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Results for "

orally active

" in TargetMol Product Catalog
  • Inhibitors & Agonists
    3129
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SEW​2871
SEW2871
T2171256414-75-2
SEW 2871 is an orally available, highly selective S1P1 agonist with an EC50 of 13.8 nM.It reduces the number of lymphocytes in the blood and is used in studies related to diabetes, Alzheimer's disease, liver fibrosis, and inflammation. It activates ERK, Akt and Rac signaling pathways and induces S1P1 internalization and recycling.
  • $48
In Stock
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TargetMol | Inhibitor Hot
Upadacitinib
ABT-494
T75031310726-60-3
Upadacitinib (ABT-494) (ABT-494) is a selective Janus kinase (JAK) 1 inhibitor, which is being studied for the treatment of several autoimmune disorders in the IC50 of 43 nM.
  • $53
In Stock
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TargetMol | Inhibitor Hot
LB42708
T2678226929-39-1In house
LB42708 is an orally active farnesyltransferase (FTase) inhibitor (IC50: 0.8/1.2/2.0 nM toward H/N/K-ras).
  • $35
In Stock
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Pilsicainide HCl
SUN 1165
T781188069-49-2In house
Pilsicainide HCl (SUN 1165) is a pure sodium channel blocker
  • $31 TargetMol
In Stock
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Sumatriptan succinate
GR 43175
T0203103628-48-4
Sumatriptan succinate (GR 43175), a serotonin1 (5-HT1) receptor agonist, is used in the acute treatment of a migraine headache.
  • $31
In Stock
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Lamivudine
GR109714X, BCH-189
T0682134678-17-4
Lamivudine (BCH-189) is a reverse transcriptase inhibitor and ZALCITABINE analog in which a sulfur atom replaces the 3' carbon of the pentose ring. It is used to treat HIV disease.
  • $53
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Ganciclovir
RS-21592, BW 759, 2'-Nor-2'-deoxyguanosine
T068882410-32-0
Ganciclovir (2'-Nor-2'-deoxyguanosine) is an ACYCLOVIR analog that is a potent inhibitor of the Herpesvirus family including cytomegalovirus. Ganciclovir is used to treat complications from AIDS-associated cytomegalovirus infections.
  • $51
In Stock
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Allopurinol
Zyloric, Zyloprim, Lopurin
T0692315-30-0
Allopurinol (Zyloric) is a Xanthine Oxidase Inhibitor. The mechanism of action of allopurinol is as a Xanthine Oxidase Inhibitor.
  • $50
In Stock
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Gentamicin sulfate
SCH9724, NSC-82261, Gentamycin sulfate
T13261405-41-0
Gentamicin sulfate (SCH9724) is a wide-spectrum, aminoglycoside antibiotic used to inhibit protein synthesis in sensitive organisms.
  • $31
In Stock
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Prednisolone
Predonine, Metacortandralone, Hydroretrocortine
T156050-24-8
Prednisolone (Hydroretrocortine) is a synthetic glucocorticoid with anti-inflammatory and immunomodulating properties.
  • $29
In Stock
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Isotretinoin
13-cis-Retinoic acid
T16114759-48-2
Isotretinoin (13-cis-Retinoic acid) binds to and activates nuclear retinoic acid receptors (RARs), which act as transcription factors that promote cell differentiation and apoptosis. This naturally occurring retinoic acid has potential antineoplastic activity, exhibits immunomodulatory and anti-inflammatory responses, and inhibits ornithine decarboxylase, thereby decreasing polyamine synthesis and keratinization.
  • $36
In Stock
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Hydralazine hydrochloride
Hydralazine HCl, Apresoline
T1613304-20-1
Hydralazine hydrochloride (Apresoline) is the hydrochloride salt of hydralazine, a phthalazine derivative with antihypertensive and potential antineoplastic activities. Hydralazine alters intracellular calcium release and interferes with smooth muscle cell calcium influx, resulting in arterial vasodilatation. This agent also inhibits the phosphorylation of myosin protein and chelation of trace metals required for smooth muscle contraction, resulting in an increase in heart rate, stroke volume, and cardiac output. In addition to its cardiovascular effects, hydralazine inhibits DNA methyltransferase, which may result in inhibition of DNA methylation in tumor cells.
