T8304 |
Anisodamine Hydrobromide
|
55449-49-5
|
98%
|
|
Anisodamine Hydrobromide is an anticholinergic and α1-adrenergic receptor antagonist used in the treatment of acute circulatory shock.
|
TN5061 |
Stephanine
|
517-63-5
|
98%
|
|
l-Stephanine is a potent and highly selective alpha 1 adrenoceptor blocker, inhibits anococcygeus muscle contraction induced by phenylephrine with pA2 values of ...
|
T12815 |
(S)-Terazosin
|
109351-33-9
|
98%
|
|
(S)-Terazosin is an active S-enantiomer of Terazosin. (S)-Terazosin is a potent and high-affinity antagonist of α-adrenoceptor(α1a, α1b and α1d-adrenoceptor with...
|
T6860 |
ICI-118551 Hydrochloride
|
1217094-53-5
|
98%
|
|
ICI-118551 is a highly selective β2-adrenergic receptor antagonist with Ki values of 0.7, 49.5 and 611 nM for β2, β1 and β3 receptors, respectively.
|
T11036 |
Diacetolol D7
|
1346604-19-0
|
98%
|
|
Diacetolol D7 is deuterium-labeled diacetone Roller. Diacetol is the main metabolite of Acetolol. Diacetololβ-adrenoceptor shielding and anti-arrhythmic agent.
|
T15943 |
M443
|
1820684-31-8
|
98%
|
|
M443 is an irreversible and specific MRK inhibitor (IC50<125 nM).
|
T6562 |
Latrepirdine dihydrochloride
|
97657-92-6
|
98%
|
|
Latrepirdine is an orally active, and neuroactive antagonist of multiple drug targets, including histamine receptors, GluR, and 5-HT receptors, used as an antihi...
|
T1769 |
Pardoprunox
|
269718-84-5
|
98%
|
|
Pardoprunox is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist properties. Pardoprunox has been used in trials studying the...
|
T10778 |
CGP 20712 A
|
105737-62-0
|
98%
|
|
CGP 20712 A (CGP 20712 mesylate) is a highly selective antagonist of β1-adrenoceptor (IC50: 0.7 nM). It shows ~10,000-fold selectivity over β2-adrenoceptors.
|
TN3507 |
Beta-Yohimbine
|
549-84-8
|
98%
|
|
Beta-Yohimbine has approximately twice as toxic as yohimbine and corynanthine about one fifth as toxic. Beta-yohimbine has alpha-1 and alpha-2 adrenoceptor block...
|
T12343 |
Benzquinamide
|
63-12-7
|
98%
|
|
Benzquinamide is an antiemetic, can bind to the α2A, α2B, and α2C adrenergic receptors (α2-AR) (Ki of 1,365, 691, and 545 nM, respectively).
|
T11010 |
Detomidine carboxylic acid
|
115664-39-6
|
98%
|
|
Detomidine carboxylic acid is the main urine metabolite of detomidine. Detomidine is a synthetic α2-adrenergic agonist and an animal analgesic. Detomidine also h...
|
T14287 |
Ancarolol
|
75748-50-4
|
98%
|
|
Ancarolol is a blocking agent of beta-adrenergic.
|
T23397 |
ST 91
|
4749-61-5
|
98%
|
|
ST-91 is an agonist of α2-adrenoceptor with a mixed α-adrenergic receptor type/subtype selection profile.
|
TN3368 |
Akuammigine
|
642-17-1
|
98%
|
|
Akuammigine has in vitro antimalarial activity. Akuammigine competitively antagonizes the effect of noradrenaline on postsynaptic alpha-adrenoceptors, yielding p...
|
T15042 |
D2343
|
72734-63-5
|
98%
|
|
D2343 is an agonist of β2-adrenoceptor. It also is an inhibitor of α1- adrenoceptor.
|
TN2267 |
Tetrahydroalstonine
|
6474-90-4
|
98%
|
|
Tetrahydroalstonine and Raubasine preferentially block the pressor responses of post-synaptic alpha-adrenergic receptor activation due to exogenous and endogenou...
|
TN4882 |
Quinine HCl
|
130-89-2
|
98%
|
|
Quinine HCl produces alpha-adrenergic blockade. Quinine modifies catecholamine- and calcium-induced myocardial contractile force responses.
|
T1728 |
Lofexidine hydrochloride
|
21498-08-8
|
98%
|
|
Lofexidine (hydrochloride) is a selective α2-receptor agonist, commonly used to alleviate the physical symptoms of heroin and other types of opioid withdrawal [1...
|
T10364 |
Arbutamine
|
128470-16-6
|
98%
|
|
Arbutamine is a short-acting synthetic potent nonselective β-adrenoceptor agonist that increases cardiac contractility, heart rate, and systolic blood pressure.
|