Search Result

Search Results for " selectivity "

Targets

903

Compounds

Natural Products

Recombinant Proteins

Libraries

Cat No.	Product Name	Synonyms	Targets
T9339	Stafia-1		STAT
	Stafia-1 is a potent STAT5a inhibitor ( IC50=22.2 μM). Stafia-1 displays high selectivity over STAT5b and other STAT family members.		STAT
T11960	MBM-55		GSK-3 , MAPK , DYRK , Akt , Chk , Bcr-Abl , CDK , S6 Kinase , Aurora Kinase
	MBM-55 is an effective inhibitor of NIMA related kinase 2 (NEK2) with an IC50 of 1 nM. MBM-55 effectively inhibits the proliferation of cancer cells by inducing cell cycle arrest and apoptosis.
T9020	GSK620		Epigenetic Reader Domain
	GSK620 is a pan-BD2 inhibitor, which shows an anti-inflammatory phenotype in human whole blood with excellent broad selectivity, developability, and in vivo oral pharmacokinetics.GSK620 is highly selective for the BET-BD...		Epigenetic Reader Domain
T21331	SAR-020106		Chk
	SAR-020106 is a potent, ATP-competitive, and selective CHK1 inhibitor with an IC50 of 13.3 nmol/L on the isolated human enzyme.		Chk
T9470	HPK1-IN-7		MAPK
	HPK1-IN-7 is an orally active HPK1 inhibitor. It shows selectivity against IRAK4 (59 nM) and GLK (140 nM).		MAPK
T28628	RVX-297	RVX297	Epigenetic Reader Domain
	RVX-297 is a BD2 selective inhibitor of BET bromodomains. RVX-297 preferentially binds to the BD2 domains of the BET bromodomain and Extra Terminal (BET) family of protein.		Epigenetic Reader Domain
T11696	Ivachtin	Caspase-3 Inhibitor VII	Caspase
	Ivachtin (Caspase-3 Inhibitor VII) is a nonpeptide, noncompetitive and reversibl caspase-3 inhibitor(IC50 = 23 nM) and is a modest inhibitor of the remaining caspases.		Caspase
T4199	Desmethyl-VS-5584		PI3K , mTOR
	Desmethyl-VS-5584 is a dimethyl analog of VS-5584, which is a novel and highly selective PI3K/mTOR kinase inhibitor for the treatment of cancer.		PI3K , mTOR
T28352	PDE9-IN-(S)-C33	(S)-C33	PDE
	PDE9-IN-(S)-C33 ((S)-C33) is a potent and selective inhibitor of PDE9 (IC50 = 11 nM). PDE9-IN-(S)-C33 can be used for central nervous system diseases and diabetes research.		PDE
T5405	BI-1347		CDK
	BI-1347 is a potent, selective inhibitor of CDK8/cyclinC (IC50: 1 nM). It shows tumor growth inhibition in an in vivo xenograft model.		CDK
T15418	GS-6201	CVT-6883	Adenosine Receptor
	GS-6201 (CVT-6883) is a selective antagonist of adenosine A2B receptor. GS-6201 shows high affinity and selectivity for the human adenosine A2B receptors with a Ki of 22 nM.		Adenosine Receptor
T9564	IRE1α kinase-IN-1		IRE1
	IRE1α kinase-IN-1 is a highly selective IRE1α (ERN1) inhibitor, with an IC50 of 77 nM. It displays 100-fold selectivity for IRE1α over the IRE1β isoform. It inhibits ER stress-induced IRE1α oligomerization and autophosph...		IRE1
T1885	Siramesine hydrochloride	Lu 28-179 hydrochloride	Ferroptosis , Sigma receptor , lysosomal autophagy
	Siramesine hydrochloride (Lu 28-179 hydrochloride) is a selective sigma-2 receptor agonist, which has been shown to trigger cell death of Y cells and to exhibit a potent anticancer activity in vivo.		Ferroptosis , Sigma receptor , lysosomal autophagy
T6658	SB-408124		OX Receptor
	SB408124 is a non-peptide antagonist for OX1 receptor with Ki of 57 nM and 27 nM in both whole cell and membrane, respectively, exhibits 50-fold selectivity over OX2 receptor.		OX Receptor
T6493	Escitalopram Oxalate	Cipralex,(S)-(+)Citalopram oxalate	Others , 5-HT Receptor , Serotonin Transporter
	Escitalopram Oxalate ((S)-(+)Citalopram oxalate) is a selective serotonin (5-HT) reuptake inhibitor (SSRI) with Ki of 0.89 nM.		Others , 5-HT Receptor , Serotonin Transporter
T4620	Siramesine	Lu 28-179	Sigma receptor
	Siramesine (Lu 28-179)(Lu 28-179) is a selective sigma-2 receptor agonist, which has been shown to trigger cell death of cancer cells and to exhibit a potent anticancer activity in vivo.lysosome-destabilizing agent siram...		Sigma receptor
