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TargetMol | Compound Library

Orally Active Compound Library

Catalog No. L9850

Oral administration is the first choice for clinical drug delivery, especially for long-term use. It is also the safest, most convenient, and most economical method of drug delivery. Oral bioavailability is the percentage of the absorbed drug dose successfully passed through the mucosa of the gastrointestinal tract and entered the bloodstream through the liver, to the original given oral dose. Drugs with high oral bioavailability can achieve efficacy at lower doses and effectively reduce toxic side effects; while when bioavailability is too low, even compounds with good pharmacological activity are unable to be fully exposed and utilized at the target site, resulting in therapeutic failure or high dose with large toxic side effects, which eventually leads to drug development failure and limits the application. TargetMol has carefully collected 3160 compounds with publicly reported oral activity that can be used for drug repurposing and development of orally active drugs.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L9850

Orally Active Compound Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 3160 of orally active compounds for high-throughput screening and high-content screening.
  • Some drugs are approved or are in clinical trials with validated biological activity and safety.
  • Detailed specifications, compound structures, target information, activity descriptions, etc.
  • NMR and HPLC detection techniques to ensure high product purity.
  • All compounds are available in stock.

Packaging And Storage Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
  • This compound library is provided at a concentration of 10 mM in DMSO. A small number of compounds may be provided in different solvents or concentrations due to solubility or stability requirements. Please refer to the specific product information for details.

