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Lenalidomide-acetylene-Br

🥰Excellent
Catalog No. T210445Cas No. 2619512-84-2

Lenalidomide-acetylene-Br is the PROTAC linker that makes up HJM-561. HJM-561 is an effective, selective, and orally active EGFR PROTAC that can inhibit the triple mutation of EGFR which is resistant to Osimertinib.

Lenalidomide-acetylene-Br

Lenalidomide-acetylene-Br

🥰Excellent
Catalog No. T210445Cas No. 2619512-84-2
Lenalidomide-acetylene-Br is the PROTAC linker that makes up HJM-561. HJM-561 is an effective, selective, and orally active EGFR PROTAC that can inhibit the triple mutation of EGFR which is resistant to Osimertinib.
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Product Introduction

Bioactivity
Description
Lenalidomide-acetylene-Br is the PROTAC linker that makes up HJM-561. HJM-561 is an effective, selective, and orally active EGFR PROTAC that can inhibit the triple mutation of EGFR which is resistant to Osimertinib.
Chemical Properties
Molecular WeightO=C1NC(=O)C(N2C(=O)C=3C=CC=C(C#CCCBr)C3C2)CC1
FormulaC17H15BrN2O3
Cas No.2619512-84-2
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

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Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH2OTargetMol | reagent mix well and clarify
For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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