T39573	GSK251		PI3K
	GSK251 is a novel, orally bioavailable inhibitor of PI3Kδ, exhibiting high potency and selectivity, with a unique binding mode.		PI3K
T14547	JWG-071	JWG071,JWG 071	ERK , Epigenetic Reader Domain
	JWG-071, the first reported chemical probe for ERK5 kinase selectivity, is a BET-selective inhibitor with a 1 μM BRD4 IC that enhances both ERK5 activity and BRD4 selectivity.		ERK , Epigenetic Reader Domain
T6940	PHA-767491 hydrochloride	CAY10572,PHA-767491,PHA767491 HCl,CAY-10572 hydrochloride	Apoptosis , GSK-3 , CDK
	PHA-767491 hydrochloride (CAY-10572 hydrochloride) is an effective ATP-competitive dual Cdc7/CDK9 inhibitor (IC50: 10/34 nM). It has ~20-fold selectivity against GSK3-β and CDK1/2, 50-fold selectivity against CDK5 and MK...		Apoptosis , GSK-3 , CDK
T14947	CHDI-390576		HDAC
	CHDI-390576 is a CNS penetrant class IIa HDAC inhibitor (IC50s: 54 nM, 60 nM, 31 nM, 50 nM for class IIa HDAC4, HDAC5, HDAC7, HDAC9). It shows >500-fold selectivity over class I HDACs (1, 2, 3) and ~150-fold selectivity ...		HDAC
T10277	AL 8697		p38 MAPK
	AL 8697 is a selective p38α MAPK inhibitor (IC50 = 6 nM) with 14-fold selectivity over p38β (IC50 = 82 nM) and 300-fold selectivity over a panel of 91 kinases. AL 8697 has anti-inflammatory activity.		p38 MAPK
T19671	AZ31	AZ 31,AZ-31	ATM/ATR
	AZ31 is an ATM inhibitor with potency, high selectivity, and oral activity.AZ31 inhibits ATM enzymes, intracellular ATM, with IC50 values of <1.2 nM and 46 nM, respectively.AZ31 exhibits excellent ATR selectivity, PIKK f...		ATM/ATR
T10778	CGP 20712 A	CGP 20712 mesylate	Adrenergic Receptor
	CGP 20712 A (CGP 20712 mesylate) is a highly selective antagonist of β1-adrenoceptor (IC50: 0.7 nM). It shows ~10,000-fold selectivity over β2-adrenoceptors.		Adrenergic Receptor
T2435	EPZ011989		Histone Methyltransferase
	EPZ011989 is a effective, specific orally bioavailable EZH2 inhibitor with Ki < 3 nM for EZH2 Y646 and EZH2 wt; 15-fold selectivity over EZH1 and >3000-fold selectivity over other HMTase.		Histone Methyltransferase
T2356	Ro-3306		Apoptosis , ERK , SGK , PKA , CDK , PKC
	RO-3306 is a selectivity ATP-competitive CDK1 inhibitor (Ki: 20 nM). The selectivity of RO-3306 for CDK1 is >15-fold higher than a diverse panel of human kinases.		Apoptosis , ERK , SGK , PKA , CDK , PKC
T6286	RGFP966 (E-isomer)		HDAC
	RGFP966 is an HDAC3 inhibitor with IC50 of 0.08 μM, exhibits > 200-fold selectivity over other HDAC.		HDAC
T26109	Robenacoxib	Onsior	COX
	Robenacoxib (Onsior) is a non-steroidal compound with strong selectivity for cyclooxygenase-2 and anti-inflammatory activity.		COX
T3049	TPCA-1	GW683965,IKK2 Inhibitor IV,TPCA1	Apoptosis , IκB/IKK , STAT
	TPCA-1 (TPCA1) is an effective and specific IKK-2 inhibitor (IC50: 17.9 nM); shows >22-fold selectivity over IKK-1 and >550-fold selectivity over others kinases and enzymes.		Apoptosis , IκB/IKK , STAT
T6054	GSK256066		PDE
	GSK256066 is a selective PDE4B(equal affinity to isoforms A-D) inhibitor with IC50 of 3.2 pM, >380, 000-fold selectivity versus PDE1/2/3/5/6 and >2500-fold selectivity against PDE4B versus PDE7.Phase 2.		PDE
T6064	UK-383367	UK 383367	Procollagen C Proteinase
	UK-383367 is a procollagen C-proteinase inhibitor with IC50 of 44 nM, has excellent selectivity over MMPs.		Procollagen C Proteinase
T21703	4-Chlorophenylguanidine hydrochloride		Others
	4-Chlorophenylguanidine hydrochloride is a potent inhibitor of urokinase selectivity.		Others
T1830	BX795		IκB/IKK , Chk , CDK , c-Kit , PDK , Autophagy
	BX795 is an effective and selective PDK1 inhibitor (IC50: 6 nM), and its selectivity is 140- and 1600-fold for PDK1 over PKA and PKC in cell-free assays, respectively. Meanwhile, the selectivity for PDK1 is 100-fold than...		IκB/IKK , Chk , CDK , c-Kit , PDK , Autophagy
