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Adrenergic Receptor

The adrenergic receptors or adrenoceptors are a class of G protein-coupled receptors that are targets of many catecholamines like norepinephrine (noradrenaline) and epinephrine (adrenaline) produced by the body, but also many medications like beta blockers, β2 agonists and α2 agonists, which are used to treat high blood pressure and asthma, for example.
Cat. No. Product name CAS No. Purity Chemical Structure
T8304 Anisodamine Hydrobromide 55449-49-5 98%
Anisodamine Hydrobromide is an anticholinergic and α1-adrenergic receptor antagonist used in the treatment of acute circulatory shock.
TN5061 Stephanine 517-63-5 98%
l-Stephanine is a potent and highly selective alpha 1 adrenoceptor blocker, inhibits anococcygeus muscle contraction induced by phenylephrine with pA2 values of ...
T12815 (S)-Terazosin 109351-33-9 98%
(S)-Terazosin is an active S-enantiomer of Terazosin. (S)-Terazosin is a potent and high-affinity antagonist of α-adrenoceptor(α1a, α1b and α1d-adrenoceptor with...
T6860 ICI-118551 Hydrochloride 1217094-53-5 98%
ICI-118551 is a highly selective β2-adrenergic receptor antagonist with Ki values of 0.7, 49.5 and 611 nM for β2, β1 and β3 receptors, respectively.
T11036 Diacetolol D7 1346604-19-0 98%
Diacetolol D7 is deuterium-labeled diacetone Roller. Diacetol is the main metabolite of Acetolol. Diacetololβ-adrenoceptor shielding and anti-arrhythmic agent.
T15943 M443 1820684-31-8 98%
M443 is an irreversible and specific MRK inhibitor (IC50<125 nM).
T6562 Latrepirdine dihydrochloride 97657-92-6 98%
Latrepirdine is an orally active, and neuroactive antagonist of multiple drug targets, including histamine receptors, GluR, and 5-HT receptors, used as an antihi...
T1769 Pardoprunox 269718-84-5 98%
Pardoprunox is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist properties. Pardoprunox has been used in trials studying the...
T10778 CGP 20712 A 105737-62-0 98%
CGP 20712 A (CGP 20712 mesylate) is a highly selective antagonist of β1-adrenoceptor (IC50: 0.7 nM). It shows ~10,000-fold selectivity over β2-adrenoceptors.
TN3507 Beta-Yohimbine 549-84-8 98%
Beta-Yohimbine has approximately twice as toxic as yohimbine and corynanthine about one fifth as toxic. Beta-yohimbine has alpha-1 and alpha-2 adrenoceptor block...
T12343 Benzquinamide 63-12-7 98%
Benzquinamide is an antiemetic, can bind to the α2A, α2B, and α2C adrenergic receptors (α2-AR) (Ki of 1,365, 691, and 545 nM, respectively).
T11010 Detomidine carboxylic acid 115664-39-6 98%
Detomidine carboxylic acid is the main urine metabolite of detomidine. Detomidine is a synthetic α2-adrenergic agonist and an animal analgesic. Detomidine also h...
T14287 Ancarolol 75748-50-4 98%
Ancarolol is a blocking agent of beta-adrenergic.
T23397 ST 91 4749-61-5 98%
ST-91 is an agonist of α2-adrenoceptor with a mixed α-adrenergic receptor type/subtype selection profile.
TN3368 Akuammigine 642-17-1 98%
Akuammigine has in vitro antimalarial activity. Akuammigine competitively antagonizes the effect of noradrenaline on postsynaptic alpha-adrenoceptors, yielding p...
T15042 D2343 72734-63-5 98%
D2343 is an agonist of β2-adrenoceptor. It also is an inhibitor of α1- adrenoceptor.
TN2267 Tetrahydroalstonine 6474-90-4 98%
Tetrahydroalstonine and Raubasine preferentially block the pressor responses of post-synaptic alpha-adrenergic receptor activation due to exogenous and endogenou...
TN4882 Quinine HCl 130-89-2 98%
Quinine HCl produces alpha-adrenergic blockade. Quinine modifies catecholamine- and calcium-induced myocardial contractile force responses.
