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Soquinolol (Synonyms: Soquinolol mucate)

Name: Soquinolol
Brand: TargetMol
SKU: T28829
Price: 88 USD
Availability: InStock
Rating: 5 (10 reviews)

Catalog No. T28829 Copy Product Info

Purity: 98.63%

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Soquinolol (Soquinolol mucate) is a beta-adrenergic receptor antagonist with weak local anesthetic activity.Soquinolol has good enteral efficacy and a long duration of action.

Soquinolol

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🥰Excellent

Catalog No. T28829

Synonyms Soquinolol mucate

Soquinolol (Soquinolol mucate) is a beta-adrenergic receptor antagonist with weak local anesthetic activity.Soquinolol has good enteral efficacy and a long duration of action.

Cas No. 61563-18-6

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Pack Size	Price	USA Stock	Global Stock
1 mg	$88	In Stock	In Stock
5 mg	$210	In Stock	In Stock
10 mg	$318	In Stock	In Stock
25 mg	$515	In Stock	In Stock
50 mg	$747	In Stock	In Stock
100 mg	$1,050	In Stock	In Stock
200 mg	$1,420	-	In Stock

For In stock only · Estimated delivery: USA Stock (1-2 days) Global Stock (5-7 days)

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For research use only—not for human use. No sales to individuals. Use as intended only.

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Batch Information

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Purity:98.63%

ee:100%

Color:White to Yellow

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COA CSFC HNMR HPLC

Product Introduction

Bioactivity

Description	Soquinolol (Soquinolol mucate) is a beta-adrenergic receptor antagonist with weak local anesthetic activity.Soquinolol has good enteral efficacy and a long duration of action.
In vitro	Soquinolol inhibits the isoprenaline-induced tachycardia (EC50% = 48 μg/L) in the guinea-pig Langendorff heart in vitro.[2]
In vivo	Soquinolol (5.5 μg/kg; intravenous injection; conscious dog) beta 1-adrenergic blocking activity (ED 50%) and oral administration (5.8 μg/kg; oral) is about twice as great as that of pindolol and 19 times (i.v.). These results suggest 95% enteral efficacy for soquinolol (pindolol 88%, propranolol 13%). The differences in soquinolol's and propranolol's efficacy detected in vitro and in vivo are partially attributable to differences in their kinetic properties namely the lower protein binding and the higher distribution volume of soquinolol. In the conscious dog, soquinolol inhibits beta 1-(ED 50% = 4.0 μg/kg) and beta 2 receptors (ED 50% = 2.7 μg/kg) at dose levels which do not differ significantly.[2]
Synonyms	Soquinolol mucate

Chemical Properties

Molecular Weight	306.4
Formula	C₁₇H₂₆N₂O₃
Cas No.	61563-18-6
Smiles	O(CC(CNC(C)(C)C)O)C1=C2C(CN(C=O)CC2)=CC=C1
Relative Density.	1.31g/cm3

Storage & Solubility Information

Storage

Pure form: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 45 mg/mL (146.87 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	3.2637 mL	16.3185 mL	32.6371 mL	163.1854 mL
5 mM	0.6527 mL	3.2637 mL	6.5274 mL	32.6371 mL
10 mM	0.3264 mL	1.6319 mL	3.2637 mL	16.3185 mL
20 mM	0.1632 mL	0.8159 mL	1.6319 mL	8.1593 mL
50 mM	0.0653 mL	0.3264 mL	0.6527 mL	3.2637 mL
100 mM	0.0326 mL	0.1632 mL	0.3264 mL	1.6319 mL

Note : The dilution table applies only to solid products. For liquid products, please calculate the stock solution based on the stated concentration and/or density.

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the stock solution preparation method and in vivo formula preparation method:

For example, if the intended dosage is 10 mg/kg for animals weighing 20 g , with a dosing volume of 100 μL per animal, TargetMol | Animal experiments

and a total of 10 animals are to be administered, using a formulation of TargetMol | reagent

10% DMSO+ 40% PEG300+ 5% Tween 80+ 45% Saline/PBS/ddH₂O , the resulting working solution concentration would be 2 mg/mL.

Stock Solution Preparation:

Dissolve 2 mg of the compound in 100 μL DMSO TargetMol | reagent to obtain a stock solution at a concentration of 20 mg/mL . If the required concentration exceeds the compound's known solubility, please contact us for technical support before proceeding.

Preparation of the In Vivo Formulation:

1) Add 100 μL of the DMSO TargetMol | reagent stock solution to 400 μL PEG300 and mix thoroughly until the solution becomes clear.

2) Add 50 μL Tween 80 and mix well until fully clarified.

3) Add 450 μL Saline,PBS or ddH₂O TargetMol | reagent and mix thoroughly until a homogeneous solution is obtained.

This example is provided solely to demonstrate the use of the In Vivo Formulation Calculator and does not constitute a recommended formulation for any specific compound. Please select an appropriate dissolution and formulation strategy based on your experimental model and route of administration.

All co-solvents required for this protocol, includingDMSO, PEG300/PEG400, Tween 80, SBE-β-CD, and Corn oil, are available for purchase on the TargetMol website.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc