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TargetMol | Compound Library

Orally Active Compound Library

Catalog No. L9850

Oral administration is the first choice for clinical drug delivery, especially for long-term use. It is also the safest, most convenient, and most economical method of drug delivery. Oral bioavailability is the percentage of the absorbed drug dose successfully passed through the mucosa of the gastrointestinal tract and entered the bloodstream through the liver, to the original given oral dose. Drugs with high oral bioavailability can achieve efficacy at lower doses and effectively reduce toxic side effects; while when bioavailability is too low, even compounds with good pharmacological activity are unable to be fully exposed and utilized at the target site, resulting in therapeutic failure or high dose with large toxic side effects, which eventually leads to drug development failure and limits the application. TargetMol has carefully collected 3160 compounds with publicly reported oral activity that can be used for drug repurposing and development of orally active drugs.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L9850

Orally Active Compound Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 3160 of orally active compounds for high-throughput screening and high-content screening.
  • Some drugs are approved or are in clinical trials with validated biological activity and safety.
  • Detailed specifications, compound structures, target information, activity descriptions, etc.
  • NMR and HPLC detection techniques to ensure high product purity.
  • All compounds are available in stock.

Packaging And Storage | TargetMol Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

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Compound Library | TargetMol
Targetmol Compound Libraries
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Library Customization | TargetMol Library Composition