T1728 Lofexidine hydrochloride 21498-08-8 98%
Lofexidine (hydrochloride) is a selective α2-receptor agonist, commonly used to alleviate the physical symptoms of heroin and other types of opioid withdrawal [1...
T10364 Arbutamine 128470-16-6 98%
Arbutamine is a short-acting synthetic potent nonselective β-adrenoceptor agonist that increases cardiac contractility, heart rate, and systolic blood pressure.
Anisodamine Hydrobromide
T8304
Anisodamine Hydrobromide is an anticholinergic and α1-adrenergic receptor antagonist used in the treatment of acute circulatory shock.
Stephanine
TN5061
l-Stephanine is a potent and highly selective alpha 1 adrenoceptor blocker, inhibits anococcygeus muscle contraction induced by phenylephrine with pA2 values of ...
(S)-Terazosin
T12815
(S)-Terazosin is an active S-enantiomer of Terazosin. (S)-Terazosin is a potent and high-affinity antagonist of α-adrenoceptor(α1a, α1b and α1d-adrenoceptor with...
ICI-118551 Hydrochloride
T6860
ICI-118551 is a highly selective β2-adrenergic receptor antagonist with Ki values of 0.7, 49.5 and 611 nM for β2, β1 and β3 receptors, respectively.
Diacetolol D7
T11036
Diacetolol D7 is deuterium-labeled diacetone Roller. Diacetol is the main metabolite of Acetolol. Diacetololβ-adrenoceptor shielding and anti-arrhythmic agent.
M443
T15943
M443 is an irreversible and specific MRK inhibitor (IC50<125 nM).
Latrepirdine dihydrochloride
T6562
Latrepirdine is an orally active, and neuroactive antagonist of multiple drug targets, including histamine receptors, GluR, and 5-HT receptors, used as an antihi...
Pardoprunox
T1769
Pardoprunox is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist properties. Pardoprunox has been used in trials studying the...
CGP 20712 A
T10778
CGP 20712 A (CGP 20712 mesylate) is a highly selective antagonist of β1-adrenoceptor (IC50: 0.7 nM). It shows ~10,000-fold selectivity over β2-adrenoceptors.
beta-Yohimbine
TN3507
Beta-Yohimbine has approximately twice as toxic as yohimbine and corynanthine about one fifth as toxic. Beta-yohimbine has alpha-1 and alpha-2 adrenoceptor block...
Benzquinamide
T12343
Benzquinamide is an antiemetic, can bind to the α2A, α2B, and α2C adrenergic receptors (α2-AR) (Ki of 1,365, 691, and 545 nM, respectively).
Detomidine carboxylic acid
T11010
Detomidine carboxylic acid is the main urine metabolite of detomidine. Detomidine is a synthetic α2-adrenergic agonist and an animal analgesic. Detomidine also h...
Ancarolol
T14287
Ancarolol is a blocking agent of beta-adrenergic.
ST 91
T23397
ST-91 is an agonist of α2-adrenoceptor with a mixed α-adrenergic receptor type/subtype selection profile.
Akuammigine
TN3368
Akuammigine has in vitro antimalarial activity. Akuammigine competitively antagonizes the effect of noradrenaline on postsynaptic alpha-adrenoceptors, yielding p...
D2343
T15042
D2343 is an agonist of β2-adrenoceptor. It also is an inhibitor of α1- adrenoceptor.
Tetrahydroalstonine
TN2267
Tetrahydroalstonine and Raubasine preferentially block the pressor responses of post-synaptic alpha-adrenergic receptor activation due to exogenous and endogenou...
Quinine HCl
TN4882
Quinine HCl produces alpha-adrenergic blockade. Quinine modifies catecholamine- and calcium-induced myocardial contractile force responses.
Lofexidine hydrochloride
T1728
Lofexidine (hydrochloride) is a selective α2-receptor agonist, commonly used to alleviate the physical symptoms of heroin and other types of opioid withdrawal [1...
Arbutamine
T10364
Arbutamine is a short-acting synthetic potent nonselective β-adrenoceptor agonist that increases cardiac contractility, heart rate, and systolic blood pressure.
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