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Apoptosis
Autophagy
Antibacterial
Antibiotic
Endogenous Metabolite
5-HT Receptor
Adrenergic Receptor
Dopamine Receptor
Histamine Receptor
Parasite
COX
AChR
DNA/RNA Synthesis
HIV Protease
Potassium Channel
VEGFR
EGFR
Calcium Channel
Cytochromes P450
Sodium Channel
SARS-CoV
PDE
CDK
PDGFR
Estrogen/progestogen Receptor
Reactive Oxygen Species
Glucocorticoid Receptor
FLT
Dehydrogenase
c-Kit
Virus Protease
p38 MAPK
RAAS
Estrogen Receptor/ERR
PI3K
NF-κB
Ferroptosis
HCV Protease
Antifungal
Topoisomerase
JAK
Mitophagy
Ras
Src
FGFR
Microtubule Associated
HBV
iGluR
Influenza Virus
c-Met/HGFR
PPAR
Serotonin Transporter
Reverse Transcriptase
HDAC
Bcr-Abl
GABA Receptor
TRP/TRPV Channel
Prostaglandin Receptor
GPCR
Proteasome
GluR
Androgen Receptor
Akt
Phosphatase
Epigenetic Reader Domain
mTOR
TNF
Histone Methyltransferase
ERK
Raf
Norepinephrine
LPL Receptor
Interleukin
ALK
Progesterone Receptor
Tyrosine Kinases
Nucleoside Antimetabolite/Analog
MMP
Adenosine Receptor
PARP
Cholinesterase (ChE)
HSV
MAPK
Beta Amyloid
Monoamine Oxidase
Transferase
Caspase
Mitochondrial Metabolism
ROS
Angiotensin-converting Enzyme (ACE)
P-gp
HSP
STAT
Integrin
GSK-3
Opioid Receptor
DPP-4
Antiviral
c-Fms
ribosome
HIF/HIF Prolyl-Hydroxylase
Kras
Proton pump
Bcl-2 Family
NO Synthase
S1P Receptor
HER
Factor Xa
NMDAR
Trk receptor
MEK
Thrombin
Leukotriene Receptor
ROCK
Aurora Kinase
Lipoxygenase
Retinoid Receptor
c-RET
Syk
PKC
MAO
Drug Metabolite
Endothelin Receptor
SGLT
Phospholipase
TAM Receptor
ROS Kinase
ATPase
Carbonic Anhydrase
MRP
Wnt/beta-catenin
Gamma-secretase
CCR
CXCR
Acyltransferase
AMPK
Cannabinoid Receptor
Thyroid hormone receptor(THR)
DHFR
Reductase
NADPH
Serine Protease
E1/E2/E3 Enzyme
Isocitrate Dehydrogenase (IDH)
Fatty Acid Synthase
IL Receptor
IGF-1R
TGF-beta/Smad
ATM/ATR
MDM-2/p53
Anti-infection
JNK
CSF-1R
DNA gyrase
Nrf2
Complement System
HMG-CoA Reductase
BTK
ROR
Glutathione Peroxidase
PKA
Glucagon Receptor
P2X Receptor
Antifection
Molecular Glues
Guanylate cyclase
TLR
RSV
Ligand for E3 Ligase
Neurokinin receptor
CFTR
Antioxidant
DNA Alkylator/Crosslinker
Histone Demethylase
PERK
Serine/threonin kinase
FXR
ABC Transporter
Hedgehog/Smoothened
Vasopressin Receptor
Xanthine Oxidase
CaMK
Beta-Secretase
Hydroxylase
PLK
IRAK
FAK
P2Y Receptor
LTR
Antifolate
OX Receptor
Aminopeptidase
Casein Kinase
IκB/IKK
Aromatase
GHSR
HIF
DNA Methyltransferase
NOD-like Receptor (NLR)
PD-1/PD-L1
YAP
GNRH Receptor
Pim
Cysteine Protease
Aryl Hydrocarbon Receptor
IDO
IAP
Glucosidase
Smo
DNA Alkylation
Stearoyl-CoA Desaturase (SCD)
Chk
Indoleamine 2,3-Dioxygenase (IDO)
OXPHOS
transporter
ASK
Sigma receptor
ADC Cytotoxin
IKZF
Mdm2
NOS
DNA-PK
CRM1
Amino Acids and Derivatives
BACE
Lipase
Melatonin Receptor
MAGL
PAK
Thrombopoietin Receptor
Telomerase
Porcupine
Ephrin Receptor
Histone Acetyltransferase
PAI-1
NADPH-oxidase
p53
Monocarboxylate transporter
IFNAR
Cholecystokinin Receptor
FLAP
MT Receptor
GlyT
Monoamine Transporter
Neuropeptide Y Receptor
FAAH
DNA
DUB
PGE Synthase
Sirtuin
Neprilysin
GST
Oxytocin Receptor
S6 Kinase
Protease-activated Receptor
AhR
MicroRNA
MTP
Tie-2
TOPK
CaSR
Glucokinase
Glutaminase
Annexin A
RIP kinase
UGT
PAFR
Hexokinase
Bradykinin Receptor
PAD
Epoxide Hydrolase
OAT
Free radical scavengers
FKBP
LPA Receptor
PI4K
SGK
Discoidin Domain Receptor (DDR)
NOD
Melanin-concentrating Hormone Receptor (MCHR)
Advanced Glycation End Products
PROTACs
MALT
NEDD8
Ligands for Target Protein for PROTAC
Cell wall
Necroptosis
OCT
c-Myc
Galectin
Rho
Hck
Liver X Receptor
Neurotensin Receptor
Vitamin
LDLR
NR4A
SIK
IRE1
LDL
Na-K-Cl cotransporter
Integrase
Mucin
ATP Citrate Lyase
Lipid
BCRP
MNK
Survivin
STING
LRRK2
GPCR19
GluCls
Hippo pathway
Acetyl-CoA Carboxylase
PDK
Adenosine Deaminase
CGRP Receptor
Cuproptosis
Gap Junction Protein
Platelet aggregation
BMI-1
Tyrosinase
MLK
Imidazoline Receptor
Kinesin
Chloride channel
Taste receptor
GSNOR
NPC1L1
Hydrogenase
CD38
ASBT
Arginase
Na+/Ca2+ Exchanger
DYRK
MIF
GTPase
AAK1
ATG
NAMPT
PYK2
Immunology/Inflammation related
Prolyl Endopeptidase (PREP)
Myosin
Adiponectin Receptor
Haspin Kinase
GRK
PACAP
AAK1 (AP2 associated kinase 1)
Arp2/3 Complex
PROTAC Linker
HCN Channel
ACK1
PTEN
Somatostatin
cAMP
Wee1
Glutathione reductase
Decarboxylase
Pyroptosis
Methionine Adenosyltransferase (MAT)
p62
GPX
Melanocortin Receptor
CRISPR/Cas9
FOXO
RXFP receptor
DAPK
p97
PKM
Ferroportin
Sodium-dependent phosphate transporter

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