Search Result

Search Results for " mer "

Targets

Libraries

Traditional Chinese Medicine Monomer Library Anti-Alzheimer's Disease Compound Library Anti-virus Traditional Chinese Medicine Monomer Library

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Compounds

Cat No.	Product Name
T38936	KRAS G13D peptide, 25 mer
	KRAS G13D peptide, a 25-mer sequence, is derived from the KRAS activating oncogene mutation and serves as an immune pote...
T72574	Axl/Mer/CSF1R-IN-1
	Axl/Mer-IN-1 is an Axl/Mer receptor tyrosine kinase ( Axl/Mer RTK ) and CSF1R inhibitor with K d s of <0.1 μM .
T26296	Triparanol	NSC-65345,NSC 65345,NSC65345,MER-29	Apoptosis , Hedgehog/Smoothened
	Triparanol interferes with posttranslational modification of Hedgehog signaling molecules as well as the sterol sensing ...		Apoptosis , Hedgehog/Smoothened
T0318	Azacyclonol	MER 17,γ-pipradol,MDL 4829,Ataractan	5-HT Receptor
	Azacyclonol is a drug used to diminish hallucinations in psychotic individuals.		5-HT Receptor
T13074	TAM-IN-2		TAM Receptor
	TAM-IN-2 is an inhibitor of TAM.		TAM Receptor
T1968	UNC2250		TAM Receptor
	UNC2250 is an effective and specific Mer inhibitor (IC50=1.7 nM).		TAM Receptor
T2311	LDC1267		TAM Receptor
	LDC1267 is a excellently specific TAM(Tyro3, Axl and Mer) kinase inhibitor, for Mer( IC50<5 nM), Tyro3(IC50=8 nM), and A...		TAM Receptor
T17205	UNC2541		Others , FLT , TAM Receptor
	UNC2541 is a potent and Mer tyrosine kinase (MerTK)-specific inhibitor. It also binds in the MerTK ATP pocket (IC50: 4.4...		Others , FLT , TAM Receptor
T6982	SGI-7079		Src , c-RET , c-Met/HGFR , FLT , TAM Receptor
	SGI-7079 is a new selective Axl inhibitor. SGI-7079 can be a dose-dependent manner inhibited growth of tumors. It is als...		Src , c-RET , c-Met/HGFR , FLT , TAM Receptor
T2005	Dubermatinib	TP0903	TAM Receptor , Apoptosis
	TP-0903 is a potent and selective Axl kinase inhibitor.		TAM Receptor , Apoptosis
T6907	NPS-1034	NPS 1034,NPS1034	Apoptosis , TAM Receptor , c-Met/HGFR
	NPS-1034 is a dual Met/Axl inhibitor with IC50 of 48 nM and 10.3 nM, respectively.		Apoptosis , TAM Receptor , c-Met/HGFR
T70265	AL-6556
	AL-6556 is a prostaglandin DP receptor agonist.
T6269	Bemcentinib	BGB324,R428	TAM Receptor
	R428 is a selective inhibitor of Axl (IC50: 14 nM) and has been investigated for the treatment of NSCLC.		TAM Receptor
T2629	UNC2881		TAM Receptor
	UNC2881 is a specific Mer tyrosine kinase inhibitor (IC50: 4.3 nM). It is about 83- and 58-fold higher selectivity than ...		TAM Receptor
T7425	RU-301		TAM Receptor
	RU-301 is a novel pan-tam inhibitor		TAM Receptor
TQ0041	Ningetinib Tosylate		c-Met/HGFR , TAM Receptor , VEGFR
	Ningetinib Tosylate is an orally bioavailable tyrosine kinase inhibitor with IC50s of <1.0, 1.9 and 6.7 nM for Axl, VEGF...		c-Met/HGFR , TAM Receptor , VEGFR
T4426	CEP-40783	RXDX-106,CEP 40783	c-Met/HGFR , TAM Receptor
	CEP-40783 is an effective, specific and orally active AXL/c-Met inhibitor (IC50: 7/12 nM). It also inhibits MER and TYRO...		c-Met/HGFR , TAM Receptor
T21302	UNC569	UNC 569	TAM Receptor
	Lesinurad is a selective inhibitor of URAT1, a transporter in the kidney that regulates uric acid excretion from the bod...		TAM Receptor
T2699	BMS 777607	BMS777607,BMS-777607,BMS 817378	TAM Receptor , c-Met/HGFR
	BMS-777607 is a Met-related inhibitor for c-Met/Axl/Ron/Tyro3 (IC50: 3.9/1.1/1.8/4.3 nM). BMS-777607 has been investigat...		TAM Receptor , c-Met/HGFR
TQ0021	Ningetinib	CT053PTSA,CT-053	VEGFR , TAM Receptor , c-Met/HGFR
	Ningetinib (CT053PTSA) is an orally bioavailable tyrosine kinase inhibitor with IC50s of <1.0, 1.9 and 6.7 nM for Axl, V...		VEGFR , TAM Receptor , c-Met/HGFR