  • $36
In Stock
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Afatinib Dimaleate
BIBW2992, BIBW 2992MA2, Afatinib (BIBW2992) Dimaleate, Afatinib
T1773850140-73-7
Afatinib Dimaleate (BIBW 2992MA2) is an orally bioavailable anilino-quinazoline derivative and inhibitor of the receptor tyrosine kinase (RTK) epidermal growth factor receptor (ErbB; EGFR) family, with antineoplastic activity.
  • $33
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Ivabradine hydrochloride
S 16257-2, Ivabradine HCl
T2535148849-67-6
Ivabradine hydrochloride (S 16257-2) is a new If inhibitor (IC50: 2.9 μM). Ivabradine Hydrochloride is the hydrochloride salt form of ivabradine, an orally bioavailable, hyperpolarization-activated, cyclic nucleotide-gated (HCN) channel blocker, with negative chronotropic activity. Upon administration, ivabradine selectively binds to the intracellular portion of the HCN channel pore and blocks HCN channels in the pacemaker cells within the sinoatrial (SA) node. This inhibits the If (funny) pacemaker ion current, prevents the inward flow and intracellular accumulation of positively charged ions, reduces pacemaker activity and slows diastolic depolarization.
  • $33
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Didanosine
ddI, 2',3'-Dideoxyinosine
T257869655-05-6
Didanosine (ddI) is a nucleoside reverse transcriptase inhibitor analog of adenosine (IC50: 0.49 μM).
  • $33
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Succinic acid
Wormwood acid, Butanedioic acid, Asuccin, Amber acid, 1,4-Butandioic Acid, 1,2-Ethanedicarboxylic acid
T2719110-15-6
Succinic acid (1, 2-ethanedicarboxylic acid) is a product of anaerobic metabolism and an intermediate of the tricarboxylic acid cycle.
  • $33
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NADH disodium salt
NADH, disodium salt hydrate, Disodium NADH
T5283606-68-8
NADH disodium salt (Disodium NADH) hydrate is the reduced form of nicotinamide adenine dinucleotide (NAD) that can donate electrons in a reducing reaction, becoming oxidized to produce NAD+. Various enzymes utilize NADH disodium salt hydrate plus H+ to reduce substrates, generating NAD+ and the reduced product.
  • $45
In Stock
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Fidaxomicin
Tiacumicin B, PAR-101, OPT-80, Clostomicin B1
T6194873857-62-6
Fidaxomicin (Tiacumicin B) is a semisynthetic macrolide antibiotic used to treat Clostridium difficile-associated diarrhea in adults. Fidaxomicin has minimal systemic absorption and has not been linked to serum enzyme elevations during therapy or to instances of clinically apparent, acute liver injury.
  • $40
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IDRA-21
T782322503-72-6
IDRA-21 is a positive AMPA receptor modulator.
  • $31
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Brexpiprazole HCl
OPC 34712 dihydrochloride
T8690913612-38-1
Brexpiprazole HCl (OPC 34712 dihydrochloride) is a new antipsychotic drug.
  • $133
In Stock
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Choline
T8734123-41-1
Choline is a ubiquitous water soluble nutrient, often associated with the B vitamins
  • $29
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AS057278
3-Methylpyrazole-5-carboxylic acid
T7476402-61-9
AS057278 (3-Methylpyrazole-5-carboxylic acid) is an D-amino acid oxidase (DAAO) inhibitor.
  • $30
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TargetMol | Inhibitor Sale
Tiapride hydrochloride
T129251012-33-0
Tiapride is a selective blocker of D2/3 dopamine receptors in the brain. It is used in the therapy of various psychiatric and neurological disorders containing dyskinesia, negative symptoms of psychosis, alcohol withdrawal syndrome, and aggression and agitation in the elderly.
  • $36
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RX-3117
TV-1360, fluorocyclopentenylcytosine
T16813865838-26-2
RX-3117 (fluorocyclopentenylcytosine) is a novel a cytidine analog. RX-3117 displays anticancer activity in several cancer cell lines, including gemcitabine-resistant variants.
  • $159
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