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TargetMol | Compound Library

Orally Active Compound Library

Catalog No. L9850

Oral administration is the first choice for clinical drug delivery, especially for long-term use. It is also the safest, most convenient, and most economical method of drug delivery. Oral bioavailability is the percentage of the absorbed drug dose successfully passed through the mucosa of the gastrointestinal tract and entered the bloodstream through the liver, to the original given oral dose. Drugs with high oral bioavailability can achieve efficacy at lower doses and effectively reduce toxic side effects; while when bioavailability is too low, even compounds with good pharmacological activity are unable to be fully exposed and utilized at the target site, resulting in therapeutic failure or high dose with large toxic side effects, which eventually leads to drug development failure and limits the application. TargetMol has carefully collected 3160 compounds with publicly reported oral activity that can be used for drug repurposing and development of orally active drugs.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L9850

Orally Active Compound Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 3160 of orally active compounds for high-throughput screening and high-content screening.
  • Some drugs are approved or are in clinical trials with validated biological activity and safety.
  • Detailed specifications, compound structures, target information, activity descriptions, etc.
  • NMR and HPLC detection techniques to ensure high product purity.
  • All compounds are available in stock.

Packaging And Storage Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
  • This compound library is provided at a concentration of 10 mM in DMSO. A small number of compounds may be provided in different solvents or concentrations due to solubility or stability requirements. Please refer to the specific product information for details.

Packaging And Storage | TargetMol Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

Library Customization | TargetMol Library Customization

Compound Library | TargetMol
Targetmol Compound Libraries
can be highly customized!
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Library Customization | TargetMol Library Composition

