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Compounds

Cat No. Product Name
T12316 Oral antiplatelet agent 1 Others
Oral antiplatelet agent 1 is a potent antiplatelet agent with an IC50 of 2.94 μM in vitro.
T20764 Dienestrol diacetate NSC81279,Cycladiene,Retalon-oral,NSC-81279,NSC 81279,Oestrasid C
Dienestrol diacetate, a derivative of the synthetic non-steroid phenolic compound, DIENESTROL, exhibits estrogenic activ...
T14358 Avoralstat BCX4161 Others
Avoralstat 是血浆激肽释放酶(PKK)抑制剂,具有口服活性,可用于遗传性血管性水肿的研究。
TN1148 Isopsoralenoside Antibacterial , Estrogen Receptor/ERR , Estrogen/progestogen Receptor
Isopsoralenoside 是补骨脂多糖中的一种苯并呋喃苷。它在消化道内容物中可迅速代谢为补骨脂素。它具有雌激素样活性、促进成骨细胞增殖活性、抗肿瘤活性和抗菌活性。
TN1008 Psoralenoside Calcium Channel , CaMK , Histamine Receptor
Psoralenoside 是源于补骨脂中的苯并呋喃苷,具有抗肿瘤、抗菌、促进成骨细胞增殖和雌激素样活性。它对组胺 H1、钙调素和电压门控 l 型钙通道具有较高的亲和力。
T3399 Psoralidin Reactive Oxygen Species , Antibacterial , Others , Akt , Gamma-secretase , COX , Estrogen/progestogen Receptor , Lipoxygenase
Psoralidin 是COX-2和5-LOX 的抑制剂,有抗癌,抗菌和抗炎作用。它显著下调NOTCH1信号传导,还极大地诱导活化氧产生。
T1251 Dicloralurea DCU,Dichlorolurea,双(三氯乙醛基)脲,双 (三氯乙醛基) 脲 Others
DCU 是一种兽用的食品添加剂,可用作生长刺激剂。
TN1343 8-Geranyloxypsoralen 8-香叶草氧基补骨脂素 P450 , Anti-infection , BACE
8-Geranyloxypsoralen 是一种呋喃香豆素,分离自葡萄柚,是 P450 3A4 的有效抑制剂(IC50:3.93 μM)。
T31011 Coralyne chloride Topoisomerase
Coralyne chloride 是一种具有强抗癌活性的原小檗碱化合物。它可用于制备 Coralyne 衍生物,是一种基于荧光 DNA 的分子整流剂,通过位点特异性插入构建成 DNA 双链体。它可作为一种拓扑异构酶 I 毒性分子,诱导拓扑...
T2942 Psoralen 补骨脂素,psoralene,Furocoumarin,Ficusin HIV Protease , Apoptosis , Influenza Virus , DNA/RNA Synthesis
Psoralen 是从补骨脂种子中提取的一种香豆素。它具有如抗癌、抗氧化、抗抑郁、抗癌、抗菌、抗病毒等多种生物学特性。
TN6298 8-[(6,7-Dihydroxy-3,7-dimethyloct-2-en-1-yl)oxy]psoralen
T40859 5-Hydroxy-8-methoxypsoralen 5-Hydroxy-8-methoxypsoralen,5-Hydroxyxanthotoxin
5-Hydroxy-8-methoxypsoralen (5-Hydroxyxanthotoxin) is a metabolite derived from Xanthotoxin, which acts as a potent tric...
TN3281 8-Hydroxy-5-O-beta-D-glucopyranosylpsoralen Others
Standard reference
TN3267 8-(7-Hydroxy-3,7-dimethyl-2,5-octadienyloxy)psoralen Others
TN2425 5,8-Dihydroxypsoralen Others
5,8-Dihydroxypsoralen is a natural product from Pueraria lobata (Willd.) Ohwi
TP2339 Goralatide
Goralatide, isolated from fetal calf bone marrow, exerts a high inhibitory activity on the proliferation of hematopoieti...
T9001 Desketoraloxifene Phospholipase
Desketoraloxifene 是一种选择性雌激素受体调节剂,可抑制哺乳动物 PLD(PLD1 和 PLD2)。
T76834 Toralizumab
Toralizumab (IDEC-131) 是一种针对 CD40L (CD154)的人源化单克隆抗体 (mAb),由人 γ1 重链和人 kappa 轻链组成。Toralizumab 特异性结合 T 细胞上的人 CD40L,从而阻止 CD4...
T30740 Carbocloral Prodorm,Uralium,Uraline,Chloralurethane,Carbochloral
Carbocloral is a bio-active chemical.
T131510 Isopsoralidin
Oral antiplatelet agent 1
T12316
synonym:
Target:
Dienestrol diacetate
T20764
synonym: NSC81279,Cycladiene,Retalon-oral,NSC-81279,NSC 81279,Oestrasid C
Target:
Avoralstat
T14358
synonym: BCX4161
Target:
Isopsoralenoside
TN1148
synonym:
Target:
Psoralenoside
TN1008
synonym:
Target:
Psoralidin
T3399
synonym:
Target:
Dicloralurea
T1251
synonym: DCU,Dichlorolurea,双(三氯乙醛基)脲,双 (三氯乙醛基) 脲
Target:
8-Geranyloxypsoralen
TN1343
synonym: 8-香叶草氧基补骨脂素
Target:
Coralyne chloride
T31011
synonym:
Target:
Psoralen
T2942
synonym: 补骨脂素,psoralene,Furocoumarin,Ficusin
Target:
8-[(6,7-Dihydroxy-3,7-dimethyloct-2-en-1-yl)oxy]psoralen
TN6298
synonym:
Target:
5-Hydroxy-8-methoxypsoralen
T40859
synonym: 5-Hydroxy-8-methoxypsoralen,5-Hydroxyxanthotoxin
Target:
8-Hydroxy-5-O-beta-D-glucopyranosylpsoralen
TN3281
synonym:
Target:
8-(7-Hydroxy-3,7-dimethyl-2,5-octadienyloxy)psoralen
TN3267
synonym:
Target:
5,8-Dihydroxypsoralen
TN2425
synonym:
Target:
Goralatide
TP2339
synonym:
Target:
Desketoraloxifene
T9001
synonym:
Target:
Toralizumab
T76834
synonym:
Target:
Carbocloral
T30740
synonym: Prodorm,Uralium,Uraline,Chloralurethane,Carbochloral
Target:
Isopsoralidin
T131510
synonym:
Target:
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