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3-Bromocytisine

🥰Excellent
Catalog No. T10108Cas No. 207390-14-5
Alias 3-Br-cytisine, (-)-9-Bromocytisine, (-)-3-Bromocytisine

3-Bromocytisine ((-)-3-Bromocytisine) is an effective agonist of nAChR (IC50s: 0.28, 0.30 and 31.6 nM for hα4β4, hα4β2, and hα7).

3-Bromocytisine

3-Bromocytisine

🥰Excellent
Purity: 99.974%
Catalog No. T10108Alias 3-Br-cytisine, (-)-9-Bromocytisine, (-)-3-BromocytisineCas No. 207390-14-5
3-Bromocytisine ((-)-3-Bromocytisine) is an effective agonist of nAChR (IC50s: 0.28, 0.30 and 31.6 nM for hα4β4, hα4β2, and hα7).
Pack SizePriceAvailabilityQuantity
1 mg$92In Stock
5 mg$225In Stock
10 mg$325In Stock
25 mg$548In Stock
50 mg$788In Stock
100 mg$1,080In Stock
200 mg$1,450In Stock
1 mL x 10 mM (in DMSO)$198In Stock
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This molecule is a custom-made product. TargetMol has an excellent synthesis team with the experience and capability to provide you with cost-effective products. However, due to objective factors, there is a small probability that the synthesis may not be successful during the R&D process. We appreciate your understanding. If you have any questions, please feel free to contact us. We are committed to serving you wholeheartedly.
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Purity:99.974%
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COA HNMR LCMS

Product Introduction

Bioactivity
Description
3-Bromocytisine ((-)-3-Bromocytisine) is an effective agonist of nAChR (IC50s: 0.28, 0.30 and 31.6 nM for hα4β4, hα4β2, and hα7).
Targets&IC50
α7 (human):31.6 nM , α4β4 (human):0.28 nM , α4β2 (human):0.30 nM
In vitro
3-Bromocytisine shows different effects on high and low ACh sensitivity α4β2 nAChRs with EC50s are 8 and 50 nM, respectively [2].
Synonyms3-Br-cytisine, (-)-9-Bromocytisine, (-)-3-Bromocytisine
Chemical Properties
Molecular Weight269.14
FormulaC11H13BrN2O
Cas No.207390-14-5
SmilesO=C1N2C([C@@]3(C[C@](C2)(CNC3)[H])[H])=CC=C1Br
Relative Density.1.61 g/cm3 (Predicted)
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
Solubility Information
DMSO: 50 mg/mL (185.78 mM), Sonication is recommended.
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM3.7155 mL18.5777 mL37.1554 mL185.7769 mL
5 mM0.7431 mL3.7155 mL7.4311 mL37.1554 mL
10 mM0.3716 mL1.8578 mL3.7155 mL18.5777 mL
20 mM0.1858 mL0.9289 mL1.8578 mL9.2888 mL
50 mM0.0743 mL0.3716 mL0.7431 mL3.7155 mL
100 mM0.0372 mL0.1858 mL0.3716 mL1.8578 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
TargetMol | Animal experimentsFor example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH2O. So your working solution concentration is 2 mg/mL。
Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH2OTargetMol | reagent mix well and clarify
For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.
1 Enter information below:
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2 Enter the in vivo formulation:
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Dose Conversion

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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc

Keywords

nAChR9-Bromocytisine3-Bromocytisine
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