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Cat No. | Product Name | Synonyms | Targets |
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T9061 | EN4 | EN4 MYC inhibitor | c-Myc |
EN4 (EN4 MYC inhibitor) MYC inhibitor is a covalent ligand that targets cysteine 171 (C171) of MYC. It is selective for c-MYC over N-MYC and L-MYC, and inhibits MYC transcriptional activity, downregulates MYC targets, an... | |||
TP1315 | C-Myc Peptide Trifluoroacetate | Others | |
c-Myc Peptide Trifluoroacetate is a synthetic peptide corresponding to the C-terminal amino acids (410-419) of human c-myc protein. c-Myc Peptide Trifluoroacetate participates in regulation of growth-related gene transcr... | |||
T3048 | 10058-F4 | c-Myc Inhibitor | c-Myc , Autophagy |
10058-F4 (c-Myc Inhibitor) is a cell-permeable thiazolidinone that specifically inhibits the c-Myc-Max interaction and prevents transactivation of c-Myc target gene expression; induces cell-cycle arrest and apoptosis. | |||
TP2311 | C-MYC PEPTIDE EPITOPE TFA | Others | |
C-MYC PEPTIDE EPITOPE TFA, the product of the c-myc proto-oncogene, is a helix-loop-helix leucine zipper phosphoprotein that regulates gene transcription in cell proliferation, cell differentiation and apoptosis. This pe... | |||
T39751 | MYC-IN-2 | ||
MYC-IN-2 is a protein-protein inhibitor targeting the MYC protein, designed for use in cancer research. | |||
T72040 | C-Myc inhibitor 7 | ||
C-Myc Inhibitor 7, serving as both a c-Myc inhibitor and a multi-target protein degrader, effectively degrades proteins c-MYC, CK1α, GSPT1, and IKZF1/2/3 across various tumor cell types. It holds potential for research i... | |||
TP2179 | C-Myc tag Peptide | Others | |
c-Myc Peptide is a useful displacement of c-Myc-tagged fusion proteins bound to anti-c-Myc antibodies in immunoassays. The successful inhibition of antibody binding by c-Myc peptide demonstrates binding is specific. c-My... | |||
T3686 | 10074-G5 | c-Myc , Autophagy | |
10074-G5 is an inhibitor of c-Myc-Max dimerization. | |||
T4252 | ML327 | c-Myc , Autophagy | |
ML327 is a MYC blocker. ML327 can also de-repress E-cadherin transcription and reverse Epithelial-to-Mesenchymal Transition (EMT). | |||
T15665 | KJ Pyr 9 | c-Myc , Autophagy | |
KJ Pyr 9 is an MYC inhibitor (Kd: 6.5 nM in vitro assay). | |||
T9628 | 10074-A4 | c-Myc | |
10074-A4 is a c-Myc binding compound that associates with c-Myc370–409 and behaves like a “ligand cloud” around a “protein cloud”, with distinct features from that of a non-binding ligand. | |||
T12132 | MYCi361 | NUCC-0196361 | c-Myc |
MYCi361 (NUCC-0196361) is an inhibitor of MYC (binding to MYC with Kd of 3.2 μM). | |||
T4367 | Mycro 3 | Mycro-3 | c-Myc , Autophagy |
Mycro 3 is potent and selective for c-Myc in whole cell assays. | |||
T12134 | MYCMI-6 | NSC354961 | Apoptosis , c-Myc |
MYCMI-6 (NSC-354961) is a potent and selective inhibitor of endogenous MYC:MAX protein interactions,reduces proliferation and induces massive apoptosis in tumor tissue from a MYC-driven xenograft tumor model without seve... | |||
T60019 | VPC-70063 | Thiourea, N-[3,5-bis(trifluoromethyl)phenyl]-N'-(phenylmethyl)- | Apoptosis , PARP , c-Myc |
VPC-70063 (Thiourea, N-[3,5-bis(trifluoromethyl)phenyl]-N'-(phenylmethyl)-) is an inhibitor of c-Myc-MAX. VPC-70063 exhibits Myc-Max transcriptional activity inhibition of 106% with an IC50 of 8.9 μM and Myc-Max/UBE2C do... | |||
T9033 | BTYNB | MDK6620,BTYNB IMP1 Inhibitor | Others , c-Myc , NF-κB |
BTYNB (MDK6620) is an inhibitor of the oncofetal mRNA-binding protein IMP1 (IC50 = 5 μM for IMP1 binding to c-Myc mRNA). MDK6620 downregulates β-TrCP1 mRNA and reduces activation of nuclear transcriptional factors-kappa ... | |||
T78055 | MYC-RIBOTAC | c-Myc | |
MYC-RIBOTAC, a ribonuclease-targeting chimera (RIBOTAC) specific to the MYC internal ribosome entry site (IRES), comprises an MYC mRNA-binding element tethered to a small molecule that recruits and activates RNase L1. Th... | |||
T10352 | APTO-253 | LOR-253,LT-253 | Apoptosis , c-Myc , KLF |
APTO-253 (LOR-253) inhibits c-Myc expression, stabilizes G-quadruplex DNA, and induces cell cycle arrest and apoptosis in acute myeloid leukemia cells. APTO-253 mediates anticancer activity through the induction of the K... | |||
T74460 | C-Myc inhibitor 5 | ||
