Home Tools
Log in
Cart

Adrenergic Receptor

The adrenergic receptors or adrenoceptors are a class of G protein-coupled receptors that are targets of many catecholamines like norepinephrine (noradrenaline) and epinephrine (adrenaline) produced by the body, but also many medications like beta blockers, β2 agonists and α2 agonists, which are used to treat high blood pressure and asthma, for example.
Signaling Pathways | Target | TargetMol
Cat. No. Product name CAS No. Purity Chemical Structure
T0143 Bisoprolol hemifumarate 104344-23-2 99.95%
Bisoprolol hemifumarate
Bisoprolol, a selective beta-1 adrenergic receptor antagonist, selectively and competitively binds to and blocks beta-1 adrenergic receptors in the heart, thereb...
T0487 Metoprolol tartrate 56392-17-7 99.72%
Metoprolol tartrate
Metoprolol Tartrate is a blocker of the cardioselective β-adrenergic receptor.
TN7042 N-methyltyramine 370-98-9 99.59%
N-methyltyramine
N-methyltyramine is an alkaloid isolated from the leguminous plant Acacia grandiflora.It is an α2-adrenoceptor antagonist that regulates adrenergic receptors thr...
T13106 TD-5471 hydrochloride 530084-35-6 99.57%
TD-5471 hydrochloride
TD-5471 hydrochloride is a selective and potent long-acting human β2-adrenergic receptor agonist for the treatment of chronic obstructive pulmonary disease (COPD...
T1503 Esmolol hydrochloride 81161-17-3 99.48%
Esmolol hydrochloride
Esmolol is a cardioselective beta-blocker used in parenteral forms in the treatment of arrhythmias and severe hypertension. Esmolol has not been linked to instan...
T2645 Vilanterol 503068-34-6 99.46%
Vilanterol
Vilanterol is a selective long-acting beta2-adrenergic agonist (LABA) used in the treatment of COPD and asthma.
T15742 Levobunolol hydrochloride 27912-14-7 98.49%
Levobunolol hydrochloride
Levobunolol hydrochloride is a non-selective blocker of β-adrenergic receptor and can be used in studies about managing glaucoma and superior oblique myokymia.
T3457 Olodaterol 868049-49-4 98%
Olodaterol
Olodaterol is a novel, long-acting beta2-adrenergic agonist (LABA) that exerts its pharmacological effect by binding and activating beta2-adrenergic receptors lo...
T12596 (4E)-SUN9221 222318-55-0 97.79%
(4E)-SUN9221
(4E)-SUN9221 is a potent dual α1-adrenergic receptor and 5-HT2 receptor antagonist that shows antihypertensive and antiplatelet aggregation activity in hypertens...
T10812 Cicloprolol hydrochloride 63686-79-3 97.26%
Cicloprolol hydrochloride
Cicloprolol hydrochloride is a new potent and selective beta 1-adrenoceptor antagonist with partial agonist activity for the study of coronary heart disease.
TCS2185 Yohimbine 146-48-5
Yohimbine
Yohimbine is a nonselective alpha 2-adrenergic receptor (AR) antagonist(IC50 : 0.6 μM)
T1244 Celiprolol hydrochloride 57470-78-7
Celiprolol hydrochloride
Celiprolol hydrochloride (Selectrol) is a cardioselective beta-1 adrenergic antagonist that has intrinsic sympathomimetic activity. It is used in the management ...
T1203 Nadolol 42200-33-9
Nadolol
Nadolol is a non-selective beta-adrenergic antagonist with antihypertensive and antiarrhythmic activities. Nadolol competitively blocks beta-1 adrenergic recepto...
T1769 Pardoprunox 269718-84-5
Pardoprunox
Pardoprunox (SLV-308) is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist properties. Pardoprunox has been used in trials st...
TN4882 Quinine HCl 130-89-2 98%
Quinine HCl
Quinine HCl produces alpha-adrenergic blockade. Quinine modifies catecholamine- and calcium-induced myocardial contractile force responses.
T5450 DL-071-IT 55104-39-7 98%
DL-071-IT
DL-071-IT (Afurolol Hydrochloride) is a potent non-selective beta-adrenoceptor antagonist. DL-071-IT showed intrinsic sympathomimetic activity and weak membrane ...
T13470 (±)-Levomepromazine-d6 1189805-51-3 98%
(±)-Levomepromazine-d6
(±)-Methotrimeprazine (D6) is the deuterium labeled Methotrimeprazine, which is an antagonist of D3 dopamine and Histamine H1 receptor.
