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UFP-101 acetate

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Catalog No. TP2105L
Alias UFP-101 acetate(849024-68-6 free base)

UFP-101 acetate is a selective and competitive antagonist of the NOP receptor (pKi = 10.24) with >3000-fold selectivity over δ, μ, and κ opioid receptors.

UFP-101 acetate
Other Forms of UFP-101 acetate:

UFP-101 acetate

🥰Excellent
Purity: 95.92%
Catalog No. TP2105LAlias UFP-101 acetate(849024-68-6 free base)
UFP-101 acetate is a selective and competitive antagonist of the NOP receptor (pKi = 10.24) with >3000-fold selectivity over δ, μ, and κ opioid receptors.
Pack SizePriceUSA WarehouseGlobal WarehouseQuantity
1 mg$317-In Stock
2 mg$573-In Stock
5 mg$897-In Stock
10 mg$1,230-In Stock
25 mg$1,820-In Stock
50 mg$2,460-In Stock
100 mg$3,290-In Stock
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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]
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Purity:95.92%
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COA HPLC MS

Product Introduction

Bioactivity
Description
UFP-101 acetate is a selective and competitive antagonist of the NOP receptor (pKi = 10.24) with >3000-fold selectivity over δ, μ, and κ opioid receptors.
In vivo
In mice submitted to the forced swimming test, UFP-101 acetate elicits a pronounced acute and dose-dependent antidepressant-like effect[2].
SynonymsUFP-101 acetate(849024-68-6 free base)
Chemical Properties
Molecular Weight1968.23
FormulaC84H142N32O23
SmilesCC(O)=O.O=C(N)[C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC(CNC([C@@H](NC([C@@H](NC(CNC(CNC(CNCC1=CC=CC=C1)=O)=O)=O)CC2=CC=CC=C2)=O)[C@H](O)C)=O)=O)C)=O)CCCNC(N)=N)=O)CCCCN)=O)CO)=O)C)=O)CCCNC(N)=N)=O)CCCCN)=O)CCCNC(N)=N)=O)CCCCN)=O)CC(N)=O)=O)CCC(N)=O
Relative Density.no data available
SequenceGly-Gly-Gly-Phe-Thr-Gly-Ala-Arg-Lys-Ser-Ala-Arg-Lys-Arg-Lys-Asn-Gln
Sequence ShortGGGFTGARKSARKRKNQ
Storage & Solubility Information
Storagekeep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
Solubility Information
H2O: 83.3 mg/mL (42.32 mM), Sonication is recommended.
Solution Preparation Table
H2O
1mg5mg10mg50mg
1 mM0.5081 mL2.5404 mL5.0807 mL25.4035 mL
5 mM0.1016 mL0.5081 mL1.0161 mL5.0807 mL
10 mM0.0508 mL0.2540 mL0.5081 mL2.5404 mL
20 mM0.0254 mL0.1270 mL0.2540 mL1.2702 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
TargetMol | Animal experimentsFor example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH2O. So your working solution concentration is 2 mg/mL。
Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH2OTargetMol | reagent mix well and clarify
For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.
1 Enter information below:
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2 Enter the in vivo formulation:
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Keywords

UFP-101 AcetateUFP101 acetateUFP101 AcetateUFP 101 AcetateUFP 101 acetateOpioidReceptorOpioid ReceptorNOP receptor
Related Tags: buy UFP-101 acetate | purchase UFP-101 acetate | UFP-101 acetate cost | order UFP-101 acetate | UFP-101 acetate chemical structure | UFP-101 acetate in vivo | UFP-101 acetate formula | UFP-101 acetate molecular weight
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