Adrenergic Receptor

The adrenergic receptors or adrenoceptors are a class of G protein-coupled receptors that are targets of many catecholamines like norepinephrine (noradrenaline) and epinephrine (adrenaline) produced by the body, but also many medications like beta blockers, β2 agonists and α2 agonists, which are used to treat high blood pressure and asthma, for example.

Cat. No.	Product name	CAS No.	Purity
TCS2185	Yohimbine	146-48-5
TCS2185	Yohimbine is a nonselective alpha 2-adrenergic receptor (AR) antagonist(IC50 : 0.6 μM)
T1769	Pardoprunox	269718-84-5
T1769	Pardoprunox is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist properties. Pardoprunox has been used in trials studying the...
TN4882	Quinine HCl	130-89-2	98%
TN4882	Quinine HCl produces alpha-adrenergic blockade. Quinine modifies catecholamine- and calcium-induced myocardial contractile force responses.
TN4323	Isorauhimbine	483-09-0	98%
TN4323	3-Epi-alpha-yohimbine(Isorauhimbine) has alpha adrenoceptor blocking activities,it also has cardiovascular effects.
T5450	DL-071-IT	55104-39-7	98%
T5450	DL 071-IT is a potent non-selective beta-adrenoceptor antagonist. DL 071 IT showed intrinsic sympathomimetic activity and weak membrane stabilizing activity.
T13470	(±)-Levomepromazine-d6	1189805-51-3	98%
T13470	(±)-Methotrimeprazine (D6) is the deuterium labeled Methotrimeprazine, which is an antagonist of D3 dopamine and Histamine H1 receptor.
TN1797	Isorhoifolin	552-57-8	98%
TN1797	Isorhoifolin and vicenin II are main compounds of ethyl acetate fraction (EAcF) obtained from Erythrina velutina leaves, EAcF increases the cardiac contractile f...
T15042	D2343	72734-63-5	98%
T15042	D2343 is an agonist of β2-adrenoceptor. It also is an inhibitor of α1- adrenoceptor.
T12343	Benzquinamide	63-12-7	98%
T12343	Benzquinamide is an antiemetic, can bind to the α2A, α2B, and α2C adrenergic receptors (α2-AR) (Ki of 1,365, 691, and 545 nM, respectively).
T6663	Scopine hydrochloride	85700-55-6	98%
T6663	Scopine HCl salt is the metabolite of anisodine, which is a α1-adrenergic receptor agonist and used in the treatment of acute circulatory shock.
T16769	Ro 363	74513-77-2	98%
T16769	RO 363 is an effective inotropic stimulant and is a cardiovascular modulator that decreases diastolic blood pressure and pronounces increases in myocardial contr...
TN2267	Tetrahydroalstonine	6474-90-4	98%
TN2267	Tetrahydroalstonine is an indole alkaloid extracted from the fruit of Rhazya stricta and is a selective α2-adrenoceptor antagonist. tetrahydroalstonine has shown...
TN3368	Akuammigine	642-17-1	98%
TN3368	Akuammigine has in vitro antimalarial activity. Akuammigine competitively antagonizes the effect of noradrenaline on postsynaptic alpha-adrenoceptors, yielding p...
T10364	Arbutamine	128470-16-6	98%
T10364	Arbutamine is a short-acting synthetic potent nonselective β-adrenoceptor agonist that increases cardiac contractility, heart rate, and systolic blood pressure.
T11786	KUL-7211 racemate	911196-40-2	98%
T11786	KUL 7211 is a selective β-adrenoceptor agonist. KUL 7211 racemate is the racemate of KUL 7211.
T12815	(S)-Terazosin	109351-33-9	98%
T12815	(S)-Terazosin is an active S-enantiomer of Terazosin. (S)-Terazosin is a potent and high-affinity antagonist of α-adrenoceptor(α1a, α1b and α1d-adrenoceptor with...
T13285	Vatinoxan hydrochloride	130466-38-5	98%
T13285	Vatinoxan hydrochloride is an antagonist of the peripheral α2 adrenergic receptors.
T11894	Lusaperidone	214548-46-6	98%
T11894	Lusaperidone is an α2 adrenergic receptor antagonist, with Kis of 0.13 and 0.15 nM for α2A and α2C, respectively.
T6562	Latrepirdine dihydrochloride	97657-92-6	98%
T6562	Latrepirdine is an orally active, and neuroactive antagonist of multiple drug targets, including histamine receptors, GluR, and 5-HT receptors, used as an antihi...
T11036	Diacetolol D7	1346604-19-0	98%
T11036	Diacetolol D7 is deuterium-labeled diacetone Roller. Diacetol is the main metabolite of Acetolol. Diacetololβ-adrenoceptor shielding and anti-arrhythmic agent.