TCS2185 |
Yohimbine
|
146-48-5
|
|
|
Yohimbine is a nonselective alpha 2-adrenergic receptor (AR) antagonist(IC50 : 0.6 μM)
|
T1769 |
Pardoprunox
|
269718-84-5
|
|
|
Pardoprunox is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist properties. Pardoprunox has been used in trials studying the...
|
TN4882 |
Quinine HCl
|
130-89-2
|
98%
|
|
Quinine HCl produces alpha-adrenergic blockade. Quinine modifies catecholamine- and calcium-induced myocardial contractile force responses.
|
TN4323 |
Isorauhimbine
|
483-09-0
|
98%
|
|
3-Epi-alpha-yohimbine(Isorauhimbine) has alpha adrenoceptor blocking activities,it also has cardiovascular effects.
|
T5450 |
DL-071-IT
|
55104-39-7
|
98%
|
|
DL 071-IT is a potent non-selective beta-adrenoceptor antagonist. DL 071 IT showed intrinsic sympathomimetic activity and weak membrane stabilizing activity.
|
T13470 |
(±)-Levomepromazine-d6
|
1189805-51-3
|
98%
|
|
(±)-Methotrimeprazine (D6) is the deuterium labeled Methotrimeprazine, which is an antagonist of D3 dopamine and Histamine H1 receptor.
|
TN1797 |
Isorhoifolin
|
552-57-8
|
98%
|
|
Isorhoifolin and vicenin II are main compounds of ethyl acetate fraction (EAcF) obtained from Erythrina velutina leaves, EAcF increases the cardiac contractile f...
|
T15042 |
D2343
|
72734-63-5
|
98%
|
|
D2343 is an agonist of β2-adrenoceptor. It also is an inhibitor of α1- adrenoceptor.
|
T12343 |
Benzquinamide
|
63-12-7
|
98%
|
|
Benzquinamide is an antiemetic, can bind to the α2A, α2B, and α2C adrenergic receptors (α2-AR) (Ki of 1,365, 691, and 545 nM, respectively).
|
T6663 |
Scopine hydrochloride
|
85700-55-6
|
98%
|
|
Scopine HCl salt is the metabolite of anisodine, which is a α1-adrenergic receptor agonist and used in the treatment of acute circulatory shock.
|
T16769 |
Ro 363
|
74513-77-2
|
98%
|
|
RO 363 is an effective inotropic stimulant and is a cardiovascular modulator that decreases diastolic blood pressure and pronounces increases in myocardial contr...
|
TN2267 |
Tetrahydroalstonine
|
6474-90-4
|
98%
|
|
Tetrahydroalstonine is an indole alkaloid extracted from the fruit of Rhazya stricta and is a selective α2-adrenoceptor antagonist. tetrahydroalstonine has shown...
|
TN3368 |
Akuammigine
|
642-17-1
|
98%
|
|
Akuammigine has in vitro antimalarial activity. Akuammigine competitively antagonizes the effect of noradrenaline on postsynaptic alpha-adrenoceptors, yielding p...
|
T10364 |
Arbutamine
|
128470-16-6
|
98%
|
|
Arbutamine is a short-acting synthetic potent nonselective β-adrenoceptor agonist that increases cardiac contractility, heart rate, and systolic blood pressure.
|
T11786 |
KUL-7211 racemate
|
911196-40-2
|
98%
|
|
KUL 7211 is a selective β-adrenoceptor agonist. KUL 7211 racemate is the racemate of KUL 7211.
|
T12815 |
(S)-Terazosin
|
109351-33-9
|
98%
|
|
(S)-Terazosin is an active S-enantiomer of Terazosin. (S)-Terazosin is a potent and high-affinity antagonist of α-adrenoceptor(α1a, α1b and α1d-adrenoceptor with...
|
T13285 |
Vatinoxan hydrochloride
|
130466-38-5
|
98%
|
|
Vatinoxan hydrochloride is an antagonist of the peripheral α2 adrenergic receptors.
|
T11894 |
Lusaperidone
|
214548-46-6
|
98%
|
|
Lusaperidone is an α2 adrenergic receptor antagonist, with Kis of 0.13 and 0.15 nM for α2A and α2C, respectively.
|
T6562 |
Latrepirdine dihydrochloride
|
97657-92-6
|
98%
|
|
Latrepirdine is an orally active, and neuroactive antagonist of multiple drug targets, including histamine receptors, GluR, and 5-HT receptors, used as an antihi...
|
T11036 |
Diacetolol D7
|
1346604-19-0
|
98%
|
|
Diacetolol D7 is deuterium-labeled diacetone Roller. Diacetol is the main metabolite of Acetolol. Diacetololβ-adrenoceptor shielding and anti-arrhythmic agent.
|