c-Myc Inhibitor 5 (DA3) is a fluorescent bispurine compound with a long-chain bridge that selectively binds to the c-MYC G-quadruplex, exhibiting a dissociation constant (K D) of 16 μM. Unlike other G4-driven oncogenes, ... | |||
T72619 | C-Myc inhibitor 8 | ||
C-Myc Inhibitor 8 is an effective compound for cancer research, inhibiting cell viability across a range of cancer types and demonstrating growth suppression in human prostate and lung cancers within mouse models. This i... | |||
T9032 | MGH-CP1 | Others | |
MGH-CP1 is a potent and selective inhibitor TEAD palmitoylation. It exhibits dose-dependent and potent inhibition of TEAD2/4 auto-palmitoylation in vitro with IC50 of 710 nM and 672 nM, respectively. | |||
T9370 | DCBP-1 | Epigenetic Reader Domain , Ligand for E3 Ligase | |
dCBP-1 is a chemical degrader of p300/CBP. dCBP-1 hijacks the E3 ubiquitin ligase CRBN for selective degradation of p300/CBP. Degradation of p300/CBP by dCBP-1 leads to effective multiple myeloma cell killing. | |||
T63359 | C-Myc inhibitor 4 | ||
c-Myc inhibitor 4 is a potent, orally active c-Myc-reducing compound. c-Myc is an important proto-oncogene, which is closely associated with the development of many tumors. | |||
T79439 | C-Myc inhibitor 12 | c-Myc | |
Compound 67h, also known as c-Myc inhibitor 12, is a potent inhibitor of c-Myc, exhibiting a pEC50 value of 6.4 [1]. | |||
T72620 | C-Myc inhibitor 9 | ||
c-Myc Inhibitor 9 (Compound 332) is an effective c-Myc inhibitor, exhibiting a logEC50 of ≥6, and demonstrating significant tumor growth inhibition in nude mouse models. This compound is utilized in cancer research. | |||
T79438 | C-Myc inhibitor 11 | c-Myc | |
c-Myc inhibitor 11 (Compound 67e), a c-MYC inhibitor (p EC 50 : 6.4), exhibits high clearance, a moderate volume of distribution, and a short half-life in rat pharmacokinetic assays, making it suitable for cancer researc... | |||
T75239 | C-Myc inhibitor 10 | ||
C-Myc Inhibitor 10 (compound 17), exhibiting enhanced cellular potency, benefits from increased permeability due to the methylation of the morpholine nitrogen [1]. | |||
T9093 | NY2267 | Acetic acid, 2-[[6-[2-(cyclohexylamino)-1-[[(4-methoxyphenyl)methyl](2-pyridinylcarbonyl)amino]-2-oxoethyl]-2-naphthalenyl]oxy]-, 1,1-dimethylethyl ester | c-Myc |
NY2267 (Acetic acid, 2-[[6-[2-(cyclohexylamino)-1-[[(4-methoxyphenyl)methyl](2-pyridinylcarbonyl)amino]-2-oxoethyl]-2-naphthalenyl]oxy]-, 1,1-dimethylethyl ester) is a disruptor of Myc-Max interaction, with an IC50 of 36... | |||
T20533 | NNK | Nicotine-derived nitrosamine ketone | Lipoxygenase |
NNK (Nicotine-derived nitrosamine ketone) is a procarcinogen and a major tobacco-specific toxicant. It inhibits the expression of lysyl oxidase which is a tumor suppressor. | |||
T11284 | FIDAS-3 | Others , Wnt/beta-catenin , Methionine Adenosyltransferase (MAT) | |
FIDAS-3, a stilbene derivative and potent Wnt inhibitor with an IC50 of 4.9 μM for methionine S-adenosyltransferase 2A (MAT2A), exhibits anticancer activities by effectively competing with S-adenosylmethionine (SAM) for ... | |||
T11285 | FIDAS-5 | Others | |
FIDAS-5, a potent and orally active methionine S-adenosyltransferase 2A (MAT2A) inhibitor with an IC50 of 2.1 μM, competitively inhibits S-adenosylmethionine (SAM) binding to MAT2A. It exhibits anticancer activities. | |||
T10760 | Ceramides Mixture | Telomerase | |
Ceramides Mixture, an endogenous ceramide, consists of hydroxy and non-hydroxy fatty acid-containing ceramides. It is involved in the regulation of cell cycle arrest, growth inhibition, and modulation of telomerase activ... | |||
T6010 | Idarubicin hydrochloride | Idamycin,4-demethoxydaunorubicin (NSC256439, 4-DMDR) HCl,4-Demethoxydaunorubicin hydrochloride,Idarubicin HCl,Zavedos | Topoisomerase , Antibacterial , Autophagy , Antifungal |
Idarubicin hydrochloride (Zavedos), a hydrochloride salt form of Idarubicin, is a DNA topoisomerase II (topo II) inhibitor for MCF-7 cells ( IC50: 3.3 ng/mL). | |||
T8658 | NEO2734 | EP31670 | Epigenetic Reader Domain , Histone Acetyltransferase |
NEO2734 (EP31670) is an orally active and selective inhibitor of p300/CBP and BET bromodomain(IC50 of <30 nM for both p300/CBP and BET bromodomains). | |||
T10765 | Eragidomide | CC-90009,Cereblon modulator 1 | Apoptosis , Ligand for E3 Ligase , Molecular Glues |
Eragidomide (CC-90009; Cereblon modulator 1) is a cereblon (CRBN) E3 ligase modulator. Eragidomide specifically binds to CRBN, thereby affecting the activity of the ubiquitin E3 ligase complex. | |||
T6203 | Saxagliptin | BMS-477118,Onglyza | Proteasome , DPP-4 |
Saxagliptin (BMS-477118) is a selective and reversible DPP4 inhibitor with IC50 of 26 nM. | |||
T0178 | Saxagliptin hydrate | Onglyza hydrate,BMS-477118 hydrate | Proteasome , DPP-4 |
Saxagliptin hydrate (Onglyza hydrate) is a selective and reversible DPP4 inhibitor (IC50: 26 nM; Ki: 1.3 nM). | |||
T12133 | MYCi975 | NUCC-0200975 | c-Myc |
MYCi975 (NUCC-0200975) is an orally active inhibitor of MYC. | |||
T3131 | Fosfomycin calcium | Phosphomycin calcium salt,Fosmicin | Antibacterial , Antibiotic |
Fosfomycin calcium (Phosphomycin calcium salt) is a blood-brain barrier penetrating, broad-spectrum antibiotic by irreversibly inhibiting an early stage in cell wall synthesis. | |||
T6448 | Clindamycin hydrochloride | Sobelin HCl,Cleocin,Clindamycin HCl,Clinimycin HCl | Antibacterial , Antibiotic |
Clindamycin hydrochloride (Clinimycin HCl) inhibits protein synthesis by acting on the 50S ribosomal. It is the hydrochloride salt form of clindamycin, a semi-synthetic, chlorinated broad-spectrum antibiotic produced by ... | |||
T6297 | Alvespimycin hydrochloride | BMS 826476,NSC 707545,KOS-1022,17-DMAG hydrochloride,Alvespimycin (17-DMAG) HCl | Apoptosis , HSP |
Alvespimycin hydrochloride (BMS 826476) is a potent HSP90 inhibitor with IC50 of 62 nM. Phase 2. | |||
T1557 | Acetylspiramycin | Spiramycin II,Foromacidin B,ASPM,Spiramycin B | ribosome , Antibacterial , Antibiotic |
Acetylspiramycin (Spiramycin B) targets 50S ribosome to inhibit protein synthesis. | |||
T26308 | Lipoxamycin hemisulfate | Lipoxamycin, sulfate (2:1),U-26146D,U26146D,U 26146D,Lipoxamycin | Antifungal |
Lipoxamycin hemisulfate (Lipoxamycin) is an inhibitor of serine palmitoyltransferase (IC50 = 21 nM) with antifungal activity. | |||
T13303 | Virginiamycin M1 | Pristinamycin IIA,Ostreogrycin A | Antibacterial |
Virginiamycin M1 (Pristinamycin IIA) is a macrocyclic lactone peptide antibiotic and is a member of the streptogramin A group of antibiotics. | |||
T11120 | Duocarmycin TM | DNA Alkylation , Antibiotic | |
Duocarmycin TM is a DNA alkylator. Duocarmycin TM is an exceptionally potent antitumor antibiotic. | |||
T0788L | Spectinomycin dihydrochloride pentahydrate | Trobicin,Spectogard,Spectinomycin hydrochloride hydrate | ribosome , Antibacterial , Antibiotic |
Spectinomycin dihydrochloride pentahydrate (Spectogard) is an antibiotic produced by Streptomyces spectabilis. It is active against gram-negative bacteria and used for the treatment of gonorrhea. | |||
T2096 | Framycetin sulfate | Neomycin Sulphate B,Framycetin sulphate | Antibacterial , Antibiotic |
Framycetin sulfate (Neomycin Sulphate B) belongs to aminoglycoside class of antibiotics that contain two or more aminosugars connected by glycosidic bonds. | |||
T12284 | O-Propargyl-Puromycin | OP-puro,O-Propargylpuromycin | Others |
O-Propargyl-Puromycin (OP-puro) is a potent protein synthesis inhibitor, a puromycin acetylene analog. | |||
T15735 | Leptomycin B | CI 940,LMB | CRM1 , Antibiotic , Antifungal |
Leptomycin B (LMB) is a potent inhibitor of the nuclear export of proteins and is a potent antifungal antibiotic blocking the eukaryotic cell cycle. Leptomycin B inactivates CRM1/exportin 1 by covalent modification at a ... | |||
T11315 | Fosmidomycin sodium salt | FR-31564 sodium salt | Antibiotic , Parasite |
Fosmidomycin sodium salt (FR-31564 sodium salt) is an anti-infective antibiotic with anti-malarial activity that inhibits both Gram-negative and Gram-positive bacteria. |
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
TN1892 | Lusianthridin | Others , c-Myc | |
Lusianthridin is a natural product from Dendrobium venustum. Lusianthridin exhibits anti-migratory property at nontoxic concentrations. Lusianthridin enhances c-Myc degradation through the inhibition of Src-STAT3 signali... | |||
T21065 | Artemisitene | Others | |
Artemisitene is the oxidized form of Artemisinin and is an antimalarial agent. Artemisinin precursors are the important basic substances for biosynthesis of Artemisinin, including Artemisinin B, Artemisitene, Artemisini... | |||
T3673 | Mollugin | Rubimaillin | HER , JAK |
Mollugin (Rubimaillin) may be a JAK2 inhibitor and inhibits LPS-induced inflammatory responses by blocking the activation of the JAK-STAT pathway. Mollugin as a candidate for a chemotherapeutic agent in OSCCs via the upr... | |||
