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TargetMol | Compound Library

Orally Active Compound Library

Catalog No. L9850

Oral administration is the first choice for clinical drug delivery, especially for long-term use. It is also the safest, most convenient, and most economical method of drug delivery. Oral bioavailability is the percentage of the absorbed drug dose successfully passed through the mucosa of the gastrointestinal tract and entered the bloodstream through the liver, to the original given oral dose. Drugs with high oral bioavailability can achieve efficacy at lower doses and effectively reduce toxic side effects; while when bioavailability is too low, even compounds with good pharmacological activity are unable to be fully exposed and utilized at the target site, resulting in therapeutic failure or high dose with large toxic side effects, which eventually leads to drug development failure and limits the application. TargetMol has carefully collected 3160 compounds with publicly reported oral activity that can be used for drug repurposing and development of orally active drugs.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L9850

Orally Active Compound Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 3160 of orally active compounds for high-throughput screening and high-content screening.
  • Some drugs are approved or are in clinical trials with validated biological activity and safety.
  • Detailed specifications, compound structures, target information, activity descriptions, etc.
  • NMR and HPLC detection techniques to ensure high product purity.
  • All compounds are available in stock.

Packaging And Storage | TargetMol Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

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Compound Library | TargetMol
Targetmol Compound Libraries
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Library Customization | TargetMol Library Composition

Autophagy
Apoptosis
Antibacterial
Antibiotic
5-HT Receptor
Endogenous Metabolite
Adrenergic Receptor
Histamine Receptor
Dopamine Receptor
COX
AChR
HIV Protease
Parasite
VEGFR
DNA/RNA Synthesis
EGFR
Potassium Channel
Sodium Channel
PDE
Calcium Channel
SARS-CoV
Estrogen/progestogen Receptor
Cytochromes P450
CDK
PDGFR
Glucocorticoid Receptor
FLT
Dehydrogenase
c-Kit
RAAS
PI3K
Estrogen Receptor/ERR
HCV Protease
Antifungal
Ferroptosis
Topoisomerase
JAK
Src
FGFR
Reactive Oxygen Species
Microtubule Associated
Mitophagy
PPAR
c-Met/HGFR
HBV
Bcr-Abl
Reverse Transcriptase
NF-κB
p38 MAPK
Serotonin Transporter
GluR
HDAC
GABA Receptor
Proteasome
TRP/TRPV Channel
Androgen Receptor
Prostaglandin Receptor
Influenza Virus
iGluR
Epigenetic Reader Domain
GPR
Histone Methyltransferase
Phosphatase
Norepinephrine
Raf
ALK
Adenosine Receptor
Tyrosine Kinases
Cholinesterase (ChE)
mTOR
Progesterone Receptor
PARP
HER
Integrin
ROS
MMP
TNF
Nucleoside Antimetabolite/Analog
Opioid Receptor
HSV
MAPK
ribosome
Transferase
GSK-3
ERK
DPP-4
Antiviral
HIF/HIF Prolyl-Hydroxylase
S1P Receptor
Proton pump
LPL Receptor
NMDAR
P-gp
Trk receptor
Beta Amyloid
Thrombin
Factor Xa
Virus Protease
Akt
Retinoid Receptor
STAT
c-Fms
c-RET
MEK
Syk
Monoamine Oxidase
ROCK
MAO
Mitochondrial Metabolism
Endothelin Receptor
Aurora Kinase
Lipoxygenase
SGLT
Carbonic Anhydrase
Reductase
MRP
CCR
CXCR
HSP
Phospholipase
Cannabinoid Receptor
TAM Receptor
Thyroid hormone receptor(THR)
ATPase
DHFR
Wnt/beta-catenin
Fatty Acid Synthase
IL Receptor
Interleukin
Acyltransferase
AMPK
ROS Kinase
NADPH
PKC
CSF-1R
Gamma-secretase
DNA gyrase
ATM/ATR
HMG-CoA Reductase
BTK
ROR
Caspase
E1/E2/E3 Enzyme
P2X Receptor
Guanylate cyclase
IGF-1R
TGF-beta/Smad
TLR
Ligand for E3 Ligase
Neurokinin receptor
CFTR
NO Synthase
Antioxidant
Histone Demethylase
Glutathione Peroxidase
PKA
Glucagon Receptor
ABC Transporter
Antifection
Hedgehog/Smoothened
Bcl-2 Family
RSV
PLK
FAK
P2Y Receptor
LTR
Antifolate
Serine/threonin kinase
Cysteine Protease
FXR
Leukotriene Receptor
Vasopressin Receptor
OX Receptor
Xanthine Oxidase
CaMK
Beta-Secretase
Aminopeptidase
Nrf2
Aromatase
Hydroxylase
HIF
Complement System
IRAK
Sigma receptor
Mdm2
DNA Alkylator/Crosslinker
BACE
PERK
GNRH Receptor
Pim
IAP
Smo
Indoleamine 2,3-Dioxygenase (IDO)
transporter
ASK
Casein Kinase
GHSR
DNA Methyltransferase
Ras
PD-1/PD-L1
Kras
NOS
DNA-PK
YAP
Lipase
Melatonin Receptor
Serine Protease
Aryl Hydrocarbon Receptor
Isocitrate Dehydrogenase (IDH)
DNA Alkylation
PAK
Stearoyl-CoA Desaturase (SCD)
Chk
Ephrin Receptor
IκB/IKK
NADPH-oxidase
p53
ADC Cytotoxin
CRM1
Cholecystokinin Receptor
Drug Metabolite
MT Receptor
Glucosidase
Monoamine Transporter
Molecular Glues
Neuropeptide Y Receptor
FAAH
DNA
DUB
PGE Synthase
Porcupine
PAI-1
Neprilysin
MicroRNA
Monocarboxylate transporter
Amino Acids and Derivatives
IFNAR
CETP
JNK
CaSR
Liver X Receptor
Glucokinase
Annexin A
FLAP
RIP kinase
UGT
GlyT
Hexokinase
PAD
Epoxide Hydrolase
Thrombopoietin Receptor
OXPHOS
Free radical scavengers
Sirtuin
GST
LPA Receptor
PI4K
Oxytocin Receptor
CGRP Receptor
Discoidin Domain Receptor (DDR)
NOD
S6 Kinase
Protease-activated Receptor
AhR
NOD-like Receptor (NLR)
Melanin-concentrating Hormone Receptor (MCHR)
Advanced Glycation End Products
PROTACs
MALT
NEDD8
Ligands for Target Protein for PROTAC
Cell wall
Tie-2
TOPK
Rho
Hck
Glutaminase
IDO
SIK
IRE1
PAFR
LDL
Na-K-Cl cotransporter
Integrase
Bradykinin Receptor
Telomerase
Lipid
OAT
MNK
STING
LRRK2
Histone Acetyltransferase
GluCls
Hippo pathway
Acetyl-CoA Carboxylase
PDK
Adenosine Deaminase
SGK
Gap Junction Protein
Platelet aggregation
BMI-1
Tyrosinase
MLK
Imidazoline Receptor
Kinesin
Vitamin
Chloride channel
Taste receptor
GSNOR
NPC1L1
Hydrogenase
CD38
Arginase
Na+/Ca2+ Exchanger
DYRK
Necroptosis
GTPase
OCT
c-Myc
Galectin
AAK1
Neurotensin Receptor
PYK2
NAMPT
FOXO1
Prolyl Endopeptidase (PREP)
Myosin
Adiponectin Receptor
Haspin Kinase
GRK
PACAP
PROTAC Linker
HCN Channel
ACK1
Angiotensin-converting Enzyme (ACE)
Somatostatin
cAMP
Mucin
Wee1
ATP Citrate Lyase
BCRP
Glutathione reductase
Survivin
GPCR19
Decarboxylase
Pyroptosis
Methionine Adenosyltransferase (MAT)
GPX
Melanocortin Receptor
CRISPR/Cas9
RXFP receptor
Anti-infection
p97
PKM
Sodium-dependent phosphate transporter

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