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TargetMol | Compound Library

Orally Active Compound Library

Catalog No. L9850

Oral administration is the first choice for clinical drug delivery, especially for long-term use. It is also the safest, most convenient, and most economical method of drug delivery. Oral bioavailability is the percentage of the absorbed drug dose successfully passed through the mucosa of the gastrointestinal tract and entered the bloodstream through the liver, to the original given oral dose. Drugs with high oral bioavailability can achieve efficacy at lower doses and effectively reduce toxic side effects; while when bioavailability is too low, even compounds with good pharmacological activity are unable to be fully exposed and utilized at the target site, resulting in therapeutic failure or high dose with large toxic side effects, which eventually leads to drug development failure and limits the application. TargetMol has carefully collected 3160 compounds with publicly reported oral activity that can be used for drug repurposing and development of orally active drugs.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L9850

Orally Active Compound Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 3160 of orally active compounds for high-throughput screening and high-content screening.
  • Some drugs are approved or are in clinical trials with validated biological activity and safety.
  • Detailed specifications, compound structures, target information, activity descriptions, etc.
  • NMR and HPLC detection techniques to ensure high product purity.
  • All compounds are available in stock.

Packaging And Storage Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
  • This compound library is provided at a concentration of 10 mM in DMSO. A small number of compounds may be provided in different solvents or concentrations due to solubility or stability requirements. Please refer to the specific product information for details.