T4S1173 | Agrimol B | Sirtuin , PPAR | |
1. Agrimol B is a main active ingredient isolated from Agrimonia pilosa Ledeb. | |||
T2764 | (S)-10-Hydroxycamptothecin | 10-Hydroxycamptothecin,10-HCPT | Apoptosis , Topoisomerase |
(S)-10-Hydroxycamptothecin (10-HCPT) is a DNA topoisomerase I inhibitor, utilized as a clinical therapy agent against hepatoma. | |||
T0060 | Streptomycin sulfate | Plantomycin,Estreptomicina,Phytomycin | ribosome , Antibacterial , Antibiotic |
Streptomycin sulfate (Phytomycin) is a sulfate salt of streptomycin that is a protein synthesis inhibitor. | |||
T8118 | Bekanamycin | Kanamycin B | Antibacterial , Antibiotic |
Bekanamycin (Kanamycin B) is an aminoglycoside antibiotic. | |||
T21820 | Resistomycin | Geliomycin,Heliomycin | Antibiotic |
Resistomycin (Geliomycin), a pentacyclic polyketide antibiotic, exhibits potent anticancer properties by triggering apoptosis. | |||
T12540 | Pristinamycin IA | Mikamycin IA,Mikamycin B | Others , Antibiotic , P-gp |
Pristinamycin IA (Mikamycin B) is a substrate for the P-glycoprotein and a cyclo-peptidic macrolactone antibiotic. | |||
T0474 | Erythromycin ethylsuccinate | EES | ribosome , HIV Protease , Antibacterial , Antibiotic , Autophagy |
Erythromycin ethylsuccinate (EES) is a macrolide antibiotic, produced by Streptomyces erythreus. | |||
T0971 | Dirithromycin | Dirithromycinum,ASE 136,LY237216,Diritromicina,Dirithromycine | ribosome , Antibacterial , Antibiotic |
Dirithromycin (LY237216) is a macrolide glycopeptide antibiotic. It is used to treat many different types of bacterial infections, such as bronchitis, pneumonia, tonsillitis, and even skin infections. | |||
T1032 | Erythromycin | E-Mycin | ribosome , Antibacterial , Antibiotic |
Erythromycin (E-Mycin) is a Macrolide and Macrolide Antimicrobial. The physiologic effect of erythromycin is by means of Decreased Sebaceous Gland Activity. | |||
T1235 | Lincomycin hydrochloride monohydrate | Lincomycin hydrochloride hydrate | ribosome , Antibacterial , Antibiotic |
Lincomycin hydrochloride monohydrate (Lincomycin hydrochloride hydrate) is an antibiotic produced by Streptomyces lincolnensis var. lincolnensis. It has been used in the treatment of staphylococcal, streptococcal, and Ba... | |||
T3629 | Gamithromycin | ML-1709460 | Antibacterial , Antibiotic |
Gamithromycin (ML-1709460) is a macrolide compound with antibacterial activity. | |||
T1419 | Azithromycin hydrate | CP-62993 dihydrate,Azithromycin dihydrate | ribosome , Antibacterial , Antibiotic , Autophagy |
Azithromycin hydrate (CP-62993 dihydrate) is a semi-synthetic macrolide antibiotic structurally related to ERYTHROMYCIN. It has been used in the treatment of Mycobacterium avium intracellulare infections, toxoplasmosis, ... | |||
T1335 | Mycophenolic acid | Mycophenolate,RS-61443 | Apoptosis , Dehydrogenase , Endogenous Metabolite , Antibacterial , Antibiotic , UGT , Antifungal |
Mycophenolic acid (Mycophenolate) is an inosine monophosphate dehydrogenase(IMPDH) inhibitor with anti-proliferative activity. | |||
T17143 | Toyocamycin | Vengicide | Apoptosis , Others , IRE1 , Antibiotic , Antifungal |
Toyocamycin (Vengicide) is an adenosine analog produced by Actinomycete, acts as an XBP1 inhibitor, inhibits IRE1α-induced ATP-dependent XBP1 mRNA cleavage (IC50: 80 nM). Toyocamycin induces apoptosis. | |||
TP1072 | Valinomycin | NSC 122023 | Apoptosis , PTEN , Antibacterial , Antibiotic , Autophagy |
Valinomycin (NSC-122023) is a cyclic depsipeptide antibiotic and a potassium-specific ionophore.Valinomycin induces PINK1 activation and promotes Parkin phosphorylation at Ser65. | |||
T20699 | Daunomycinone | Daunomycinon,Leukaemomycinone C,NSC 109351,NSC-109351,NSC109351 | Antibiotic |
Daunomycinone (NSC-109351) is a glycan of daunomycin, which belongs to the antibiotic class and is a representative glycan of tumour-inhibiting anthracyclines, used in the treatment of cancer and leukaemia. | |||
T1084 | Apramycin sulfate | Nebramycin II,Ai3-29795 | Antibacterial , Antibiotic |
Apramycin sulfate (Nebramycin II) is an aminoglycoside antibiotic. | |||
T5003 | Rifamycin sodium | Rifamycin sodium salt | Antibacterial , Antibiotic |
Rifamycin sodium (Rifamycin sodium salt) salt is an antibiotic that inhibits bacterial DNA-dependent RNA polymerase. It is effective against Gram-positive bacteria. | |||
