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Compounds

Cat No. Product Name
T12551 PROTAC BRD4 ligand-1 Epigenetic Reader Domain
PROTAC BRD4 ligand-1 是 PROTAC GNE-987 靶向 BRD4 蛋白的配体,也是一种 BET 的抑制剂。
T5835 PROTAC ERRα ligand 2 Estrogen/progestogen Receptor , Estrogen Receptor/ERR
PROTAC ERRα ligand 2 是雌激素相关受体 α (ERRα)反向激动剂。它对 ERRα (IC50=5.67 nM) 的抑制作用比 XCT790 (IC50=61.3 nM) 高效约 11 倍。
T15191 PROTAC ERRα ligand 1 Estrogen Receptor/ERR , Estrogen/progestogen Receptor
PROTAC ERRα ligand 1 是一种雌激素相关受体 α (ERRα) 拮抗剂,能够作用于 ERRα (IC50:0.04 μM)和 ERRγ (IC50:2.8 μM)。
T5437 Gefitinib-based PROTAC 3 EGFR
Gefitinib-based PROTAC 3 通过 linker 将 EGFR 结合元件与 von Hippel-Lindau 配体结合,在 HCC827(外显子 19 del)和 H3255(L858R 突变)细胞中诱导 EGFR 降...
T13722 Homo-PROTAC pVHL30 degrader 1 Others
Homo-PROTAC pVHL30 degrader 1 是一种基于 PROTAC 的 pVHL30 降解剂。
T13721 Homo-PROTAC cereblon degrader 1 Others
Homo-PROTAC cereblon degrader 1 (compound 15a) 是一种高效 cereblon 降解剂,对 IKZF1 和 IKZF3 的影响很小。
T13848 SMARCA-BD ligand 1 for Protac Epigenetic Reader Domain
SMARCA-BD ligand 1 for Protac 能够与 BAF ATPase 亚基 SMARCA2 结合,可用于 PROTAC 技术,用于降解 SMARCA2。
T8745 PROTAC BRAF-V600E degrader-1 Compound 23,Compound 23 Raf
PROTAC BRAF-V600E degrader-1 选择性地诱导 BRAF-V600E 的降解,而不是野生型 BRAF。
T13890 SMARCA-BD ligand 1 for Protac dihydrochloride Epigenetic Reader Domain
SMARCA-BD ligand 1 for Protac dihydrochloride 是一种能够与 BAF ATPase 亚基 SMARCA2 结合的化合物,基于 PROTAC 技术,使 SMARCA2 降解。
T34168 PROTAC-I PROTAC I
PROTAC-I targets steroid hormone receptors for ubiquitination and degradation.
T34167 PROTAC-12 PROTAC12,PROTAC 12
PROTAC-12 is a SirReal-based PROTAC which induces isotype-selective Sirt2 degradation, resulting in the hyperacetylation...
T39920 PROTAC IRAK4 degrader-3 PROTAC IRAK4 degrader-3
PROTAC IRAK4 degrader-3 is a PROTAC-induced IRAK4 degrader based on von Hippel-Lindau.
T36242 PROTAC BRD4 Degrader-5 PROTAC BRD4 Degrader-5
PROTAC BRD4 Degrader-5 is a PROTAC-based BRD4 degrader. PROTAC BRD4 Degrader-5 can potent degrade BRD4 in HER2 positive ...
T40074 PROTAC BRD4 Degrader-15 PROTAC BRD4 Degrader-15
PROTAC BRD4 Degrader-15 is a chemical compound consisting of a PROteolysis TArgeting Chimera (PROTAC) linked to ligands ...
T39902 PROTAC IRAK4 degrader-5 PROTAC IRAK4 degrader-5
PROTAC IRAK4 degrader-5 is a Cereblon-based IRAK4 degrader derived from patent US20190192668A1, compound I-171.
T39903 PROTAC IRAK4 degrader-6 PROTAC IRAK4 degrader-6
PROTAC IRAK4 degrader-6 is a potent Cereblon-based compound designed to degrade interleukin-1 receptor-associated kinase...
T39901 PROTAC IRAK4 degrader-4 PROTAC IRAK4 degrader-4
PROTAC IRAK4 degrader-4 (US20190192668A1, compound I-127) is a Cereblon-based PROTAC specifically designed to target and...
T40073 PROTAC BRD4 Degrader-10 PROTAC BRD4 Degrader-10
PROTAC BRD4 Degrader-10, also known as compound 8b, is a dual ligand-based PROTAC that combines ligands for von Hippel-L...
T40334 PROTAC IRAK3 degrade-1 PROTAC IRAK3 degrade-1
PROTAC IRAK3 degrade-1 is a potent and selective degrader of IRAK3 ( IC 50 = 5 nM).
T39997 PROTAC CDK9 ligand-1 PROTAC CDK9 ligand-1
PROTAC CDK9 ligand-1 is a CDK9 ligand that can be used in the synthesis of PROTACs.
PROTAC BRD4 ligand-1
T12551
synonym:
Target:
PROTAC ERRα ligand 2
T5835
synonym:
Target:
PROTAC ERRα ligand 1
T15191
synonym:
Target:
Gefitinib-based PROTAC 3
T5437
synonym:
Target:
Homo-PROTAC pVHL30 degrader 1
T13722
synonym:
Target:
Homo-PROTAC cereblon degrader 1
T13721
synonym:
Target:
SMARCA-BD ligand 1 for Protac
T13848
synonym:
Target:
PROTAC BRAF-V600E degrader-1
T8745
synonym: Compound 23,Compound 23
Target:
SMARCA-BD ligand 1 for Protac dihydrochloride
T13890
synonym:
Target:
PROTAC-I
T34168
synonym: PROTAC I
Target:
PROTAC-12
T34167
synonym: PROTAC12,PROTAC 12
Target:
PROTAC IRAK4 degrader-3
T39920
synonym: PROTAC IRAK4 degrader-3
Target:
PROTAC BRD4 Degrader-5
T36242
synonym: PROTAC BRD4 Degrader-5
Target:
PROTAC BRD4 Degrader-15
T40074
synonym: PROTAC BRD4 Degrader-15
Target:
PROTAC IRAK4 degrader-5
T39902
synonym: PROTAC IRAK4 degrader-5
Target:
PROTAC IRAK4 degrader-6
T39903
synonym: PROTAC IRAK4 degrader-6
Target:
PROTAC IRAK4 degrader-4
T39901
synonym: PROTAC IRAK4 degrader-4
Target:
PROTAC BRD4 Degrader-10
T40073
synonym: PROTAC BRD4 Degrader-10
Target:
PROTAC IRAK3 degrade-1
T40334
synonym: PROTAC IRAK3 degrade-1
Target:
PROTAC CDK9 ligand-1
T39997
synonym: PROTAC CDK9 ligand-1
Target:
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