T22990	ML-090	Fluoflavine	NADPH-oxidase , Others
	ML-090 is NOX1-specific inhibitor(IC50 = 90 nM) which is >100 selectivity for NOX1 over NOX2, NOX3, NOX4 (all IC50s >10 μM).		NADPH-oxidase , Others
T6378	AMG-458	AMG 458	c-Met/HGFR
	AMG-458 is a potent c-Met inhibitor with Ki of 1.2 nM, ~350-fold selectivity for c-Met than VEGFR2 in cells.		c-Met/HGFR
T13312L	Seviteronel	VT-464	Others
	Seviteronel is an effective CYP17 lyase inhibitor (h-Lyase IC50=69 nM). In a hamster model of androgen biosynthesis inhibition, it demonstrated both exceptional in vitro lyase/hydroxylase selectivity (~10-fold) and oral...		Others
T19917	Gepirone		5-HT Receptor
	Gepirone is a 5-HT1A receptor agonist belonging to the buspirone family. Gepirone HCl possesses greater selectivity for the 5-HT1A receptor than SSRIs.		5-HT Receptor
T36287	Pirtobrutinib		BTK
	Pirtobrutinib (LOXO-305) is an advanced BTK inhibitor that displays high selectivity and operates through a non-covalent mechanism. This compound effectively inhibits various BTK C481 substitution mutations, leading to t...		BTK
T16936	SS-208		HDAC
	SS-208 is a selective inhibitor of HDAC6 (IC50 = 12 nM) with anti-tumor activity. SS-208 shows selectivity over other HDAC subtypes.		HDAC
T68134	Ro-3201195		p38 MAPK
	Ro-3201195 is a novel orally available p38 MAPK inhibitor with high selectivity.		p38 MAPK
T8651	CAL-101	(S)-2-(1-(9H-Purin-6-ylamino)ethyl)-5-fluoro-3-phenylquinazolin-4(3H)-one,GS-1101,Idelalisib	PI3K
	CAL-101 (Idelalisib) is a selective inhibitor of p110δ(IC50 : 2.5 nM; in cell-free assays); shown to have 40- to 300-fold greater selectivity for p110δ than p110α/β/γ, and 400- to 4000-fold more selectivity to p110δ than...		PI3K
T16777	ROC-325		Apoptosis , Autophagy
	ROC-325 is an effective and orally active inhibitor of autophagy with anticancer activity. ROC-325 induces renal cell carcinoma apoptosis and exhibits favorable selectivity.		Apoptosis , Autophagy
T6306	Erteberel	LY500307	Estrogen Receptor/ERR , Estrogen/progestogen Receptor
	Erteberel (LY500307) is a potent, selective estrogen receptor β agonist with EC50 of 0.66 nM, 32-fold selectivity against estrogen receptor α. Phase 2.		Estrogen Receptor/ERR , Estrogen/progestogen Receptor
T5503	IPSU		OX Receptor
	IPSU is an antagonist of OX2 receptor. IPSU Exhibits approximately six-fold selectivity for OX2 versus OX1 receptors.		OX Receptor
T6358	1-Azakenpaullone	azakenpaullone	GSK-3
	1-Azakenpaullone (azakenpaullone) is a potent and selective GSK-3β inhibitor with IC50 of 18 nM, >100-fold selectivity over CDK1/cyclin B and CDK5/p25.		GSK-3
T36631	BAY-6035		MEK , Histone Methyltransferase
	BAY-6035 is an inhibitor of SET and MYND domain-containing protein 3 (SMYD3). BAY-6035 has more than 100-fold selectivity over other histone methyltransferases.		MEK , Histone Methyltransferase
T6757	AMG319		PI3K
	AMG319 is a potent and selective PI3Kδ inhibitor with IC50 of 18 nM, >47-fold selectivity over other PI3Ks. Phase 2.		PI3K
T6578	ME0328		PARP
	ME0328 is a potent and selective PARP inhibitor with IC50 of 0.89 μM for PARP3, about 7-fold selectivity over PARP1.		PARP
T6774	AZD-8835	AZD8835	PI3K
	AZD-8835 is a mixed inhibitor of PI3Kα/δ (IC50: 6.2/5.7 nM), also with selectivity against PI3Kβ/γ (IC50: 431/90 nM).		PI3K
T16803	RS 8359		MAO
	RS 8359 is a reversible inhibitor of monoamine oxidase A (MAO-A) with a selectivity ratio of about 2200 for the A:B enzyme types. RS 8359 has antidepressant activity.		MAO
T6655	SB-269970 hydrochloride	SB-269970A,SB269970 HCl	5-HT Receptor
	SB-269970 hydrochloride (SB-269970A) , a hydrochloride salt form of SB-269970, is a 5-HT7 receptor antagonist (pKi of 8.3) and exhibits >50-fold selectivity against other receptors.		5-HT Receptor