T2481 | Ascomycin | FK520,Immunomycin,FR-900520 | Phosphatase , Others , Antibiotic , Parasite , Antifungal |
Ascomycin (Immunomycin)(Immunomycin, FR-900520, FK520) is an ethyl analog of tacrolimus (FK506) with strong immunosuppressant properties. | |||
T0950 | Neomycin sulfate | Framycin sulfate | Phospholipase , ribosome , Antibacterial , Antibiotic |
Neomycin sulfate (Framycin sulfate) is a broad-spectrum aminoglycoside antibiotic that blocks the synthesis of bacterial proteins in order to exert antimicrobial activity. Neomycin sulfate is commonly used to screen prok... | |||
T21344 | 1-Deoxynojirimycin hydrochloride | Moranoline,AT2220,Duvoglustat hydrochloride,1-Deoxynojirimycin,DNJ,deoxynojirimycin | PI3K , Antibacterial , Antibiotic , Glucosidase |
1-Deoxynojirimycin hydrochloride (Moranoline) is a potent and selective inhibitor of alpha-glucosidase, most commonly found in mulberry leaves. Duvoglustat is used to suppress the elevation of postprandial hyperglycemia. | |||
T36818 | Questiomycin A | GPR , Antibacterial | |
Questiomycin A is an antibiotic produced in crème fraiche with antibacterial and anticancer activities. Questiomycin A suppresses expression of GRP78, a cell-protective ER chaperone protein. | |||
T9605 | Sangivamycin | BA-90912,NSC 65346 | Nucleoside Antimetabolite/Analog , PKC |
Sangivamycin (NSC-65346) is an effective inhibitor of protein kinase C (PKC, Ki = 10 μM). Sangivamycin exhibits antiproliferative activity against a variety of human cancers. | |||
T60104 | Mycophenolic acid-β-D-glucuronide solution | Others | |
Mycophenolic acid glucuronide is the glucuronide metabolite of mycophenolic acid in human plasma. | |||
T21494 | Oligomycin | HIF | |
Oligomycin is an antifungal antibiotic that is an inhibitor of H+-ATP synthetase. The Oligomycin blocks oxidative phosphorylation and the electron transport chain. Oligomycin inhibited HIF-1alpha expression in hypoxic tu... | |||
T13229 | Tunicamycin | Influenza Virus , Antibacterial , Antibiotic , Antifungal | |
Tunicamycin is a mixture of antibiotics that inhibit N-linked glycosylation by blocking GlcNAc phosphotransferase (GPT). Tunicamycin has antitumor activity, as well as anti-bacterial, anti-fungal, and anti-viral activity... | |||
T6740 | Bafilomycin A1 | Apoptosis , Proton pump , Antibacterial , Antibiotic , Autophagy | |
Bafilomycin A1 belongs to the macrolide class of antibiotics and is a V-ATPase (IC50=0.44 nM) that is specific and reversible. Bafilomycin A1 is an inhibitor of the late phase of autophagy, blocking the fusion of autopha... | |||
T1381 | Milbemycin oxime | Others , Antibiotic , Parasite | |
Milbemycin oxime is a broad spectrum antiparasitic, used as a veterinary drug. | |||
T3675 | 1-Deoxynojirimycin | Duvoglustat,Moranoline,moranolin | PI3K , Glucosidase |
1-Deoxynojirimycin (Moranoline) is a potent α-glucosidase inhibitor, suppressing postprandial blood glucose, thereby possibly preventing diabetes mellitus. | |||
T8262 | Fosfomycin sodium | Fosfomycin Disodium | Antibacterial , Antibiotic |
Fosfomycin sodium is a bactericidal, low-molecular weight, broad-spectrum antibiotic, with putative activity against several bacteria, including multidrug-resistant Gram-negative bacteria, by irreversibly inhibiting an e... | |||
T1441 | Capreomycin sulfate | Capastat sulfate | ribosome , Antibacterial , Antibiotic |
Capreomycin sulfate (Capastat sulfate) , a cyclic peptide antibiotic, binds to the 70S ribosomal unit leading to inhibition of protein synthesis. | |||
T1104 | Paromomycin Sulfate | Aminosidine sulfate,Paromomycin sulfate salt | Antibacterial , Antibiotic , Parasite |
Paromomycin binds specifically to the RNA oligonucleotide at the A site of bacterial 30S ribosomes, thereby causing misreading and premature termination of translation of mRNA and inhibition of protein synthesis followed... | |||
T14854 | Caerulomycin A | Cerulomycin,Caerulomycin | Antifungal |
Caerulomycin A (Caerulomycin) (Cerulomycin; Caerulomycin) is an antifungal compound. Which induces generation of T cells, enhances TGF-β-Smad3 protein signaling via suppressing interferon-γ-induced STAT1 signaling. Antif... | |||
T0788 | Spectinomycin dihydrochloride | Spectinomycin 2HCl,Actinospectacin | ribosome , Antibacterial , Antibiotic |
Spectinomycin dihydrochloride (Actinospectacin) is an antibiotic produced by Streptomyces spectabilis. It is active against gram-negative bacteria and used for the treatment of gonorrhea. | |||
