Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Firazorexton hydrate (TAK-994) is a brain-penetrant and orally active agonist of the orexin type 2 receptor (OX2R) with a potent EC50 of 19 nM. It effectively reduces wakefulness fragmentation and cataplexy-like episodes in mouse models of narcolepsy [1].
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Description | Firazorexton hydrate (TAK-994) is a brain-penetrant and orally active agonist of the orexin type 2 receptor (OX2R) with a potent EC50 of 19 nM. It effectively reduces wakefulness fragmentation and cataplexy-like episodes in mouse models of narcolepsy [1]. |
Synonyms | TAK-994 |
Molecular Weight | 497.53 |
Formula | C22H25F3N2O4S.3/2H2O |
CAS No. | 2861934-86-1 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
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Firazorexton hydrate 2861934-86-1 TAK-994 inhibitor inhibit