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CYN 154806 TFA

Name: CYN 154806 TFA
Brand: TargetMol
SKU: TP1346
Price: 147 USD
Availability: InStock
Rating: 5 (10 reviews)

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Catalog No. TP1346Cas No. 2828432-46-6

Alias CYN 154806 TFA

CYN 154806 TFA is a cyclic octapeptide and an effective selective somatostatin sst2 receptor antagonist. For the recombinant sst2, sst1, sst3, sst4 and sst5 receptors, the pIC50 values are 8.58, 5.41, 6.07, 5.76 and 6.48, respectively.

CYN 154806 TFA

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Purity: 99.7%

Catalog No. TP1346Alias CYN 154806 TFACas No. 2828432-46-6

Pack Size	Price	USA Warehouse	Global Warehouse
1 mg	$147	In Stock	In Stock
5 mg	$478	In Stock	In Stock
10 mg	$689	In Stock	In Stock
25 mg	$1,080	In Stock	In Stock
50 mg	$1,480	In Stock	In Stock
100 mg	$1,960	In Stock	In Stock

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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]

All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.

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Purity:99.7%

Appearance:Solid

Color:White

Resource Download

COA LCMS HNMR

Product Introduction

Bioactivity

Description	CYN 154806 TFA is a cyclic octapeptide and an effective selective somatostatin sst2 receptor antagonist. For the recombinant sst2, sst1, sst3, sst4 and sst5 receptors, the pIC50 values are 8.58, 5.41, 6.07, 5.76 and 6.48, respectively.
Synonyms	CYN 154806 TFA

Chemical Properties

Molecular Weight	1311.36
Formula	C₅₈H₆₉F₃N₁₂O₁₆S₂
Cas No.	2828432-46-6
Smiles	C[C@@H](O)[C@H]1C(N[C@H](C(N[C@@H](C(N)=O)CC2=CC=C(O)C=C2)=O)CSSC[C@@H](NC([C@@H](NC(C)=O)CC3=CC=C([N+]([O-])=O)C=C3)=O)C(N[C@@H](CC4=CC=C(O)C=C4)C(N[C@H](CC5=CNC6=CC=CC=C65)C(N[C@@H](CCCCN)C(N1)=O)=O)=O)=O)=O.OC(C(F)(F)F)=O
Relative Density.	no data available
Sequence	Ac-FCYWKTCY-NH2 (Disulfide bridge: Cys2-Cys7)
Sequence Short	Phe-Cys-Tyr-Trp-Lys-Thr-Cys-Tyr (Disulfide bridge: Cys2-Cys7)

Storage & Solubility Information

Storage

keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

H2O: 50 mg/mL (38.13 mM), Sonication is recommended.

Solution Preparation Table

H2O

	1mg	5mg	10mg	50mg
1 mM	0.7626 mL	3.8128 mL	7.6257 mL	38.1284 mL
5 mM	0.1525 mL	0.7626 mL	1.5251 mL	7.6257 mL
10 mM	0.0763 mL	0.3813 mL	0.7626 mL	3.8128 mL
20 mM	0.0381 mL	0.1906 mL	0.3813 mL	1.9064 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the stock solution preparation method and in vivo formula preparation method:

For example, if the intended dosage is 10 mg/kg for animals weighing 20 g , with a dosing volume of 100 μL per animal, TargetMol | Animal experiments

and a total of 10 animals are to be administered, using a formulation of TargetMol | reagent

10% DMSO+ 40% PEG300+ 5% Tween 80+ 45% Saline/PBS/ddH₂O , the resulting working solution concentration would be 2 mg/mL.

Stock Solution Preparation:

Dissolve 2 mg of the compound in 100 μL DMSO TargetMol | reagent to obtain a stock solution at a concentration of 20 mg/mL . If the required concentration exceeds the compound's known solubility, please contact us for technical support before proceeding.

Preparation of the In Vivo Formulation:

1) Add 100 μL of the DMSO TargetMol | reagent stock solution to 400 μL PEG300 and mix thoroughly until the solution becomes clear.

2) Add 50 μL Tween 80 and mix well until fully clarified.

3) Add 450 μL Saline,PBS or ddH₂O TargetMol | reagent and mix thoroughly until a homogeneous solution is obtained.

This example is provided solely to demonstrate the use of the In Vivo Formulation Calculator and does not constitute a recommended formulation for any specific compound. Please select an appropriate dissolution and formulation strategy based on your experimental model and route of administration.

All co-solvents required for this protocol, includingDMSO, PEG300/PEG400, Tween 80, SBE-β-CD, and Corn oil, are available for purchase on the TargetMol website.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc