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  • Methionine Adenosyltransferase (MAT)
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Results for "

mat

" in TargetMol Product Catalog
  • Inhibitors & Agonists
    633
    TargetMol | Inhibitors_Agonists
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    TargetMol | Inhibitors_Agonists
MAT2A-IN-10
T789462924825-23-8
MAT2A-IN-10 (Compound 28), an orally active inhibitor of MAT2A, exhibits an IC50 of 26 nM and is utilized in cancer research [1].
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8-10 weeks
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MAT2A-IN-11
T79349
MAT2A Allosteric Inhibitor 1, also known as Compound 5, is a selective inhibitor of methionine adenosyltransferase (MAT) demonstrating potent activity with an IC50 value of 6.8 nM [1].
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MAT2A-IN-12
T79350631897-75-1
MAT2A Allosteric Inhibitor 2 is a potent, selective inhibitor exhibiting an IC50 of 5 nM and demonstrates nanomolar efficacy (IC50 = 5 μM) in proliferation assays utilizing the MTAP - - cell line [1].
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8-10 weeks
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MAT2A-IN-9
IDE397, GSK-4362676
T731402439277-80-0
MAT2A-IN-9, a 2-oxoquinazoline derivative, is a potent MAT2A (methionine adenylyltransferase 2A) inhibitor.MAT2A-IN-9 has antitumor activity for the treatment of lymphomas and solid tumors.
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6-8 weeks
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TargetMol | Inhibitor Sale
Rabies Virus Matrix Protein Fragment(RV-MAT)
T765551023648-37-4
Rabies Virus Matrix Protein Fragment (RV-MAT), a polypeptide, selectively binds to the acetylcholine receptor (AChR) on the cell surface [1].
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MAT-POS-e194df51-1
T81849
MAT-POS-e194df51-1 is an orally active, non-covalent, non-peptide inhibitor of the SARS-CoV-2 main protease (M^pro) with an IC_50 of 37 nM. It exhibits cytotoxicity, showing EC_50 values of 64 nM in A549-ACE2-TMPRSS2 cells and 126 nM in HeLa-ACE2 cells [1].
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Imatinib Mesylate
STI-571, ST-1571 Mesylate, CGP-57148B
T1621220127-57-1
Imatinib Mesylate (STI-571) is a tyrosine kinase receptor inhibitor with antineoplastic activity (IC50s: 0.6 μM, 0.1 μM and 0.1 μM for v-Abl, c-Kit and PDGFR, respectively).
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TargetMol | Inhibitor Hot
Palmatine chloride
T271810605-02-4
Palmatine chloride an isoquinoline alkaloid, is an important medicinal herbal extract with diverse pharmacological and biological properties.
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TargetMol | Inhibitor Hot
Fostamatinib
R788
T6115901119-35-5
Fostamatinib (R788)(IC50 of 41 nM), which is a prodrug of the active metabolite R406, is a Syk inhibitor. It does not work on Lyn.
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TargetMol | Inhibitor Hot
Nirmatrelvir
T93512628280-40-8
PF-07321332 is a potent and orally active inhibitor of SARS-CoV 3C-like protease (3CLPRO) .
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TargetMol | Inhibitor Hot
Somatostatin 1-28 acetate
Somatostatin 1-28 acetate(74315-46-1 Free base)
TP2124L
Somatostatin 1-28 acetate circulates in human plasma. Approximately 46% of the total somatostatin-like immunoreactivity in plasma is due to Somatostatin 1-28 acetate.
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TargetMol | Inhibitor Hot
Asperphenamate
T1039063631-36-7In house
Asperphenamate is a fungal metabolite of Aspergillus flatiipes. The IC50s for T47D cells, MDA-MB-231 cells, and HL-60 cells are 92.3 μM, 96.5 μM, and 97.9 μM. Asperphenamate shows an anticancer effect.