Compounds

Target: GSK-3, MAPK, DYRK, Akt, Chk, Bcr-Abl, CDK, S6 Kinase, Aurora Kinase

GSK620

T9020

Synonym:

Target: Epigenetic Reader Domain

Target: Epigenetic Reader Domain

Ivachtin

T11696

Synonym: Caspase-3 Inhibitor VII

Target: Adenosine Receptor

Siramesine hydrochloride

T1885

Synonym: Lu 28-179 hydrochloride

Target: Ferroptosis, Sigma receptor, lysosomal autophagy

Synonym: Cipralex,(S)-(+)Citalopram oxalate

Target: Others, 5-HT Receptor, Serotonin Transporter

Siramesine

T4620

Synonym: Lu 28-179

Target: Sigma receptor

Synonym: JWG071,JWG 071

Target: ERK, Epigenetic Reader Domain

PHA-767491 hydrochloride

T6940

Synonym: CAY10572,PHA-767491,PHA767491 HCl,CAY-10572 hydrochloride

Target: Apoptosis, GSK-3, CDK

Synonym: CGP 20712 mesylate

Target: Adrenergic Receptor

EPZ011989

T2435

Synonym:

Target: Histone Methyltransferase

Ro-3306

T2356

Synonym:

Target: Apoptosis, ERK, SGK, PKA, CDK, PKC

Synonym: GW683965,IKK2 Inhibitor IV,TPCA1

Target: Apoptosis, IκB/IKK, STAT

Target: Procollagen C Proteinase

4-Chlorophenylguanidine hydrochloride

Target: IκB/IKK, Chk, CDK, c-Kit, PDK, Autophagy

ML-090

T22990

Synonym: Fluoflavine

Target: NADPH-oxidase, Others

Target: 5-HT Receptor

Synonym: (S)-2-(1-(9H-Purin-6-ylamino)ethyl)-5-fluoro-3-phenylquinazolin-4(3H)-one,GS-1101,Idelalisib