T6447 | Clindamycin | Clinimycin,Sobelin,Chlolincocin | Antibacterial , Antibiotic |
Clindamycin (Sobelin) dissociates peptidyl-tRNA from the bacterial ribosome, thereby disrupting bacterial protein synthesis. Clindamycin is a semisynthetic broad-spectrum antibiotic produced by chemical modification of t... | |||
T19424 | Methyl mycophenolate | Mycophenolic Acid Methyl Ester | Others |
Methyl mycophenolate (Mycophenolic Acid Methyl Ester) is found in the marine fungus Phaeosphaeria spartinae. Methyl mycophenolate is the methyl ester form of mycophenolic acid. | |||
T0819 | Spiramycin | Espiramicin,Sequamycin,Rovamycin,Provamycin,Formacidine | Antibacterial , Antibiotic , Parasite |
Spiramycin (Rovamycin) is a macrolide antibiotic produced by Streptomyces ambofaciens. The drug is effective against gram-positive aerobic pathogens, N. gonorrhoeae, and staphylococci. It is used to treat infections caus... | |||
T5037 | Midecamycin | Antibiotic SF-837,Turimycin P3,Medecamycin A1,Rubimycin,Platenomycin B1,Espinomycin A | Antibacterial , Antibiotic |
Midecamycin (Medecamycin A1), an acetoxy-substituted macrolide antibiotic, has effective on gram-positive and gram-negative bacteria acts by inhibiting bacterial protein synthesis. | |||
T67867 | Mycaminosyltylonolide | Antibacterial | |
Mycaminosyltylonolide is a macrolide antibiotic that is tylonolide having a beta-D-mycaminosyl residue attached at position 5. Mycaminosyltylonolide is a potent antibiotic with antibacterial activity and inhibits lucifer... | |||
T67731 | Holomycin | N-Demethylthiolutin | DNA/RNA Synthesis |
Holomycin (N-Demethylthiolutin) is a secondary metabolite of dithiopyrrolidone. HolomycinHolomycin, an antibiotic secondary metabolite, is required for the biofilm formation of natural photogenic Bacillus galatheae S2753... | |||
T6995 | Ochromycinone | STA 21,STA21,STA-21 | Antibacterial , STAT |
Ochromycinone (STA 21) is a selective STAT3 inhibitor. | |||
T6290 | Tanespimycin | 17-AAG,CP 127374,NSC 330507,KOS 953 | Apoptosis , Mitophagy , HSP , Antibacterial , Antibiotic , Autophagy |
Tanespimycin (KOS 953) (17-AAG) is an inhibitor of Hsp90 that selectively inhibits BT474 tumor cell Hsp90 (IC50: 5 nM). | |||
T1277 | Lincomycin hydrochloride | Lincomycin HCl,NSC 70731,U10149A | ribosome , Antibacterial , Antibiotic |
Lincomycin hydrochloride (U10149A) is a lincosamide antibiotic identified in S.lincolnensis with activity against gram-positive cocci and anaerobic bacteria. | |||
T6323 | Oligomycin A | MCH 32 | ATPase , Antibiotic , Antifungal |
Oligomycin A (MCH 32) is an inhibitor of ATP synthase, inhibits oxidative phosphorylation and all the ATP-dependent processes occurring on the coupling membrane of mitochondria. | |||
T8641 | Vancomycin | Antibacterial , Antibiotic , Autophagy | |
Vancomycin is a glycopeptide antibiotic that exerts its antimicrobial activity by altering the permeability of cell membranes and selectively inhibiting ribonucleic acid synthesis. Vancomycin can be used for the treatmen... | |||
T1665 | Daptomycin | LY146032 | DNA/RNA Synthesis , Antibacterial , Antibiotic |
Daptomycin (LY146032) is a cyclic lipopeptide antibiotic that inhibits GRAM-POSITIVE BACTERIA. | |||
T21498 | Phleomycin | DNA/RNA Synthesis , Antibacterial , Antibiotic | |
Phleomycin is one of the anticancer glycopeptide antibiotics which cause DNA cleavage. It is similar to Bleomycin which binds and intercalates DNA to damage the integrity of the double helix. | |||
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Cat No. | Product Name | Species | Expression System |
---|---|---|---|
TMPH-02791 | C-Myc Protein, Mouse, Recombinant (GST) | Mouse | E. coli |
c-Myc Protein, Mouse, Recombinant (GST) is expressed in E. coli. | |||
TMPH-01720 | C-Myc Protein, Human, Recombinant (His) | Human | E. coli |
Transcription factor that binds DNA in a non-specific manner, yet also specifically recognizes the core sequence 5'-CAC[GA]TG-3'. Activates the transcription of growth-related genes. Binds to the VEGFA promoter, promotin... | |||
TMPH-01721 | C-Myc Protein, Human, Recombinant (Avi & His & MBP), Biotinylated | Human | E. coli |
Transcription factor that binds DNA in a non-specific manner, yet also specifically recognizes the core sequence 5'-CAC[GA]TG-3'. Activates the transcription of growth-related genes. Binds to the VEGFA promoter, promotin... | |||
