Adrenergic Receptor

The adrenergic receptors or adrenoceptors are a class of G protein-coupled receptors that are targets of many catecholamines like norepinephrine (noradrenaline) and epinephrine (adrenaline) produced by the body, but also many medications like beta blockers, β2 agonists and α2 agonists, which are used to treat high blood pressure and asthma, for example.

Cat. No.	Product name	CAS No.	Purity
T8304	Anisodamine Hydrobromide	55449-49-5	98%
T8304	Anisodamine Hydrobromide is an anticholinergic and α1-adrenergic receptor antagonist used in the treatment of acute circulatory shock.
TN5061	Stephanine	517-63-5	98%
TN5061	l-Stephanine is a potent and highly selective alpha 1 adrenoceptor blocker, inhibits anococcygeus muscle contraction induced by phenylephrine with pA2 values of ...
T12815	(S)-Terazosin	109351-33-9	98%
T12815	(S)-Terazosin is an active S-enantiomer of Terazosin. (S)-Terazosin is a potent and high-affinity antagonist of α-adrenoceptor(α1a, α1b and α1d-adrenoceptor with...
T6860	ICI-118551 Hydrochloride	1217094-53-5	98%
T6860	ICI-118551 is a highly selective β2-adrenergic receptor antagonist with Ki values of 0.7, 49.5 and 611 nM for β2, β1 and β3 receptors, respectively.
T11036	Diacetolol D7	1346604-19-0	98%
T11036	Diacetolol D7 is deuterium-labeled diacetone Roller. Diacetol is the main metabolite of Acetolol. Diacetololβ-adrenoceptor shielding and anti-arrhythmic agent.
T15943	M443	1820684-31-8	98%
T15943	M443 is an irreversible and specific MRK inhibitor (IC50<125 nM).
T6562	Latrepirdine dihydrochloride	97657-92-6	98%
T6562	Latrepirdine is an orally active, and neuroactive antagonist of multiple drug targets, including histamine receptors, GluR, and 5-HT receptors, used as an antihi...
T1769	Pardoprunox	269718-84-5	98%
T1769	Pardoprunox is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist properties. Pardoprunox has been used in trials studying the...
T10778	CGP 20712 A	105737-62-0	98%
T10778	CGP 20712 A (CGP 20712 mesylate) is a highly selective antagonist of β1-adrenoceptor (IC50: 0.7 nM). It shows ~10,000-fold selectivity over β2-adrenoceptors.
TN3507	Beta-Yohimbine	549-84-8	98%
TN3507	Beta-Yohimbine has approximately twice as toxic as yohimbine and corynanthine about one fifth as toxic. Beta-yohimbine has alpha-1 and alpha-2 adrenoceptor block...
T12343	Benzquinamide	63-12-7	98%
T12343	Benzquinamide is an antiemetic, can bind to the α2A, α2B, and α2C adrenergic receptors (α2-AR) (Ki of 1,365, 691, and 545 nM, respectively).
T11010	Detomidine carboxylic acid	115664-39-6	98%
T11010	Detomidine carboxylic acid is the main urine metabolite of detomidine. Detomidine is a synthetic α2-adrenergic agonist and an animal analgesic. Detomidine also h...
T14287	Ancarolol	75748-50-4	98%
T14287	Ancarolol is a blocking agent of beta-adrenergic.
T23397	ST 91	4749-61-5	98%
T23397	ST-91 is an agonist of α2-adrenoceptor with a mixed α-adrenergic receptor type/subtype selection profile.
TN3368	Akuammigine	642-17-1	98%
TN3368	Akuammigine has in vitro antimalarial activity. Akuammigine competitively antagonizes the effect of noradrenaline on postsynaptic alpha-adrenoceptors, yielding p...
T15042	D2343	72734-63-5	98%
T15042	D2343 is an agonist of β2-adrenoceptor. It also is an inhibitor of α1- adrenoceptor.
TN2267	Tetrahydroalstonine	6474-90-4	98%
TN2267	Tetrahydroalstonine and Raubasine preferentially block the pressor responses of post-synaptic alpha-adrenergic receptor activation due to exogenous and endogenou...
TN4882	Quinine HCl	130-89-2	98%
TN4882	Quinine HCl produces alpha-adrenergic blockade. Quinine modifies catecholamine- and calcium-induced myocardial contractile force responses.
T1728	Lofexidine hydrochloride	21498-08-8	98%
T1728	Lofexidine (hydrochloride) is a selective α2-receptor agonist, commonly used to alleviate the physical symptoms of heroin and other types of opioid withdrawal [1...
T10364	Arbutamine	128470-16-6	98%
T10364	Arbutamine is a short-acting synthetic potent nonselective β-adrenoceptor agonist that increases cardiac contractility, heart rate, and systolic blood pressure.