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PRL 2915 is a potent antagonist of the human somatostatin subtype 2 receptor (hsst 2), exhibiting a binding affinity (K_i) of 12 nM [1].
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50 mg | Inquiry | Backorder |
Description | PRL 2915 is a potent antagonist of the human somatostatin subtype 2 receptor (hsst 2), exhibiting a binding affinity (K_i) of 12 nM [1]. |
Targets&IC50 | SST2 (human):1.8 nM (rat antagonist bioassay versus somatostatin), SST3 (human):100 nM (Ki), SST2 (human):12 nM (Ki), SST5 (human):520 nM (Ki), SST4 (human):895 nM (Ki), UTII receptor (human):562 nM (Ki), SST1 (human):>1000 nM (Ki), UTII receptor (rat):293 nM (Ki) |
Molecular Weight | 1175.85 |
Formula | C59H71ClN12O8S2 |
Cas No. | 209006-18-8 |
Sequence | {Phe<4-Cl>}-{d-Cys}-{β-Ala<3-Py>}-{d-Trp}-Lys-{Val<3-Me>}-Cys-{2-Nal}-NH2(Disulfide bond) |
Sequence Short | {F<4-Cl>}-{d-C}-{β-A<3-Py>}-{d-W}-K-{V<3-Me>}-C-{A<3(2-Naph)>}-NH2 (Disulfide bridge:Cys2-Cys7) |
Storage | keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature. |
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