005) Hemagglutinin/HA Protein (R339G & S341R, His) H5N1 Baculovirus Insect Cells
Influenza A H5N1 (A/Indonesia/5/2005) Hemagglutinin/HA Protein (R339G & S341R, His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 60 kDa and the accession number is A8HWY8.
TMPY-02847 Moesin Protein, Human, Recombinant (aa 1-346, His) Human E. coli
Moesin is a member of the ERM family which includes ezrin and radixin. ERM proteins, highly related members of the larger protein 4.1 superfamily, can exist in an active or inactive conformation. It seems that ERM protei...
TMPH-00508 Pro-resilin Protein, Drosophila melanogaster, Recombinant (His & Myc) Fruit fly E. coli
Plays a central role in insect flight by providing low stiffness, high strain and efficient energy storage.
TMPY-04589 Influenza A H5N1 (A/Indonesia/5/2005) Hemagglutinin/HA-specific B cell probe Protein (His) H5N1 Baculovirus Insect Cells
Influenza A H5N1 (A/Indonesia/5/2005) Hemagglutinin/HA-specific B cell probe Protein (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 58.2 kDa and the accession number is AHJ...
Cat No. Product Name
L7900 Osteogenesis Compound Library

317 compounds
A unique collection of 317 osteogenesis related compounds for high throughput and high content screening;
L4800 Angiogenesis related Compound Library

1353 compounds
A unique collection of 1353 proangiogenic and antiangiogenic compounds for new targets identification, research in mechanisms of angiogenesis, and high throughput screening (HTS) and high content screening (HCS);
L7100 Anti-Obesity Compound Library

2247 compounds
A unique collection of 2247 anti-obesity compounds for high throughput and high content screening;
TargetMol