Autophagy
Apoptosis
Antibacterial
Antibiotic
5-HT Receptor
Endogenous Metabolite
Adrenergic Receptor
Histamine Receptor
Dopamine Receptor
COX
AChR
HIV Protease
Parasite
VEGFR
DNA/RNA Synthesis
Potassium Channel
EGFR
Sodium Channel
PDE
Calcium Channel
SARS-CoV
CDK
Cytochromes P450
Estrogen/progestogen Receptor
PDGFR
Glucocorticoid Receptor
FLT
Dehydrogenase
c-Kit
PI3K
RAAS
Estrogen Receptor/ERR
Antifungal
HCV Protease
Ferroptosis
Topoisomerase
JAK
Src
FGFR
Reactive Oxygen Species
Microtubule Associated
Mitophagy
PPAR
c-Met/HGFR
HBV
Bcr-Abl
Reverse Transcriptase
HDAC
NF-κB
Proteasome
p38 MAPK
Serotonin Transporter
TRP/TRPV Channel
GluR
GABA Receptor
Prostaglandin Receptor
Influenza Virus
GPCR
Epigenetic Reader Domain
Androgen Receptor
Histone Methyltransferase
Phosphatase
iGluR
Norepinephrine
Raf
ALK
Tyrosine Kinases
Cholinesterase (ChE)
mTOR
Adenosine Receptor
PARP
Progesterone Receptor
Integrin
ROS
TNF
Transferase
DPP-4
HSV
MMP
Antiviral
Proton pump
GSK-3
Nucleoside Antimetabolite/Analog
ERK
Opioid Receptor
MAPK
Beta Amyloid
ribosome
HIF/HIF Prolyl-Hydroxylase
S1P Receptor
HER
LPL Receptor
Akt
P-gp
Trk receptor
MEK
Thrombin
Virus Protease
NMDAR
HSP
STAT
c-Fms
c-RET
Syk
Monoamine Oxidase
Factor Xa
ROCK
MAO
Mitochondrial Metabolism
Endothelin Receptor
Aurora Kinase
SGLT
Retinoid Receptor
TAM Receptor
Carbonic Anhydrase
Reductase
MRP
CCR
CXCR
Lipoxygenase
Phospholipase
Cannabinoid Receptor
ATPase
DHFR
Wnt/beta-catenin
PKC
Fatty Acid Synthase
IL Receptor
Interleukin
Acyltransferase
ATM/ATR
AMPK
ROS Kinase
Thyroid hormone receptor(THR)
NADPH
CSF-1R
HMG-CoA Reductase
BTK
ROR
Antioxidant
Caspase
E1/E2/E3 Enzyme
Gamma-secretase
Glucagon Receptor
P2X Receptor
DNA gyrase
Guanylate cyclase
IGF-1R
TGF-beta/Smad
TLR
Ligand for E3 Ligase
Neurokinin receptor
CFTR
NO Synthase
Histone Demethylase
Glutathione Peroxidase
PKA
ABC Transporter
Antifection
Hedgehog/Smoothened
Vasopressin Receptor
Bcl-2 Family
RSV
PLK
FAK
DNA Alkylator/Crosslinker
P2Y Receptor
LTR
Antifolate
Serine/threonin kinase
Cysteine Protease
FXR
OX Receptor
Xanthine Oxidase
CaMK
Beta-Secretase
Aminopeptidase
Nrf2
Aromatase
Hydroxylase
HIF
Complement System
DNA Methyltransferase
IRAK
BACE
PERK
GNRH Receptor
Pim
Leukotriene Receptor
IAP
Smo
Chk
Indoleamine 2,3-Dioxygenase (IDO)
transporter
ASK
Casein Kinase
GHSR
Ras
Sigma receptor
PD-1/PD-L1
Kras
Mdm2
NOS
DNA-PK
YAP
Melatonin Receptor
Serine Protease
Aryl Hydrocarbon Receptor
Isocitrate Dehydrogenase (IDH)
DNA Alkylation
PAK
Stearoyl-CoA Desaturase (SCD)
Ephrin Receptor
IκB/IKK
NADPH-oxidase
p53
ADC Cytotoxin
CRM1
Lipase
Cholecystokinin Receptor
Drug Metabolite
MT Receptor
GlyT
Glucosidase
Monoamine Transporter
Molecular Glues
Neuropeptide Y Receptor
FAAH
DNA
DUB
PGE Synthase
Porcupine
PAI-1
Neprilysin
Protease-activated Receptor
AhR
MicroRNA
Monocarboxylate transporter
Amino Acids and Derivatives
IFNAR
CETP
JNK
TOPK
CaSR
Glucokinase
Annexin A
FLAP
RIP kinase
UGT
Hexokinase
PAD
Epoxide Hydrolase
Thrombopoietin Receptor
OXPHOS
Free radical scavengers
Sirtuin
GST
LPA Receptor
PI4K
Oxytocin Receptor
CGRP Receptor
Discoidin Domain Receptor (DDR)
NOD
S6 Kinase
NOD-like Receptor (NLR)
Melanin-concentrating Hormone Receptor (MCHR)
Advanced Glycation End Products
PROTACs
MALT
NEDD8
Ligands for Target Protein for PROTAC
Cell wall
Rho
Hck
Liver X Receptor
Glutaminase
IDO
SIK
IRE1
PAFR
LDL
Na-K-Cl cotransporter
Integrase
Bradykinin Receptor
Telomerase
Lipid
OAT
MNK
STING
LRRK2
Histone Acetyltransferase
GluCls
Hippo pathway
Acetyl-CoA Carboxylase
PDK
Adenosine Deaminase
SGK
Gap Junction Protein
Platelet aggregation
BMI-1
MLK
Imidazoline Receptor
Kinesin
Vitamin
Chloride channel
Taste receptor
GSNOR
NPC1L1
Hydrogenase
CD38
Arginase
Na+/Ca2+ Exchanger
DYRK
Necroptosis
Tie-2
GTPase
OCT
c-Myc
Galectin
AAK1
Neurotensin Receptor
NAMPT
PYK2
FOXO1
Prolyl Endopeptidase (PREP)
Myosin
Adiponectin Receptor
Haspin Kinase
GRK
PACAP
PROTAC Linker
HCN Channel
ACK1
Angiotensin-converting Enzyme (ACE)
PTEN
Somatostatin
cAMP
Mucin
Wee1
ATP Citrate Lyase
BCRP
Glutathione reductase
Survivin
GPCR19
Decarboxylase
Pyroptosis
Methionine Adenosyltransferase (MAT)
GPX
Melanocortin Receptor
CRISPR/Cas9
RXFP receptor
Anti-infection
Tyrosinase
p97
PKM
Sodium-dependent phosphate transporter

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