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6-8 weeks
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BMT-124110 Formate
BMT-124110 Formate(1679371-59-5 Free base)
T10572L In house
BMT-124110 Formate is a selective AAK1 inhibitor (IC50: 0.9 nM) with anti-injury sensory activity.BMT-124110 Formate inhibits the BMP-2-inducible protein kinase BIKE with an IC50: 17 nM.BMT-124110 Formate inhibits the cell-cycle protein G-related BMT-124110 Formate inhibits the cell cycle protein G-associated kinase GAK with an IC50:99 nM.
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BPO-27 racemate
BPO-27 (racemate)
T105911314873-02-3In house
BPO-27 racemate (BPO-27 (racemate)) is an effective CFTR inhibitor with IC50 of 8 nM.
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6-8 weeks
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TargetMol | Inhibitor Sale
Bucindolol Formate
Bucindolol Formate (71119-11-4 Free base)
T10631L In house
Bucindolol Formatel is a blocker of β1-adrenergic receptor. Bucindolol exhibits intrinsic sympathomimetic activity. Bucindolol can be used in the research of heart failure.
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ELN318463 racemate
ELN318463 (racemate), ELN 318463 racemate
T11178L851599-82-1In house
ELN318463 racemate (ELN 318463 racemate) is the racemate of ELN318463 which is an amyloid precursor protein (APP) selective γ-secretase inhibitor.
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6-8 weeks
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Estradiol 3-sulfamate
ES-J 995, E2MATE, BLE 00084
T11235172377-52-5In house
Estradiol 3-sulfamate (BLE 00084) is an orally active and highly potent steroidal estrone sulfatase (ES) inhibitor.Estradiol 3-sulfamate has a K(i) value of 73 nM for ES in human placental microsomes and can be used in the study of breast cancer.
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7-10 days
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JTV-519 Formate
JTV-519 Formate (145903-06-6 Free base)
T11731L In house
JTV-519 Formate is a Ca2+-dependent blocker of sarcoplasmic reticulum Ca2+-stimulated ATPase (SERCA). JTV-519 Formate is also a partial agonist of ryanodine receptors in striated muscle. JTV-519 Formate exhibits antiarrhythmic and cardioprotective properties.
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Nexopamil racemate
(Rac)-Nexopamil
T12215116759-35-4In house
Nexopamil racemate((Rac)-Nexopamil) is a racemate of Nexopamil. The Nexopamil racemate has potential anti-asthmatic and anti-ulcer activity.
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6-8 weeks
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Peliglitazar racemate
BMS 426707-01 racemate, (Rac)-Peliglitazar, (Rac)-BMS 426707-01
T12400331744-72-0In house
Peliglitazar racemate(BMS 426707-01 racemate) is the racemate of Peliglitazar.Peliglitazar racemate may be used as a potential antidiabetic and anti-obesity agent.
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6-8 weeks
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WAY127093B racemate
T13331145743-63-1In house
WAY127093B racemate is the racemic mixture of WAY127093B, a phosphodiesterase IV inhibitor with demonstrated oral activity in rats and guinea pigs.
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6-8 weeks
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TargetMol | Inhibitor Sale
Pamatolol
T1643159110-35-9In house
Pamatolol is a selective and potent beta-adrenoceptor antagonist that has not shown sympathomimetic activity in ex vivo experiments.
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6-8 weeks
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Rentiapril racemate
SA-446 racemate, (Rac)-SA-446, (Rac)-Rentiapril
T1673172679-47-1In house
Rentiapril racemate (SA-446 racemate) is the racemic form of Rentiapril, exhibiting anti-inflammatory properties and potential applications in glaucoma research.
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6-8 weeks
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Gimatecan
LBQ707, STI481
T21319292618-32-7In house
Gimatecan (STI481) is a potent topoisomerase I inhibitor. Gimatecan is an orally bioavailable camptothecin analogue with antitumor activity.
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10-14 weeks
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