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SR 16584

Name: SR 16584
Brand: TargetMol
SKU: T23388
Price: 120 USD
Availability: InStock
Rating: 5 (10 reviews)

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Catalog No. T23388Cas No. 1150153-86-8

Alias SR16584

SR 16584 is a selective α3β4 nAChR antagonist (IC50 = 10.2 μM, Ki = 0.508) that can attenuate the contractile effects induced by epibatidine.

SR 16584

🥰Excellent

Purity: 99.84%

Catalog No. T23388Alias SR16584Cas No. 1150153-86-8

SR 16584 is a selective α3β4 nAChR antagonist (IC50 = 10.2 μM, Ki = 0.508) that can attenuate the contractile effects induced by epibatidine.

Pack Size	Price	USA Warehouse	Global Warehouse
1 mg	$120	-	In Stock
5 mg	$519	-	In Stock
10 mg	$693	-	In Stock

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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]

This molecule is a custom-made product. TargetMol has an excellent synthesis team with the experience and capability to provide you with cost-effective products. However, due to objective factors, there is a small probability that the synthesis may not be successful during the R&D process. We appreciate your understanding. If you have any questions, please feel free to contact us. We are committed to serving you wholeheartedly.

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Purity:99.84%

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COA HNMR LCMS

Product Introduction

Bioactivity

Description	SR 16584 is a selective α3β4 nAChR antagonist (IC50 = 10.2 μM, Ki = 0.508) that can attenuate the contractile effects induced by epibatidine.
Targets&IC50	α3β4 nAChR:10.2μM
Synonyms	SR16584

Chemical Properties

Molecular Weight	270.37
Formula	C₁₇H₂₂N₂O
Cas No.	1150153-86-8
Smiles	O=C1N(C=2C(C1)=CC=CC2)[C@@H]3C[C@@]4(N(C)[C@](C3)(CCC4)[H])[H]
Relative Density.	1.168 g/cm3 (Predicted)

Storage & Solubility Information

Storage	store at low temperature \| Powder: -20°C for 3 years \| In solvent: -80°C for 1 year \| Shipping with blue ice/Shipping at ambient temperature.
Solubility Information	DMSO: Soluble

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

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