Target: Apoptosis, Autophagy

Erteberel

T6306

Synonym: LY500307

Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor

Synonym: azakenpaullone

Target: MEK, Histone Methyltransferase

SB-269970 hydrochloride

T6655

Synonym: SB-269970A,SB269970 HCl

Target: 5-HT Receptor

Cat No.	Product Name	Synonyms	Targets
T0185	Escitalopram	Seroplex,S-(+)-Citalopram,(S)-Citalopram	Dopamine Receptor , 5-HT Receptor , Serotonin Transporter , Adrenergic Receptor , AChR , Norepinephrine , Histamine Receptor
	Escitalopram (Seroplex) is a furancarbonitrile that is one of the SEROTONIN UPTAKE INHIBITORS used as an antidepressant. The drug is also effective in reducing ethanol uptake in alcoholics and is used in depressed patien...
T2826	Asaraldehyde	Asarylaldehyde,2,4,5-trimethoxy-Benzaldehyde,Asaronaldehyde	COX
	Asaraldehyde (2,4,5-trimethoxy-Benzaldehyde), a natural COX-2 inhibitor, exhibits 17-fold selectivity than COX-1.		COX
T3S1251	Neoruscogenin		ROR
	1. Neoruscogenin represents a universal pharmacological tool for RORα research due to its specific selectivity profile versus other nuclear receptors.		ROR
T7472	7-Hydroxyflavone		P450
	7-Hydroxyflavone is a potent inhibitor of CYP1A1 with a Ki value of 0.015 μM and exhibits 6-fold greater selectivity for CYP1A1 over CYP1A2.with anti-inflammatory activity		P450
T6512	G-418 disulfate	Geneticin,G418 Sulfate,Antibiotic G-418 sulfate,Geneticin sulfate	Antibacterial , Antibiotic
	G-418 disulfate (Geneticin sulfate) is an aminoglycoside antibiotic, an inhibitor of protein synthesis with eukaryotic selectivity. G-418 disulfate blocks peptide synthesis by inhibiting peptide chain elongation.		Antibacterial , Antibiotic
T0665	Xanthine	2,6-Dihydroxypurine,Isoxanthine	Endogenous Metabolite , Adenosine Receptor
	Xanthine (Isoxanthine) is a product on the pathway of purine degradation. Xanthine is subsequently converted to uric acid by the action of the Xanthine oxidase enzyme. Xanthine is found in most body tissues and fluids in...		Endogenous Metabolite , Adenosine Receptor
T11041	Dihydro-β-erythroidine hydrobromide	DHβE hydrobromide	Others
	Dihydro-β-erythroidine hydrobromide(DHβE) is a potent, oral active and competitive antagonist of neuronal nicotinic acetylcholine receptors (nAChRs). Dihydro-β-carotene hydrobromide showed selectivity to α4β4 and α4β2nAC...		Others
TN4788	Pierreione B		mTOR
	Pierreione B is an inhibitor of mTOR signaling with strong anticancer activity. Pierreione A and Pierreione B demonstrate solid tumor selectivity with minimal cytotoxicity.		mTOR
T74005	Urolithin D
	Urolithin D acts as a competitive and reversible antagonist for EphA receptors, displaying selectivity within its class [1].
TN1852	Lancifodilactone F		HIV Protease
	Lancifodilactone F exerts minimal cytotoxicity against C8166 cells (CC50 > 200 microg/mL) and shows anti-HIV activity with EC50 = 20.69 +/- 3.31 microg/mL and a selectivity index > 6.62.		HIV Protease
TN2360	Falcarinol	Falcarinol,Panaxynol	HSP