TMPY-02888 | MAX Protein, Human, Recombinant (His & GST) | Human | Baculovirus-Insect Cells |
MYC associated factor X contains 1 basic helix-loop-helix (bHLH) domain and belongs to the MAX family. It is highly expressed in the brain, heart, and lung while lower levels are seen in the liver, kidney, and skeletal m... | |||
TMPJ-01040 | MAX Protein, Human, Recombinant (His) | Human | E. coli |
Myc-Associated Factor X (MAX) is a member of the basic helix-loop-helix leucine zipper (bHLHZ) family of transcription factors. It contains 1 basic helix-loop-helix (bHLH) domain. It is found in the brain, heart, and lun... | |||
TMPH-03328 | Mcpt1 Protein, Rat, Recombinant (Myc) | Rat | E. coli |
Mcpt1 Protein, Rat, Recombinant (Myc) is expressed in E. coli. | |||
TMPH-02552 | BMP3 Protein, Mouse, Recombinant (Myc) | Mouse | E. coli |
Negatively regulates bone density. Antagonizes the ability of certain osteogenic BMPs to induce osteoprogenitor differentitation and ossification. | |||
TMPH-02825 | ACOX1 Protein, Mouse, Recombinant (Myc) | Mouse | E. coli |
Catalyzes the desaturation of acyl-CoAs to 2-trans-enoyl-CoAs. First enzyme of the fatty acid beta-oxidation pathway.; Shows highest activity against medium-chain fatty acyl-CoAs and activity decreases with increasing ch... | |||
TMPH-01898 | PARL Protein, Human, Recombinant (Myc) | Human | in vitro E. coli expression system |
Required for the control of apoptosis during postnatal growth. Essential for proteolytic processing of an antiapoptotic form of OPA1 which prevents the release of mitochondrial cytochrome c in response to intrinsic apopt... | |||
TMPH-01177 | CRISPLD2 Protein, Human, Recombinant (His & Myc) | Human | HEK293 |
CRISPLD2 Protein, Human, Recombinant (His & Myc) is expressed in HEK293. | |||
TMPH-02589 | COL26A1 Protein, Mouse, Recombinant (His & Myc) | Mouse | Baculovirus |
COL26A1 Protein, Mouse, Recombinant (His & Myc) is expressed in Baculovirus. | |||
TMPH-03366 | RUNX1 Protein, Rat, Recombinant (His & Myc) | Rat | Baculovirus |
RUNX1 Protein, Rat, Recombinant (His & Myc) is expressed in Baculovirus. | |||
TMPH-02033 | RPE65 Protein, Human, Recombinant (His & Myc) | Human | Baculovirus |
RPE65 Protein, Human, Recombinant (His & Myc) is expressed in Baculovirus. | |||
TMPH-01986 | PSG7 Protein, Human, Recombinant (His & Myc) | Human | HEK293 |
PSG7 Protein, Human, Recombinant (His & Myc) is expressed in HEK293. | |||
TMPH-00929 | APBA2 Protein, Human, Recombinant (His & Myc) | Human | HEK293 |
APBA2 Protein, Human, Recombinant (His & Myc) is expressed in HEK293. | |||
TMPH-01999 | RAB10 Protein, Human, Recombinant (His & Myc) | Human | Baculovirus |
RAB10 Protein, Human, Recombinant (His & Myc) is expressed in Baculovirus. | |||
TMPH-00924 | AMELX Protein, Human, Recombinant (His & Myc) | Human | Baculovirus |
AMELX Protein, Human, Recombinant (His & Myc) is expressed in Baculovirus. | |||
TMPH-02795 | Myoglobin Protein, Mouse, Recombinant (His & Myc) | Mouse | HEK293 |
Myoglobin Protein, Mouse, Recombinant (His & Myc) is expressed in HEK293. | |||
TMPH-03387 | TSHB Protein, Rat, Recombinant (His & Myc) | Rat | Yeast |
TSHB Protein, Rat, Recombinant (His & Myc) is expressed in Yeast. | |||
TMPH-02084 | SRRM2 Protein, Human, Recombinant (His & Myc) | Human | Baculovirus |
SRRM2 Protein, Human, Recombinant (His & Myc) is expressed in Baculovirus. | |||
TMPH-01981 | NPEPPS Protein, Human, Recombinant (His & Myc) | Human | Baculovirus |
NPEPPS Protein, Human, Recombinant (His & Myc) is expressed in Baculovirus. | |||
TMPH-02793 | Myocilin Protein, Mouse, Recombinant (His & Myc) | Mouse | Baculovirus |
Myocilin Protein, Mouse, Recombinant (His & Myc) is expressed in Baculovirus. | |||
TMPH-00908 | MACROD1 Protein, Human, Recombinant (His & Myc) | Human | Baculovirus |
MACROD1 Protein, Human, Recombinant (His & Myc) is expressed in Baculovirus. | |||
TMPH-01186 | CYP2C9 Protein, Human, Recombinant (His & Myc) | Human | E. coli |
CYP2C9 Protein, Human, Recombinant (His & Myc) is expressed in E. coli. | |||
TMPH-02708 | HNMT Protein, Mouse, Recombinant (His & Myc) | Mouse | E. coli |
HNMT Protein, Mouse, Recombinant (His & Myc) is expressed in E. coli. | |||
TMPH-00499 | PPP1CA Protein, Canine, Recombinant (His & Myc) | Canine | E. coli |
PPP1CA Protein, Canine, Recombinant (His & Myc) is expressed in E. coli. | |||