T78567 Moprolol 5741-22-0 98%
Moprolol
Moprolol ((±)-Moprolol) is a beta-adrenergic receptor antagonist utilized in research pertaining to essential hypertension [1] [2] [3].
T79641 (±)-N-Methylcoclaurine 1472-62-4 98%
(±)-N-Methylcoclaurine
N-Methylcoclaurine (±) acts as a selective antagonist at the α2-adrenoceptor [1].
T80175 Conopeptide rho-TIA 381725-58-2 98%
Conopeptide rho-TIA
Conopeptide rho-TIA, a peptide from Conus tulipa venom, acts as a selective, noncompetitive inhibitor at the human α1B-Adrenergic Receptor and as a competitive i...
Bisoprolol hemifumarate
T0143
Bisoprolol, a selective beta-1 adrenergic receptor antagonist, selectively and competitively binds to and blocks beta-1 adrenergic receptors in the heart, thereb...
Metoprolol tartrate
T0487
Metoprolol Tartrate is a blocker of the cardioselective β-adrenergic receptor.
N-methyltyramine
TN7042
N-methyltyramine is an alkaloid isolated from the leguminous plant Acacia grandiflora.It is an α2-adrenoceptor antagonist that regulates adrenergic receptors thr...
TD-5471 hydrochloride
T13106
TD-5471 hydrochloride is a selective and potent long-acting human β2-adrenergic receptor agonist for the treatment of chronic obstructive pulmonary disease (COPD...
Esmolol hydrochloride
T1503
Esmolol is a cardioselective beta-blocker used in parenteral forms in the treatment of arrhythmias and severe hypertension. Esmolol has not been linked to instan...
Vilanterol
T2645
Vilanterol is a selective long-acting beta2-adrenergic agonist (LABA) used in the treatment of COPD and asthma.
Levobunolol hydrochloride
T15742
Levobunolol hydrochloride is a non-selective blocker of β-adrenergic receptor and can be used in studies about managing glaucoma and superior oblique myokymia.
Olodaterol
T3457
Olodaterol is a novel, long-acting beta2-adrenergic agonist (LABA) that exerts its pharmacological effect by binding and activating beta2-adrenergic receptors lo...
(4E)-SUN9221
T12596
(4E)-SUN9221 is a potent dual α1-adrenergic receptor and 5-HT2 receptor antagonist that shows antihypertensive and antiplatelet aggregation activity in hypertens...
Cicloprolol hydrochloride
T10812
Cicloprolol hydrochloride is a new potent and selective beta 1-adrenoceptor antagonist with partial agonist activity for the study of coronary heart disease.
Yohimbine
TCS2185
Yohimbine is a nonselective alpha 2-adrenergic receptor (AR) antagonist(IC50 : 0.6 μM)
Celiprolol hydrochloride
T1244
Celiprolol hydrochloride (Selectrol) is a cardioselective beta-1 adrenergic antagonist that has intrinsic sympathomimetic activity. It is used in the management ...
Nadolol
T1203
Nadolol is a non-selective beta-adrenergic antagonist with antihypertensive and antiarrhythmic activities. Nadolol competitively blocks beta-1 adrenergic recepto...
Pardoprunox
T1769
Pardoprunox (SLV-308) is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist properties. Pardoprunox has been used in trials st...
Quinine HCl
TN4882
Quinine HCl produces alpha-adrenergic blockade. Quinine modifies catecholamine- and calcium-induced myocardial contractile force responses.
DL-071-IT
T5450
DL-071-IT (Afurolol Hydrochloride) is a potent non-selective beta-adrenoceptor antagonist. DL-071-IT showed intrinsic sympathomimetic activity and weak membrane ...
(±)-Levomepromazine-d6
T13470
(±)-Methotrimeprazine (D6) is the deuterium labeled Methotrimeprazine, which is an antagonist of D3 dopamine and Histamine H1 receptor.
Moprolol
T78567
Moprolol ((±)-Moprolol) is a beta-adrenergic receptor antagonist utilized in research pertaining to essential hypertension [1] [2] [3].
(±)-N-Methylcoclaurine
T79641
N-Methylcoclaurine (±) acts as a selective antagonist at the α2-adrenoceptor [1].
Conopeptide rho-TIA
T80175
Conopeptide rho-TIA, a peptide from Conus tulipa venom, acts as a selective, noncompetitive inhibitor at the human α1B-Adrenergic Receptor and as a competitive i...
1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 18
TargetMol