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TargetMol | Compound Library

Orally Active Compound Library

Catalog No. L9850

Oral administration is the first choice for clinical drug delivery, especially for long-term use. It is also the safest, most convenient, and most economical method of drug delivery. Oral bioavailability is the percentage of the absorbed drug dose successfully passed through the mucosa of the gastrointestinal tract and entered the bloodstream through the liver, to the original given oral dose. Drugs with high oral bioavailability can achieve efficacy at lower doses and effectively reduce toxic side effects; while when bioavailability is too low, even compounds with good pharmacological activity are unable to be fully exposed and utilized at the target site, resulting in therapeutic failure or high dose with large toxic side effects, which eventually leads to drug development failure and limits the application. TargetMol has carefully collected 2427 compounds with publicly reported oral activity that can be used for drug repurposing and development of orally active drugs.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L9850

Orally Active Compound Library
sizeIn stock
  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 2427 of orally active compounds for high-throughput screening and high-content screening.
  • Some drugs are approved or are in clinical trials with validated biological activity and safety.
  • Detailed specifications, compound structures, target information, activity descriptions, etc.
  • NMR and HPLC detection techniques to ensure high product purity.
  • All compounds are available in stock.

Packaging And Storage | TargetMol Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

Library Customization | TargetMol Library Customization

Compound Library | TargetMol
Targetmol Compound Libraries
can be highly customized!
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Library Customization | TargetMol Library Composition

Autophagy
Apoptosis
Antibacterial
Antibiotic
5-HT Receptor
Endogenous Metabolite
Adrenergic Receptor
Dopamine Receptor
Histamine Receptor
COX
Parasite
HIV Protease
VEGFR
AChR
DNA/RNA Synthesis
Potassium Channel
Sodium Channel
EGFR
PDGFR
P450
Estrogen/progestogen Receptor
Calcium Channel
Glucocorticoid Receptor
c-Kit
SARS-CoV
FLT
PDE
Antifungal
CDK
Dehydrogenase
Ferroptosis
PI3K
JAK
RAAS
Reactive Oxygen Species
FGFR
HCV Protease
Topoisomerase
Src
c-Met/HGFR
Mitophagy
NF-κB
Reverse Transcriptase
PPAR
Influenza Virus
Proteasome
Estrogen Receptor/ERR
Serotonin Transporter
BTK
Bcr-Abl
HBV
mTOR
HDAC
GPR
GABA Receptor
Androgen Receptor
Prostaglandin Receptor
Microtubule Associated
p38 MAPK
TRP/TRPV Channel
Histone Methyltransferase
Phosphatase
Adenosine Receptor
PARP
Raf
Tyrosine Kinases
GluR
Progesterone Receptor
ROS
HSV
Epigenetic Reader Domain
Nucleoside Antimetabolite/Analog
Opioid Receptor
DPP-4
AChE
ribosome
MEK
TNF
ALK
HIF/HIF Prolyl-Hydroxylase
iGluR
Norepinephrine
Trk receptor
HER
Proton pump
Virus Protease
ERK
LPL Receptor
Transferase
P-gp
SGLT
MAPK
Beta Amyloid
c-RET
TAM Receptor
S1P Receptor
ROCK
c-Fms
STAT
Thrombin
MAO
MRP
MMP
Aurora Kinase
AMPK
Phospholipase
NADPH
Integrin
DNA gyrase
Interleukin
Akt
HSP
Endothelin Receptor
Retinoid Receptor
Syk
ATPase
Wnt/beta-catenin
Caspase
Mitochondrial Metabolism
PKC
CSF-1R
Gamma-secretase
Antifection
Guanylate cyclase
Fatty Acid Synthase
IL Receptor
CXCR
Acyltransferase
TLR
CCR
HMG-CoA Reductase
Ras
ROR
GSK-3
Thyroid hormone receptor(THR)
Factor Xa
E1/E2/E3 Enzyme
BCL
Lipoxygenase
IGF-1R
Complement System
Monoamine Oxidase
Carbonic Anhydrase
DHFR
DNA Alkylator/Crosslinker
ABC
Antifolate
NMDAR
Beta-Secretase
Antiviral
ATM/ATR
CFTR
NO Synthase
Nrf2
Ligand for E3 Ligase
Hydroxylase
PLK
HIF
Neurokinin receptor
ROS Kinase
P2Y Receptor
Reductase
Glutathione Peroxidase
Antioxidant
Smo
CaMK
TGF-beta/Smad
Hedgehog/Smoothened
Aminopeptidase
ASK
RSV
GHSR
FAK
BACE
Melatonin Receptor
LTR
Lipase
Serine Protease
Serine/threonin kinase
IAP
FXR
DNA Alkylation
Stearoyl-CoA Desaturase (SCD)
Isocitrate Dehydrogenase (IDH)
PAK
OX Receptor
Indoleamine 2,3-Dioxygenase (IDO)
Ephrin Receptor
IκB/IKK
Casein Kinase
Cannabinoid Receptor
DNA Methyltransferase
Sigma receptor
DNA-PK
Histone Demethylase
GNRH Receptor
PKA
Pim
Cysteine Protease
Leukotriene Receptor
Aryl Hydrocarbon Receptor
MT Receptor
P2X Receptor
Monoamine Transporter
Vasopressin Receptor
Xanthine Oxidase
PGE Synthase
transporter
IRAK
PAI-1
Aromatase
NADPH-oxidase
p53
CRM1
JNK
Mdm2
Amino Acids and Derivatives
IFNAR
PERK
CaSR
Glucokinase
Annexin A
RIP kinase
UGT
Liver X Receptor
FLAP
Drug Metabolite
Glucagon Receptor
Glucosidase
Neuropeptide Y Receptor
Chk
DNA
DUB
Free radical scavengers
Sirtuin
Molecular Glues
FAAH
PAD
Porcupine
Neprilysin
cholecystokinin
AhR
Discoidin Domain Receptor (DDR)
S6 Kinase
NOD-like Receptor (NLR)
PD-1/PD-L1
MALT
Tie-2
TOPK
advanced glycation end products
CAT
Ligands for Target Protein for PROTAC
CETP
IDO
LDL
Rho
Hck
Hexokinase
Thrombopoietin Receptor
OXPHOS
STING
LRRK2
Integrase
Telomerase
Lipid
MNK
Histone Acetyltransferase
GST
Acetyl-CoA Carboxylase
PI4K
PDK
CGRP Receptor
SGK
Protease-activated Receptor
Adenosine deaminase
Platelet aggregation
NOD
BMI-1
Tyrosinase
Imidazoline Receptor
Chloride channel
Taste receptor
NOS
Monocarboxylate transporter
DYRK
Cell wall
c-Myc
NPC1L1
Hydrogenase
NEDD8
Na+/Ca2+ Exchanger
PYK2
Prolyl Endopeptidase (PREP)
Myosin
IRE1
Adiponectin receptor
Neurotensin Receptor
NAMPT
Glutaminase
SIK
PAFR
Haspin Kinase
GRK
GlyT
Na-K-Cl cotransporter
Bradykinin Receptor
Angiotensin-converting Enzyme (ACE)
Somatostatin
cAMP
ATP Citrate Lyase
BCRP
Glutathione reductase
GPCR19
Decarboxylase
PROTAC Linker
Epoxide Hydrolase
ACK
Survivin
OAT
GluCls
Pyroptosis
Methionine Adenosyltransferase (MAT)
LPA Receptor
p97
MLK
PKM
GPX
CRISPR/Cas9
Gap Junction Protein
Anti-infection
Kinesin

Keywords