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Results for "

AChR

" in TargetMol Product Catalog
  • Inhibitors & Agonists
    503
    TargetMol | Inhibitors_Agonists
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    14
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SIB-1553A hydrochloride
T16881191611-89-9In house
SIB-1553A hydrochloride is an orally available, selective nicotinic acetylcholine receptor agonist and a selective neuronal nAChR ligand.SIB-1553A hydrochloride enhances cognition and may be useful in the study of Alzheimer's disease and cognitive impairment.
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6-8 weeks
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Anisodamine
6-Hydroxyhyoscyamine, 6-beta-Hydroxyhyoscyamine
T2153255869-99-3In house
Anisodamine (6-beta-Hydroxyhyoscyamine) is an antagonist of muscarinic and nicotinic cholinoceptor with similar affinities at the muscarinic receptor as scopolamine and atropine. Anisodamine improve the microcirculation in states of shock and can be used in studies about organophosphate poisoning.
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6-8 weeks
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Dibucaine hydrochloride
Dibucaine HCl, Cinchocaine hydrochloride, Cinchocaine HCl
T0364L61-12-1
Dibucaine hydrochloride (Cinchocaine hydrochloride), a long-acting local amide anestheticsis, is usually used for surface anesthesia.
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7-10 days
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Neostigmine methyl sulfate
Syntostigmin, Normastigmin, Hodostin
T161251-60-5
Neostigmine methyl sulfate (Syntostigmin) is a reversible inhibitor of acetylcholinesterase, can not cross the blood-brain barrier, used in the treatment of myasthenia gravis.
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Arecoline
T6895363-75-2
Arecoline is a natural alkaloid derived from areca nut in the palm family and is a potent nicotine and partial agonist of muscarinic acetylcholine receptors. Arecoline has anti-anxiety and anti-parasitic activity, can induce oxidative stress and can be used to study Alzheimer's disease and Alzheimer's disease.
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6-8 weeks
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(+)-Sparteine
Pachycarpine
T7853492-08-0
(+)-Sparteine ​​is a quinoline alkaloid extracted from Scotch broom, a sodium channel blocker and a class 1a antiarrhythmic agent. It competitively inhibits the activity of nicotinic acetylcholine receptors in nerve cells and is a ganglionic blocking agent.
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D-Menthol
Menthol, (+)-MENTHOL
TN154415356-60-2
D-Menthol ((+)-MENTHOL) is a common compound in pharmaceutical and commercial products and a popular additive to cigarettes, it attenuates α±7 mediated Ca 2+ transients in the cell body and neurite, suggests that menthol inhibits α±7-nACh receptors in a noncompetitive manner.
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Temephos
Temefos
T09973383-96-8
Temephos (Temefos) is a cholinesterase inhibitor. Temephos is an organothiophosphate insecticide, used in the therapy of water infested with disease-carrying insects including midges, mosquitoes, and black fly larvae.
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TargetMol | Inhibitor Sale
Physostigmine Salicylate
T013057-64-7
Physostigmine, a parasympathomimetic alkaloid, is a reversible cholinesterase inhibitor. It extracts from the Calabar bean.
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TargetMol | Inhibitor Sale
Nanofin
Naniopinum, Lupetidine, Lupetidin, 2,6-Lupetidine, 2,6-Dimethylpiperidine
T1007504-03-0
Nanofin (Lupetidine) is a neuropathic blocker, with antihypertensive effect.
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Cisatracurium besylate
51W89
T145996946-42-8
Cisatracurium besylate (51W89) is a nondepolarizing skeletal muscle relaxant intended for intravenous administration.
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3-Epioleanolic acid
TN124825499-90-5
3-Epioleanolic acid and oleanonic acid possess varying degrees of agonist activity on uterine smooth muscle with minor changes in the molecular structure affecting its intrinsic activity on uterine muscle.
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beta-Amyrone
β-Amyron
TN3500638-97-1
beta-Amyrone (β-Amyron) has antifungal activity against Chikungunya virus replication with an EC50 of 86 uM. beta-Amyrone has anti-inflammatory activity through inhibiting the expression of COX-2. beta-Amyrone exhibits anti-α-glucosidase inhibitory activity and moderate AChE activity. β-Amyrone can be used in the research of disease like inflammation, infection, and obesity.
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buxbodine b
TN3550390362-51-3
Buxbodine B has weak anti-AChE activity with IC50 values in the range of 10.8-98μM.
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lucidadiol
TN4456252351-95-4
Lucidadiol exhibits butyrylcholinesterase-inhibitory activity at concentrations up to 200 uM, it also possesses inhibitory activity against acetylcholinesterase (AChE) with the percentage inhibition at 100 uM. Lucidadiol shows antiviral activity against i
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Pseudotaraxasterol
TN4837464-98-2
Pseudotaraxasterol exhibits cytotoxic activity against MOLT-4 cells.
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α-Thujone
Thujone, ALPHA-(-)-THUJONE
T8193546-80-5
α-Thujone is an inhibitor of ACh with an IC50 value of 24.7μM.
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Fustin
TN165320725-03-5
Fustin is the phytogenic flavanol component of the plant Rhus verniciflua Stokes. Fustin shows protective effects on 6-hydroxydopamine-induced neuronal cell death.
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N-p-trans-Coumaroyltyramine
TN103036417-86-4
N-p-trans-Coumaroyltyramine is a natural product and an acetylcholinesterase (AChE) inhibitor with an IC50 of 122 μM. It also exhibits anti-trypanosomal activity with an IC50 of 13.3 μM for T. brucei rhodesiense.
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Anti-Human/Rat/Fish AChR Antibody (Mab35)
T9901A-531
Anti-Human Rat Fish AChR Antibody (Mab35) is an IgG1 antibody inhibitor derived from rats, targeting AChR in humans, rats, and fish.
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2-4 weeks
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mAChR-IN-1 hydrochloride
T5655119391-73-0
mAChR-IN-1 hydrochloride is a potent antagonist of muscarinic cholinergic receptors (mAChR) with an IC50 of 17 nM.
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TargetMol | Inhibitor Sale
nAChR agonist 1
DUN71755
T121651394371-75-5
nAChR agonist 1 (DUN71755) is a brain-permeable and orally efficacious positive allosteric α7 nicotinic acetylcholine receptor (α7 nAChR)modulator.
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mAChr-in-1
T5476119391-56-9
mAChR-IN-1 is muscarinic cholinergic receptor(mAChR) antagonist (IC50=17 nM).
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1-2 weeks
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M4 mAChR agonist-1 
4-Piperidinecarboxamide, 1-(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)-
T9889785705-53-5
M4 mAChR agonist-1 (4-Piperidinecarboxamide, 1-(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)-) is an effective agonist of M4 mAChR (EC50 >10 μM).
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