T12316 |
Oral antiplatelet agent 1
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Others
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Oral antiplatelet agent 1 is a potent antiplatelet agent with an IC50 of 2.94 μM in vitro. |
T20764 |
Dienestrol diacetate
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NSC81279,Cycladiene,Retalon-oral,NSC-81279,NSC 81279,Oestrasid C |
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Dienestrol diacetate, a derivative of the synthetic non-steroid phenolic compound, DIENESTROL, exhibits estrogenic activ... |
T14358 |
Avoralstat
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BCX4161 |
Others
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Avoralstat 是血浆激肽释放酶(PKK)抑制剂,具有口服活性,可用于遗传性血管性水肿的研究。 |
TN1148 |
Isopsoralenoside
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Antibacterial
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Estrogen Receptor/ERR
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Estrogen/progestogen Receptor
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Isopsoralenoside 是补骨脂多糖中的一种苯并呋喃苷。它在消化道内容物中可迅速代谢为补骨脂素。它具有雌激素样活性、促进成骨细胞增殖活性、抗肿瘤活性和抗菌活性。 |
TN1008 |
Psoralenoside
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Calcium Channel
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CaMK
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Histamine Receptor
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Psoralenoside 是源于补骨脂中的苯并呋喃苷,具有抗肿瘤、抗菌、促进成骨细胞增殖和雌激素样活性。它对组胺 H1、钙调素和电压门控 l 型钙通道具有较高的亲和力。 |
T3399 |
Psoralidin
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Reactive Oxygen Species
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Antibacterial
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Others
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Akt
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Gamma-secretase
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COX
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Estrogen/progestogen Receptor
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Lipoxygenase
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Psoralidin 是COX-2和5-LOX 的抑制剂,有抗癌,抗菌和抗炎作用。它显著下调NOTCH1信号传导,还极大地诱导活化氧产生。 |
T1251 |
Dicloralurea
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DCU,Dichlorolurea,双(三氯乙醛基)脲,双 (三氯乙醛基) 脲 |
Others
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DCU 是一种兽用的食品添加剂,可用作生长刺激剂。 |
TN1343 |
8-Geranyloxypsoralen
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8-香叶草氧基补骨脂素 |
P450
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Anti-infection
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BACE
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8-Geranyloxypsoralen 是一种呋喃香豆素,分离自葡萄柚,是 P450 3A4 的有效抑制剂(IC50:3.93 μM)。 |
T31011 |
Coralyne chloride
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Topoisomerase
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Coralyne chloride 是一种具有强抗癌活性的原小檗碱化合物。它可用于制备 Coralyne 衍生物,是一种基于荧光 DNA 的分子整流剂,通过位点特异性插入构建成 DNA 双链体。它可作为一种拓扑异构酶 I 毒性分子,诱导拓扑... |
T2942 |
Psoralen
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补骨脂素,psoralene,Furocoumarin,Ficusin |
HIV Protease
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Apoptosis
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Influenza Virus
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DNA/RNA Synthesis
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Psoralen 是从补骨脂种子中提取的一种香豆素。它具有如抗癌、抗氧化、抗抑郁、抗癌、抗菌、抗病毒等多种生物学特性。 |
TN6298 |
8-[(6,7-Dihydroxy-3,7-dimethyloct-2-en-1-yl)oxy]psoralen
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T40859 |
5-Hydroxy-8-methoxypsoralen
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5-Hydroxy-8-methoxypsoralen,5-Hydroxyxanthotoxin |
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5-Hydroxy-8-methoxypsoralen (5-Hydroxyxanthotoxin) is a metabolite derived from Xanthotoxin, which acts as a potent tric... |
TN3281 |
8-Hydroxy-5-O-beta-D-glucopyranosylpsoralen
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Others
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Standard reference |
TN3267 |
8-(7-Hydroxy-3,7-dimethyl-2,5-octadienyloxy)psoralen
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Others
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TN2425 |
5,8-Dihydroxypsoralen
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Others
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5,8-Dihydroxypsoralen is a natural product from Pueraria lobata (Willd.) Ohwi |
TP2339 |
Goralatide
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Goralatide, isolated from fetal calf bone marrow, exerts a high inhibitory activity on the proliferation of hematopoieti... |
T9001 |
Desketoraloxifene
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Phospholipase
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Desketoraloxifene 是一种选择性雌激素受体调节剂,可抑制哺乳动物 PLD(PLD1 和 PLD2)。 |
T76834 |
Toralizumab
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Toralizumab (IDEC-131) 是一种针对 CD40L (CD154)的人源化单克隆抗体 (mAb),由人 γ1 重链和人 kappa 轻链组成。Toralizumab 特异性结合 T 细胞上的人 CD40L,从而阻止 CD4... |
T30740 |
Carbocloral
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Prodorm,Uralium,Uraline,Chloralurethane,Carbochloral |
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Carbocloral is a bio-active chemical. |
T131510 |
Isopsoralidin
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