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[Tyr3]Octreotate

🥰Excellent
Catalog No. T67931Cas No. 302794-43-0

[Tyr3]Octreotate is a long peptide compound containing 8 amino acids and is a functional DOTA chelating agent with covalent bonds. [Tyr3]Octreotate binds to transmembrane receptors of SSR2-active NETs and is actively transported into cells by endocytosis, which may increase the required double-stranded DNA breaks and is a potential drug for tumor treatment.

[Tyr3]Octreotate

[Tyr3]Octreotate

🥰Excellent
Purity: 98.21%
Catalog No. T67931Cas No. 302794-43-0
[Tyr3]Octreotate is a long peptide compound containing 8 amino acids and is a functional DOTA chelating agent with covalent bonds. [Tyr3]Octreotate binds to transmembrane receptors of SSR2-active NETs and is actively transported into cells by endocytosis, which may increase the required double-stranded DNA breaks and is a potential drug for tumor treatment.
Pack SizePriceAvailabilityQuantity
1 mg$195In Stock
5 mg$447In Stock
10 mg$659In Stock
25 mg$987In Stock
50 mg$1,380In Stock
100 mg$1,890In Stock
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Purity:98.21%
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COA HPLC MS

Product Introduction

Bioactivity
Description
[Tyr3]Octreotate is a long peptide compound containing 8 amino acids and is a functional DOTA chelating agent with covalent bonds. [Tyr3]Octreotate binds to transmembrane receptors of SSR2-active NETs and is actively transported into cells by endocytosis, which may increase the required double-stranded DNA breaks and is a potential drug for tumor treatment.
Chemical Properties
Molecular Weight1049.22
FormulaC49H64N10O12S2
Cas No.302794-43-0
SmilesC(C=1C=2C(NC1)=CC=CC2)[C@H]3NC(=O)[C@H](CC4=CC=C(O)C=C4)NC(=O)[C@@H](NC([C@@H](CC5=CC=CC=C5)N)=O)CSSC[C@@H](C(N[C@@H]([C@@H](C)O)C(O)=O)=O)NC(=O)[C@]([C@@H](C)O)(NC(=O)[C@H](CCCCN)NC3=O)[H]
Relative Density.1.44 g/cm3 (Predicted)
SequenceH-D-Phe-Cys(1)-Tyr-D-Trp-Lys-Thr-Cys(1)-Thr-OH
Sequence ShortFCYWKTCT
Storage & Solubility Information
Storagestore at low temperature,keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
Solubility Information
DMSO: 100 mg/mL (95.31 mM), Sonication is recommended.
H2O: 100 mg/mL (95.31 mM), Sonication is recommended.
Solution Preparation Table
DMSO/H2O
1mg5mg10mg50mg
1 mM0.9531 mL4.7654 mL9.5309 mL47.6544 mL
5 mM0.1906 mL0.9531 mL1.9062 mL9.5309 mL
10 mM0.0953 mL0.4765 mL0.9531 mL4.7654 mL
20 mM0.0477 mL0.2383 mL0.4765 mL2.3827 mL
50 mM0.0191 mL0.0953 mL0.1906 mL0.9531 mL

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Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH2OTargetMol | reagent mix well and clarify
For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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Keywords

[Tyr3]Octreotateacetate(freebase)[Tyr3]Octreotate
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