	Falcarinol, also known as Panaxynol, is a naturally occurring compound that acts as an orally active inhibitor of Hsp90. It effectively targets both the N-terminal and C-terminal regions of Hsp90, displaying high selecti...		HSP
TN3428	Aphadilactone C		Others
	Aphadilactone C shows significant antimalarial activity with the IC50 value of 170 ± 10 nM. It shows potent and selective inhibition against the diacylglycerol O-acyltransferase-1 (DGAT-1) enzyme (IC50 = 0.46 ± 0.09 uM, ...		Others
T36303	Psammaplin A
	Psammaplin A, a marine metabolite, functions as a robust inhibitor of HDAC and DNA methyltransferases, displaying notable potency and selectivity as a DAC1 inhibitor, with an IC50 value of 0.9 nM. It exhibits antimicrobi...
T75651	Rivulariapeptolides 988
	Rivulariapeptolides 988 demonstrates significant potency and selectivity as a serine protease inhibitor, exhibiting IC50 values of 95.46 nM for chymotrypsin, 15.29 nM for elastase, and 85.50 nM for proteinase K [1].
T75630	Ganoderic acid Mf
	Ganoderic acid Mf, an antitumor triterpenoid, selectively induces apoptosis in cancer cells through a mitochondria-mediated pathway while demonstrating high selectivity between normal and cancer cells. It also arrests th...
T72802	Spongionellol A
	Spongionellol A, an inhibitor of MDR1 (p-glycoprotein), exhibits significant cytotoxicity and selectivity towards prostate cancer cells through the induction of caspase-dependent apoptosis. This compound is valuable for ...
T79975	Dihydrodehydrodiconiferyl alcohol 9-O-α-L-rhamnopyranoside		HBV
	Dihydrodehydrodiconiferyl alcohol 9-O-α-L-rhamnopyranoside (Compound 1), a lignan with anti-HBV activity, exhibits selectivity by targeting the HBV surface antigen (HBsAg) with an IC50 of 0.58 mM, whereas its activity ag...		HBV
T73072	PTP1B-IN-20
	PTP1B-IN-20 is a selective PTP1B (protein tyrosine phosphatase 1B) inhibitor, exhibiting an IC50 of 1.05 μM, and demonstrates selectivity over TCPTP (T-cell protein tyrosine phosphatase), which has an IC50 of 78.0 μM. Th...
T82031	Isoguaiacin
	Isoguaiacin, a natural product [1], exhibits (hass) the potential to be (to exist as) an (a) effective pharmacological agent due to its (its) ability to inhibit (the inhibition of) mushroom tyrosinase. This (The) inhibit...
T75436	Jatrorrhizine hydroxide
	Jatrorrhizine hydroxide, an alkaloid derived from Coptis chinensis, exhibits a range of biological activities including neuroprotective, antimicrobial, antiplasmodial, and antioxidant properties [1]. It acts as a potent ...
T83913	Mitraciliatine
	Mitraciliatine, an alkaloid discovered in M. speciosa (Kratom in Thai), acts as a partial agonist for the μ-opioid receptor (MOR) and an agonist for the κ-opioid receptor (KOR), demonstrating selectivity for these recept...
T37876	Fengycin
	Fengycin, a cyclic lipopeptide, functions as an agricultural fungicide by exhibiting an anti-fungal infection effect through damaging the target's cell membrane[1].