TMPH-01901 | DDX53 Protein, Human, Recombinant (His & Myc) | Human | E. coli |
DDX53 Protein, Human, Recombinant (His & Myc) is expressed in E. coli. | |||
TMPH-00968 | ATP5C1 Protein, Human, Recombinant (His & Myc) | Human | E. coli |
ATP5C1 Protein, Human, Recombinant (His & Myc) is expressed in E. coli. | |||
TMPH-02072 | SEPHS2 Protein, Human, Recombinant (His & Myc) | Human | E. coli |
SEPHS2 Protein, Human, Recombinant (His & Myc) is expressed in E. coli. | |||
TMPH-02750 | LTBP4 Protein, Mouse, Recombinant (His & Myc) | Mouse | E. coli |
LTBP4 Protein, Mouse, Recombinant (His & Myc) is expressed in E. coli. | |||
TMPH-01952 | SPRY2 Protein, Human, Recombinant (His & Myc) | Human | E. coli |
SPRY2 Protein, Human, Recombinant (His & Myc) is expressed in E. coli. | |||
TMPH-01185 | CYP2C19 Protein, Human, Recombinant (His & Myc) | Human | E. coli |
CYP2C19 Protein, Human, Recombinant (His & Myc) is expressed in E. coli. | |||
TMPH-01178 | CDA Protein, Human, Recombinant (His & Myc) | Human | E. coli |
CDA Protein, Human, Recombinant (His & Myc) is expressed in E. coli. | |||
TMPH-00942 | AP1B1 Protein, Human, Recombinant (His & Myc) | Human | E. coli |
AP1B1 Protein, Human, Recombinant (His & Myc) is expressed in E. coli. | |||
TMPH-01915 | PREB Protein, Human, Recombinant (His & Myc) | Human | E. coli |
PREB Protein, Human, Recombinant (His & Myc) is expressed in E. coli. | |||
TMPH-01993 | PDHX Protein, Human, Recombinant (His & Myc) | Human | E. coli |
PDHX Protein, Human, Recombinant (His & Myc) is expressed in E. coli. | |||
TMPH-00993 | SLC4A1 Protein, Human, Recombinant (His & Myc) | Human | E. coli |
SLC4A1 Protein, Human, Recombinant (His & Myc) is expressed in E. coli. | |||
TMPH-03372 | Sharpin Protein, Rat, Recombinant (His & Myc) | Rat | E. coli |
Sharpin Protein, Rat, Recombinant (His & Myc) is expressed in E. coli. | |||
TMPH-02730 | ITIH2 Protein, Mouse, Recombinant (His & Myc) | Mouse | E. coli |
ITIH2 Protein, Mouse, Recombinant (His & Myc) is expressed in E. coli. | |||
TMPH-01912 | PIBF1 Protein, Human, Recombinant (His & Myc) | Human | E. coli |
PIBF1 Protein, Human, Recombinant (His & Myc) is expressed in E. coli. | |||
TMPH-03340 | NEFH Protein, Rat, Recombinant (His & Myc) | Rat | E. coli |
NEFH Protein, Rat, Recombinant (His & Myc) is expressed in E. coli. | |||
TMPH-02051 | RNF207 Protein, Human, Recombinant (His & Myc) | Human | E. coli |
RNF207 Protein, Human, Recombinant (His & Myc) is expressed in E. coli. | |||
TMPH-01930 | CBFA2T1 Protein, Human, Recombinant (His & Myc) | Human | E. coli |
CBFA2T1 Protein, Human, Recombinant (His & Myc) is expressed in E. coli. | |||
TMPH-01983 | POTEKP Protein, Human, Recombinant (His & Myc) | Human | E. coli |
POTEKP Protein, Human, Recombinant (His & Myc) is expressed in E. coli. | |||
TMPH-01617 | SDS Protein, Human, Recombinant (His & Myc) | Human | E. coli |
SDS Protein, Human, Recombinant (His & Myc) is expressed in E. coli. | |||
TMPH-01572 | KRT34 Protein, Human, Recombinant (His & Myc) | Human | E. coli |
KRT34 Protein, Human, Recombinant (His & Myc) is expressed in E. coli. | |||
TMPH-01465 | HNRNPA2B1 Protein, Human, Recombinant (His & Myc) | Human | E. coli |
HNRNPA2B1 Protein, Human, Recombinant (His & Myc) is expressed in E. coli. | |||
TMPH-01685 | MAST4 Protein, Human, Recombinant (His & Myc) | Human | E. coli |
MAST4 Protein, Human, Recombinant (His & Myc) is expressed in E. coli. | |||
TMPH-03389 | TRPA1 Protein, Rat, Recombinant (His & Myc) | Rat | E. coli |
TRPA1 Protein, Rat, Recombinant (His & Myc) is expressed in E. coli. | |||
TMPH-01436 | FOXA1 Protein, Human, Recombinant (His & Myc) | Human | E. coli |
FOXA1 Protein, Human, Recombinant (His & Myc) is expressed in E. coli. | |||
------------------------ More ------------------------ |
Cat No. | Product Name | ||
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L2130 | Anti-Cancer Metabolism Compound Library | 1280 compounds | |
A unique collection of 1280 cancer cellular metabolism related compounds for cancer research and high throughput screening (HTS) and high content screening (HCS); | |||
L2550 | Glutamine Metabolism Compound Library | 580 compounds | |
A unique collection of 580 glutamine metabolism related compounds can be used for high throughput screening (HTS) and high content screening (HCS), and also is an effective tool for research in glutamine metabolism and ... |