hγ1

Prostaglandin H1 is the cyclooxygenase metabolite of DGLA, a CRTh2 agonist and a precursor of a family of 1 anti-inflammatory prostaglandins. Prostaglandin H1 can be used in the study of inflammation.

H1-7 (histone H1 phosphorylation site), a synthetic polypeptide, serves as a PKA substrate and demonstrates utility in various PKA substrate applications [1] [2].

Maximin H1, an antimicrobial peptide sourced from the skin secretions of the Chinese red belly toad (Bombina maxima), exhibits efficacy against several pathogens, including Escherichia coli (ATCC25922), Staphylococcus aureus (ATCC2592), Bacillus pyocyaneus (CMCCB1010), and Candida albicans (ATCC2002). Corresponding minimum inhibitory concentration (MIC) values are 9, 4.5, 9, and 4.5 μg/ml, respectively [1].

Bombinin H1, an antimicrobial peptide originating from the skin of the Bombina variegata moth, exhibits lethal concentrations of 3.8 μM against Escherichia coli D21 and 2.1 μM against Staphylococcus aureus Cowan 1 [1].

Anti-Canine PD-L1/B7-H1 Antibody (JC071) is an IgG1, κ antibody inhibitor derived from mice, targeting canine PD-L1/B7-H1.

Anti-Mouse PD-L1/B7-H1 (LALA-PG) Antibody (10F.9G2) is an IgG2a, κ antibody inhibitor derived from mice, specifically targeting and inhibiting mouse PD-L1/B7-H1.

Anti-Mouse PD-L1/B7-H1 Antibody (10F.9G2-Mouse IgG1) is an IgG1, κ inhibitory antibody derived from mice, designed to target mouse PD-L1/B7-H1.

Anti-Mouse PD-L1/B7-H1 (D265A) Antibody (10F.9G2) is an IgG1, κ inhibitor antibody derived from mice, specifically targeting and inhibiting mouse PD-L1/B7-H1.

Monamycin H1 is an ester peptide antibiotic that exhibits activity against Gram-positive bacteria.

Asperosaponin H1 is a high-purity biochemical reagent suitable for biochemical experiments and drug synthesis research.

Cimicifugoside H1 shows the protective function to cerebral neuron during cerebral ischemia.

(±)-Tazifylline is a selective and long-acting antagonist of histamine H1 receptor. Tazifylline shows much lower affinity for H2 receptors, α- and β-adrenoceptors, 5-hydroxytryptamine and muscarinic receptor subtypes.

Wy 49051 is an orally active antagonist of H1 receptor(IC50 of 44 nM).

Bamirastine inhibits ligand binding to recombinant human histamine H1 receptor (rhH1R) with an IC50 of 17.3 nM and possesses an inhibitory effect on allergic skin inflammation.

Rocastine (AHR-11325) is a selective and potent non-sedating H1 receptor antagonist.

Oxatomide (Oxatomida) is a potent and orally active dual H1 histamine receptor and P2X7 receptor antagonist with antihistamine and antiallergic activity.Oxatomide can be used to block ATP-induced currents in the human P2X7 receptor with an IC50 value of 0.95 μM.Oxatomide has an inhibitory effect on ATP-induced Ca2+ inward currents with an IC50 value of 0.43 μM.Oxatomide inhibits 5-hydroxytryptamine. Oxatomide inhibits 5-hydroxytryptamine with an IC50 of 0.43 μM.Oxatomide is used in the treatment of immune system diseases and in the study of hypersensitivity reactions.

Tecastemizole (R 43512) is a selective antagonist of H1 receptor and a major metabolite of astemizole with anti-inflammatory effects.

DF-1111301 is a novel anti-allergic compound with anti-histamine H1 and anti-PAF activity.

ReN-1869 is a novel selective histamine H(1) receptor antagonist with anti-neurogenic pain and anti-inflammatory activity for the study of neurological diseases.

Vapitadine dihydrochloride(R-129160 2HCl) is a novel, potent, selective and non-sedating compound with inhibitory effects on histamine H1.

Dimethindene (Dimetindeno) is a selective antagonist of H1 receptor and blocks K+ current. Dimethindene exhibits antihistamine and anticholinergic effects.

H1k is an eudistomin Y fluorescent derivative and lysosome-targeted antiproliferative agent that dose-dependently increases autophagy signalling and down-regulates the expression of cyclin-dependent kinase (CDK1) and cyclin B1.

Fenclozine Maleate (S 1429) is a potential histamine H1 receptor antagonist , which can be used to study fever, inflammation and pain.

(2R)-6-Methoxynaringenin is one of the potentially active components in Scutellaria baicalensis.