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Apoptosis
Autophagy
Antibacterial
Antibiotic
Endogenous Metabolite
5-HT Receptor
Adrenergic Receptor
Dopamine Receptor
Histamine Receptor
Parasite
COX
AChR
DNA/RNA Synthesis
HIV Protease
Potassium Channel
VEGFR
EGFR
Calcium Channel
Cytochromes P450
Sodium Channel
SARS-CoV
PDE
CDK
PDGFR
Estrogen/progestogen Receptor
Reactive Oxygen Species
FLT
Dehydrogenase
Glucocorticoid Receptor
c-Kit
Virus Protease
p38 MAPK
NF-κB
RAAS
Estrogen Receptor/ERR
PI3K
Ferroptosis
JAK
HCV Protease
Antifungal
Topoisomerase
Mitophagy
Ras
Src
FGFR
Microtubule Associated
HBV
PPAR
iGluR
Influenza Virus
c-Met/HGFR
Serotonin Transporter
Reverse Transcriptase
HDAC
Bcr-Abl
GABA Receptor
Proteasome
TRP/TRPV Channel
Prostaglandin Receptor
GPCR
GluR
Akt
Androgen Receptor
Interleukin
TNF
Phosphatase
ERK
Epigenetic Reader Domain
mTOR
Raf
Norepinephrine
Histone Methyltransferase
LPL Receptor
ALK
Adenosine Receptor
Progesterone Receptor
Tyrosine Kinases
Nucleoside Antimetabolite/Analog
MMP
PARP
ROS
Cholinesterase (ChE)
MAPK
Transferase
HSV
Beta Amyloid
STAT
HIF/HIF Prolyl-Hydroxylase
Monoamine Oxidase
Integrin
Caspase
Mitochondrial Metabolism
Angiotensin-converting Enzyme (ACE)
P-gp
HSP
Proton pump
GSK-3
Opioid Receptor
DPP-4
Antiviral
c-Fms
ribosome
Kras
Bcl-2 Family
MEK
S1P Receptor
HER
Factor Xa
NMDAR
Trk receptor
Retinoid Receptor
AMPK
Thrombin
NO Synthase
Leukotriene Receptor
ROCK
Aurora Kinase
Lipoxygenase
c-RET
Syk
Reductase
Wnt/beta-catenin
PKC
MAO
Drug Metabolite
Endothelin Receptor
Phospholipase
TAM Receptor
ROS Kinase
ATPase
Carbonic Anhydrase
MRP
Gamma-secretase
CCR
CXCR
SGLT
Acyltransferase
Cannabinoid Receptor
Thyroid hormone receptor(THR)
DHFR
NADPH
JNK
Serine Protease
E1/E2/E3 Enzyme
Isocitrate Dehydrogenase (IDH)
Fatty Acid Synthase
IL Receptor
IGF-1R
TGF-beta/Smad
ATM/ATR
MDM-2/p53
Anti-infection
CSF-1R
DNA gyrase
Nrf2
Complement System
HMG-CoA Reductase
BTK
ROR
Glutathione Peroxidase
PKA
Glucagon Receptor
P2X Receptor
Antifection
Molecular Glues
Guanylate cyclase
TLR
RSV
Ligand for E3 Ligase
Neurokinin receptor
CFTR
Antioxidant
DNA Alkylator/Crosslinker
Histone Demethylase
PERK
Serine/threonin kinase
FXR
ABC Transporter
Hedgehog/Smoothened
Vasopressin Receptor
Xanthine Oxidase
CaMK
Beta-Secretase
Hydroxylase
PLK
IRAK
FAK
NOD-like Receptor (NLR)
P2Y Receptor
LTR
Antifolate
Cysteine Protease
OX Receptor
Aminopeptidase
Casein Kinase
IκB/IKK
Aromatase
GHSR
HIF
DNA Methyltransferase
PD-1/PD-L1
YAP
GNRH Receptor
Pim
Aryl Hydrocarbon Receptor
IDO
IAP
Glucosidase
Smo
DNA Alkylation
Stearoyl-CoA Desaturase (SCD)
Chk
Indoleamine 2,3-Dioxygenase (IDO)
OXPHOS
Ephrin Receptor
transporter
ASK
Sigma receptor
ADC Cytotoxin
IKZF
Mdm2
NOS
DNA-PK
CRM1
Amino Acids and Derivatives
BACE
Lipase
Melatonin Receptor
MAGL
PAK
Thrombopoietin Receptor
Telomerase
Porcupine
Histone Acetyltransferase
PAI-1
NADPH-oxidase
p53
Monocarboxylate transporter
IFNAR
Cholecystokinin Receptor
FLAP
MT Receptor
GlyT
Monoamine Transporter
Neuropeptide Y Receptor
FAAH
DNA
DUB
PGE Synthase
Sirtuin
Neprilysin
GST
S6 Kinase
Protease-activated Receptor
AhR
MicroRNA
MTP
Tie-2
TOPK
CaSR
Glucokinase
Glutaminase
Annexin A
RIP kinase
UGT
PAFR
Hexokinase
Bradykinin Receptor
PAD
Epoxide Hydrolase
OAT
Free radical scavengers
FKBP
LPA Receptor
PI4K
Oxytocin Receptor
SGK
Discoidin Domain Receptor (DDR)
NOD
Melanin-concentrating Hormone Receptor (MCHR)
Advanced Glycation End Products
PROTACs
MALT
NEDD8
Ligands for Target Protein for PROTAC
Cell wall
Necroptosis
OCT
Galectin
c-Myc
Rho
Hck
Liver X Receptor
Neurotensin Receptor
Vitamin
LDLR
NR4A
SIK
IRE1
LDL
Na-K-Cl cotransporter
Integrase
Mucin
ATP Citrate Lyase
Lipid
BCRP
Survivin
MNK
STING
LRRK2
GPCR19
GluCls
Hippo pathway
Acetyl-CoA Carboxylase
PDK
Adenosine Deaminase
CGRP Receptor
Cuproptosis
Gap Junction Protein
Platelet aggregation
BMI-1
Tyrosinase
MLK
Imidazoline Receptor
Kinesin
Chloride channel
Taste receptor
GSNOR
NPC1L1
Hydrogenase
CD38
ASBT
Arginase
Na+/Ca2+ Exchanger
DYRK
MIF
GTPase
AAK1
ATG
NAMPT
PYK2
Immunology/Inflammation related
Prolyl Endopeptidase (PREP)
Myosin
Adiponectin Receptor
Haspin Kinase
GRK
PACAP
AAK1 (AP2 associated kinase 1)
Arp2/3 Complex
PROTAC Linker
HCN Channel
ACK1
PTEN
Somatostatin
cAMP
glycosidase
Wee1
Glutathione reductase
Decarboxylase
Pyroptosis
Methionine Adenosyltransferase (MAT)
p62
GPX
Melanocortin Receptor
CRISPR/Cas9
FOXO
RXFP receptor
DAPK
p97
PKM
Ferroportin
Sodium-dependent phosphate transporter

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