Autophagy
Apoptosis
Antibacterial
Antibiotic
5-HT Receptor
Endogenous Metabolite
Adrenergic Receptor
Histamine Receptor
Dopamine Receptor
COX
AChR
HIV Protease
Parasite
VEGFR
DNA/RNA Synthesis
Potassium Channel
EGFR
Sodium Channel
PDE
Calcium Channel
SARS-CoV
CDK
Cytochromes P450
PDGFR
Estrogen/progestogen Receptor
FLT
Glucocorticoid Receptor
Dehydrogenase
c-Kit
RAAS
PI3K
Antifungal
Estrogen Receptor/ERR
HCV Protease
Ferroptosis
JAK
Topoisomerase
Src
FGFR
Reactive Oxygen Species
Microtubule Associated
Mitophagy
PPAR
HDAC
Bcr-Abl
c-Met/HGFR
GABA Receptor
NF-κB
GluR
HBV
p38 MAPK
Proteasome
Reverse Transcriptase
Serotonin Transporter
TRP/TRPV Channel
Influenza Virus
Prostaglandin Receptor
Androgen Receptor
Epigenetic Reader Domain
GPCR
iGluR
Histone Methyltransferase
Norepinephrine
ALK
Raf
mTOR
Phosphatase
Tyrosine Kinases
Adenosine Receptor
Cholinesterase (ChE)
Progesterone Receptor
PARP
Integrin
ROS
TNF
Antiviral
DPP-4
HSV
MMP
ribosome
Transferase
Beta Amyloid
ERK
GSK-3
HER
HIF/HIF Prolyl-Hydroxylase
MAPK
Nucleoside Antimetabolite/Analog
Opioid Receptor
S1P Receptor
Akt
LPL Receptor
MEK
NMDAR
P-gp
Proton pump
Thrombin
Trk receptor
c-Fms
c-RET
HSP
STAT
Syk
Virus Protease
Aurora Kinase
Endothelin Receptor
Factor Xa
Mitochondrial Metabolism
Monoamine Oxidase
Retinoid Receptor
ROCK
SGLT
TAM Receptor
Cannabinoid Receptor
Carbonic Anhydrase
CCR
CXCR
Lipoxygenase
MAO
MRP
Phospholipase
Reductase
Acyltransferase
AMPK
ATM/ATR
ATPase
DHFR
Fatty Acid Synthase
IL Receptor
Interleukin
PKC
ROS Kinase
Thyroid hormone receptor(THR)
Wnt/beta-catenin
CSF-1R
Gamma-secretase
HMG-CoA Reductase
NADPH
BTK
Caspase
CFTR
DNA gyrase
E1/E2/E3 Enzyme
Glucagon Receptor
Guanylate cyclase
IGF-1R
Ligand for E3 Ligase
Neurokinin receptor
NO Synthase
P2X Receptor
ROR
TGF-beta/Smad
TLR
ABC Transporter
Antifection
DNA Alkylator/Crosslinker
FAK
Glutathione Peroxidase
Hedgehog/Smoothened
Histone Demethylase
PKA
PLK
RSV
Vasopressin Receptor
Aminopeptidase
Antifolate
Antioxidant
Aromatase
Bcl-2 Family
Beta-Secretase
CaMK
Complement System
Cysteine Protease
DNA Methyltransferase
FXR
HIF
Hydroxylase
IRAK
Leukotriene Receptor
LTR
Nrf2
OX Receptor
P2Y Receptor
Serine/threonin kinase
Xanthine Oxidase
ASK
BACE
Casein Kinase
Chk
DNA Alkylation
GHSR
IAP
Indoleamine 2,3-Dioxygenase (IDO)
PD-1/PD-L1
PERK
Pim
Ras
Sigma receptor
Smo
transporter
Kras
Aryl Hydrocarbon Receptor
DNA-PK
Ephrin Receptor
GNRH Receptor
Isocitrate Dehydrogenase (IDH)
IκB/IKK
Mdm2
Melatonin Receptor
NADPH-oxidase
NOS
p53
PAK
Serine Protease
Stearoyl-CoA Desaturase (SCD)
YAP
ADC Cytotoxin
AhR
Cholecystokinin Receptor
CRM1
DNA
Drug Metabolite
DUB
FAAH
FLAP
Glucosidase
GlyT
Lipase
Molecular Glues
Monoamine Transporter
MT Receptor
Neprilysin
Neuropeptide Y Receptor
PAI-1
PGE Synthase
Porcupine
Protease-activated Receptor
Amino Acids and Derivatives
Annexin A
CaSR
CETP
CGRP Receptor
Discoidin Domain Receptor (DDR)
Epoxide Hydrolase
Free radical scavengers
Glucokinase
GST
Hexokinase
IFNAR
JNK
LPA Receptor
MicroRNA
Monocarboxylate transporter
NOD
NOD-like Receptor (NLR)
OXPHOS
Oxytocin Receptor
PAD
PI4K
RIP kinase
S6 Kinase
Sirtuin
Thrombopoietin Receptor
TOPK
UGT
Acetyl-CoA Carboxylase
Adenosine Deaminase
Advanced Glycation End Products
BMI-1
Bradykinin Receptor
Cell wall
Gap Junction Protein
GluCls
Glutaminase
Hck
Hippo pathway
Histone Acetyltransferase
IDO
Imidazoline Receptor
Integrase
IRE1
Kinesin
LDL
Ligands for Target Protein for PROTAC
Lipid
Liver X Receptor
LRRK2
MALT
Melanin-concentrating Hormone Receptor (MCHR)
MLK
MNK
Na-K-Cl cotransporter
NEDD8
OAT
PAFR
PDK
Platelet aggregation
PROTACs
Rho
SGK
SIK
STING
Telomerase
Tyrosinase
Vitamin
AAK1
ACK1
Adiponectin Receptor
Angiotensin-converting Enzyme (ACE)
Anti-infection
Arginase
ATP Citrate Lyase
BCRP
cAMP
CD38
Chloride channel
c-Myc
CRISPR/Cas9
Decarboxylase
DYRK
FOXO1
Galectin
Glutathione reductase
GPCR19
GPX
GRK
GSNOR
GTPase
Haspin Kinase
HCN Channel
Hydrogenase
Melanocortin Receptor
Methionine Adenosyltransferase (MAT)
Mucin
Myosin
Na+/Ca2+ Exchanger
NAMPT
Necroptosis
Neurotensin Receptor
NPC1L1
OCT
p97
PACAP
PKM
Prolyl Endopeptidase (PREP)
PROTAC Linker
PTEN
PYK2
Pyroptosis
RXFP receptor
Somatostatin
Survivin
Taste receptor
Tie-2
Wee1
Sodium-dependent phosphate transporter

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