Natural Products

Escitalopram

T0185

Synonym: Seroplex,S-(+)-Citalopram,(S)-Citalopram

Target: Dopamine Receptor, 5-HT Receptor, Serotonin Transporter, Adrenergic Receptor, AChR, Norepinephrine, Histamine Receptor

Asaraldehyde

T2826

Synonym: Asarylaldehyde,2,4,5-trimethoxy-Benzaldehyde,Asaronaldehyde

Synonym: Geneticin,G418 Sulfate,Antibiotic G-418 sulfate,Geneticin sulfate

Target: Antibacterial, Antibiotic

Xanthine

T0665

Synonym: 2,6-Dihydroxypurine,Isoxanthine

Target: Endogenous Metabolite, Adenosine Receptor

Dihydro-β-erythroidine hydrobromide

T11041

Synonym: DHβE hydrobromide

Synonym: Falcarinol,Panaxynol

Rivulariapeptolides 988

Dihydrodehydrodiconiferyl alcohol 9-O-α-L-rhamnopyranoside

Jatrorrhizine hydroxide

Recombinant Proteins

Species：

Expression System：

Tag：

Cat No.	Product Name	Species	Expression System
TMPY-02975	CANT1 Protein, Human, Recombinant (hFc)	Human	HEK293
	CANT1(calcium activated nucleotidase 1) belongs to the apyrase family. Apyrase is a calcium-activated plasma membrane-bound enzyme (magnesium can also activate it) (EC 3.6.1.5) that catalyses the hydrolysis of ATP to yie...
TMPY-02710	CANT1 Protein, Human, Recombinant (His)	Human	HEK293
	CANT1(calcium activated nucleotidase 1) belongs to the apyrase family. Apyrase is a calcium-activated plasma membrane-bound enzyme (magnesium can also activate it) (EC 3.6.1.5) that catalyses the hydrolysis of ATP to yie...
TMPJ-00922	DCK Protein, Human, Recombinant (His & T7)	Human	E. coli
	Deoxycytidine Kinase (DCK) is a member of the DCK/DGK family. DCK exists as a homodimer and is localized to the nucleus. DCK is required for the phosphorylation of the deoxyribonucleosides deoxycytidine (dC), deoxyguanos...
TMPJ-01001	CCL11 Protein, Human, Recombinant	Human	E. coli
	C-C Motif Chemokine 11 (CCL11) is a secreted protein that belongs to the intercrine beta (chemokine CC) family. In response to the presence of allergens, CCL11 selectively recruits eosinophils, a prominent feature of all...
TMPY-01891	ECE2 Protein, Human, Recombinant (His)	Human	HEK293
	Endothelin-converting enzyme 2, also known as ECE-2, is a metalloprotease that possesses many properties consistent with it being a neuropeptide-processing enzyme. Endothelin-converting enzymes (ECEs) are the key enzy...
TMPY-00782	ECE2 Protein, Human, Recombinant (hFc)	Human	HEK293
	Endothelin-converting enzyme 2, also known as ECE-2, is a metalloprotease that possesses many properties consistent with it being a neuropeptide-processing enzyme. Endothelin-converting enzymes (ECEs) are the key enzy...
TMPH-02301	VPS35 Protein, Human, Recombinant (His & Myc)	Human	E. coli
	Acts as component of the retromer cargo-selective complex (CSC). The CSC is believed to be the core functional component of retromer or respective retromer complex variants acting to prevent missorting of selected transm...
TMPH-00818	Delta-theraphotoxin-Hm1a Protein, Heteroscodra maculata, Recombinant (His & Myc & SUMO)	Heteroscodra maculata	E. coli
	Gating-modifier toxin that potently inhibits inactivation of the mammalian Nav1.1/SCN1A sodium channel (EC(50)=38 nM). Also moderately inhibits inactivation of Nav1.2/SCN2A (EC(50)=236 nM) and Nav1.3/SCN3A (EC(50)=220 nM...

CANT1 Protein, Human, Recombinant (hFc)

TMPY-02975

Species: Human

Expression System: HEK293

CANT1 Protein, Human, Recombinant (His)

TMPY-02710

Species: Human

Expression System: HEK293

DCK Protein, Human, Recombinant (His & T7)

TMPJ-00922

Species: Human

Expression System: E. coli

CCL11 Protein, Human, Recombinant

TMPJ-01001

Species: Human

Expression System: E. coli

ECE2 Protein, Human, Recombinant (His)

TMPY-01891

Species: Human

Expression System: HEK293

ECE2 Protein, Human, Recombinant (hFc)

TMPY-00782

Species: Human

Expression System: HEK293

VPS35 Protein, Human, Recombinant (His & Myc)

TMPH-02301

Species: Human

Expression System: E. coli

Delta-theraphotoxin-Hm1a Protein, Heteroscodra maculata, Recombinant (His & Myc & SUMO)

TMPH-00818

Species: Heteroscodra maculata

Expression System: E. coli

Cat No.	Product Name
L9411	Cysteine Covalent Library	72 compounds
	The cysteine covalent library contains 72 compounds.
L2152	Targeted Therapy Drug Library	121 compounds
	121 tumor-targeted drugs that can be used for high-throughput and high-content screening.
L9610	Cyclic Peptide Library	58 compounds
	58 species of cyclic peptide molecules for high-throughput and high-content screening;
L7400	Sodium Channel Blocker Library	128 compounds
	A unique collection of 128 sodium channel blockers and agonists for high throughput and high content screening;
L9600	Peptide Compound Library	800 compounds
	800 peptides can be used in peptide drug development and signaling transduction and mechanism study;

Libraries

Cysteine Covalent Library

L9411

Compounds: 72

Targeted Therapy Drug Library

L2152

Compounds: 121

Cyclic Peptide Library

L9610

Compounds: 58

Sodium Channel Blocker Library

L7400

Compounds: 128

Peptide Compound Library

L9600

Compounds: 800