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AChR

An acetylcholine receptor (abbreviated AChR) is an integral membrane protein that responds to the binding of acetylcholine, a neurotransmitter.
Cat. No. Product name CAS No. Purity Chemical Structure
T13772 MHP 133 147340-43-0 98%
MHP 133 is a drug with multiple CNS targets(AChE with Ki of 69 μM).
T10914 Cyclodrine hydrochloride 78853-39-1 98%
Cyclone hydrochloride is a cholinergic (muscarinic, nicotinic) (mAChR and nAChR) receptor antagonist.
T5476 MAChr-in-1 119391-56-9 98%
mAChR-IN-1 is muscarinic cholinergic receptor(mAChR) antagonist (IC50=17 nM).
T12446 Phenserine 101246-66-6 98%
Phenserine is a derivative of Physostigmine and is annoncompetitive, long-acting and selective inhibitor of AChE.
T10731 CDD0102 146422-58-4 98%
CDD0102 is a potent agonist of M1 Muscarinic receptor.
TN1409 Asimilobine 6871-21-2 98%
(-)-Asimilobine shows antioxidative, anti-acetylcholinesterase (AChE), anti-α±-glucosidase, anti-leishmanial and anti-fungal activities; it displays weak inhibit...
T1484 Perindoprilat 95153-31-4 98%
Perindoprilat is an angiotensin-converting enzyme inhibitor.
T12868 Sch412348 377727-26-9 98%
Sch412348 is a potent competitive the human adenosine A2A receptor antagonist with Ki of 0.6 nM and has >1000-fold selectivity over all other adenosine receptors...
TN4456 Lucidadiol 252351-95-4 98%
Lucidadiol exhibits butyrylcholinesterase-inhibitory activity at concentrations up to 200 uM, it also possesses inhibitory activity against acetylcholinesterase ...
T13256 UP202-56 163838-04-8 98%
UP202-56 is an adenosinergic agonist and is an adenosine analog.
T16417 Oxitropium Bromide 30286-75-0 98%
Oxitropium bromide is a mAChR antagonist. It is used as an anticholinergic bronchodilator drug for the treatment of asthma and chronic obstructive pulmonary dise...
TN4812 Pluviatolide 28115-68-6 98%
(-)-Pluviatolide can inhibit electrically-induced and acetylcholine-induced contraction in the isolated guinea-pig ileum.
TN2504 1,5-Dihydroxyxanthone 14686-65-8 98%
1,5-Dihydroxyxanthone exhibits the epidermal growth factor receptor (EGFR) -tyrosine kinase inhibitory activity, with the IC50 value of 90.34 nM. It may have ant...
T19623 α-Muricholic acid 2393-58-0 98%
α-Muricholic acid is the most abundant primary bile acid in rodents.
T12191 NBTGR 13153-27-0 98%
NBTGR is a potent nucleoside transport inhibitor(adenosine uptake ,Ki of 70 nM).
T12525 Pozanicline dihydrochloride 161416-61-1 98%
Pozanicline dihydrochloride is an orally bioavailable agonist of nicotinic acetylcholine receptor (nAChR) (Ki of 16.7 nM)
TN2067 Picfeltarraegenin X 1391826-61-1 98%
Picfeltarraenin X shows stronger AChE inhibition than the known AChE inhibitor Tacrine.
TN3875 Dipterocarpol 471-69-2 98%
Dipterocarpol is a dammarane-type triterpenoid, as are the major bioactive compounds of ginseng. Dipterocarpol A shows moderate acetylcholinesterase inhibitory a...
T16563 Pozanicline 161417-03-4 98%
Pozanicline reverses nicotine withdrawal-induced cognitive deficits, may be an effective component of novel therapeutic strategies for nicotine addiction. Pozani...
TN3744 Cyclomorusin 62596-34-3 98%
Cyclomorusin exhibits competitive inhibition toward monophenolase activity of mushroom tyrosinase, the IC50 value of 0.092 microM. It evokes the stimulation of s...
MHP 133
T13772
MHP 133 is a drug with multiple CNS targets(AChE with Ki of 69 μM).
Cyclodrine hydrochloride
T10914
Cyclone hydrochloride is a cholinergic (muscarinic, nicotinic) (mAChR and nAChR) receptor antagonist.
mAChr-in-1
T5476
mAChR-IN-1 is muscarinic cholinergic receptor(mAChR) antagonist (IC50=17 nM).
Phenserine
T12446
Phenserine is a derivative of Physostigmine and is annoncompetitive, long-acting and selective inhibitor of AChE.
CDD0102
T10731
CDD0102 is a potent agonist of M1 Muscarinic receptor.
Asimilobine
TN1409
(-)-Asimilobine shows antioxidative, anti-acetylcholinesterase (AChE), anti-α±-glucosidase, anti-leishmanial and anti-fungal activities; it displays weak inhibit...
Perindoprilat
T1484
Perindoprilat is an angiotensin-converting enzyme inhibitor.
Sch412348
T12868
Sch412348 is a potent competitive the human adenosine A2A receptor antagonist with Ki of 0.6 nM and has >1000-fold selectivity over all other adenosine receptors...
Lucidadiol
TN4456
Lucidadiol exhibits butyrylcholinesterase-inhibitory activity at concentrations up to 200 uM, it also possesses inhibitory activity against acetylcholinesterase ...
UP202-56
T13256
UP202-56 is an adenosinergic agonist and is an adenosine analog.
Oxitropium Bromide
T16417
Oxitropium bromide is a mAChR antagonist. It is used as an anticholinergic bronchodilator drug for the treatment of asthma and chronic obstructive pulmonary dise...
Pluviatolide
TN4812
(-)-Pluviatolide can inhibit electrically-induced and acetylcholine-induced contraction in the isolated guinea-pig ileum.
1,5-Dihydroxyxanthone
TN2504
1,5-Dihydroxyxanthone exhibits the epidermal growth factor receptor (EGFR) -tyrosine kinase inhibitory activity, with the IC50 value of 90.34 nM. It may have ant...
α-Muricholic acid
T19623
α-Muricholic acid is the most abundant primary bile acid in rodents.
NBTGR
T12191
NBTGR is a potent nucleoside transport inhibitor(adenosine uptake ,Ki of 70 nM).
Pozanicline dihydrochloride
T12525
Pozanicline dihydrochloride is an orally bioavailable agonist of nicotinic acetylcholine receptor (nAChR) (Ki of 16.7 nM)
Picfeltarraegenin X
TN2067
Picfeltarraenin X shows stronger AChE inhibition than the known AChE inhibitor Tacrine.
Dipterocarpol
TN3875
Dipterocarpol is a dammarane-type triterpenoid, as are the major bioactive compounds of ginseng. Dipterocarpol A shows moderate acetylcholinesterase inhibitory a...
Pozanicline
T16563
Pozanicline reverses nicotine withdrawal-induced cognitive deficits, may be an effective component of novel therapeutic strategies for nicotine addiction. Pozani...
Cyclomorusin
TN3744
Cyclomorusin exhibits competitive inhibition toward monophenolase activity of mushroom tyrosinase, the IC50 value of 0.092 microM. It evokes the stimulation of s...
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