M1/M2/M4 muscarinic agonist 3

Name: M1/M2/M4 muscarinic agonist 3
Brand: TargetMol
SKU: T86843
Rating: 4.5 (1 reviews)

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Catalog No. T86843Cas No. 2640109-28-8

Muscarinic agonist 3 (compound 45) is a muscarinic mAChR M1/M2/M4 agonist with EC50 values of 3.2 nM, 32 nM, and 1.7 nM, respectively [1].

M1/M2/M4 muscarinic agonist 3

😃Good

Catalog No. T86843Cas No. 2640109-28-8

Muscarinic agonist 3 (compound 45) is a muscarinic mAChR M1/M2/M4 agonist with EC50 values of 3.2 nM, 32 nM, and 1.7 nM, respectively [1].

Pack Size	Price	Availability	Quantity
10 mg	Inquiry	10-14 weeks
50 mg	Inquiry	10-14 weeks

Bulk & Custom

With extensive experience in compound synthesis, we can provide rapid custom synthesis services for this product according to your research needs.All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.

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Product Introduction

Bioactivity

Description

Muscarinic agonist 3 (compound 45) is a muscarinic mAChR M1/M2/M4 agonist with EC50 values of 3.2 nM, 32 nM, and 1.7 nM, respectively [1].

Chemical Properties

Molecular Weight	402.50
Formula	C₂₃H₃₁FN₂O₃
Cas No.	2640109-28-8

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.

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A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

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Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

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