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PROTAC BRD9 Degrader-1

Name: PROTAC BRD9 Degrader-1
Brand: TargetMol
SKU: T12560
Rating: 4.5 (1 reviews)

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Catalog No. T12560Cas No. 2097971-01-0

PROTAC BRD9 Degrader-1 is a leading PROTAC BRD9 chemical degrader with an IC50 of 13.5 nM.

PROTAC BRD9 Degrader-1

😃Good

Catalog No. T12560Cas No. 2097971-01-0

PROTAC BRD9 Degrader-1 is a leading PROTAC BRD9 chemical degrader with an IC50 of 13.5 nM.

Pack Size	Price	Availability	Quantity
5 mg	$733	Backorder
10 mg	$1,219	Backorder

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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.

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Product Introduction

Bioactivity

Description	PROTAC BRD9 Degrader-1 is a leading PROTAC BRD9 chemical degrader with an IC50 of 13.5 nM.
Targets&IC50	BRD9:13.5 nM, BRD4:3.78 μM, CRBN-DDB1:48.9 nM
In vitro	PROTAC BRD9 Degrader-1 inhibits BRD9, BRD4, and CRBN-DDB1 (IC50s = 13.5 nM, 3.78 μM, and 48.9 nM, respectively)[1].

Chemical Properties

Molecular Weight	903.98
Formula	C₄₂H₄₅N₇O₁₂S₂
Cas No.	2097971-01-0
Relative Density.	1.56 g/cm3 (Predicted)

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 150 mg/mL (165.93 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	1.1062 mL	5.5311 mL	11.0622 mL	55.3110 mL
5 mM	0.2212 mL	1.1062 mL	2.2124 mL	11.0622 mL
10 mM	0.1106 mL	0.5531 mL	1.1062 mL	5.5311 mL
20 mM	0.0553 mL	0.2766 mL	0.5531 mL	2.7655 mL
50 mM	0.0221 mL	0.1106 mL	0.2212 mL	1.1062 mL
100 mM	0.0111 mL	0.0553 mL	0.1106 mL	0.5531 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc