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Efaroxan hydrochloride

🥰Excellent
Catalog No. T22760Cas No. 89197-00-2
Alias RX821037 hydrochloride, RX 821037 hydrochloride

Efaroxan hydrochloride is the salt form of Efaroxan, a selective, orally available α2-adrenoceptor antagonist that raises resting plasma insulin levels and significantly potentiates adrenaline-induced increases in insulin levels.

Efaroxan hydrochloride

Efaroxan hydrochloride

🥰Excellent
Catalog No. T22760Alias RX821037 hydrochloride, RX 821037 hydrochlorideCas No. 89197-00-2
Efaroxan hydrochloride is the salt form of Efaroxan, a selective, orally available α2-adrenoceptor antagonist that raises resting plasma insulin levels and significantly potentiates adrenaline-induced increases in insulin levels.
Pack SizePriceUSA WarehouseGlobal WarehouseQuantity
2 mg$29-In Stock
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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]
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Product Introduction

Bioactivity
Description
Efaroxan hydrochloride is the salt form of Efaroxan, a selective, orally available α2-adrenoceptor antagonist that raises resting plasma insulin levels and significantly potentiates adrenaline-induced increases in insulin levels.
In vitro
Efaroxan hydrochloride binds to 1-imidazoline and α2-adrenergic receptors in the ventrolateral medulla membrane of the cephalic bull with Ki values ​​of 0.15 nM and 5.6 nM, respectively. [1]
SynonymsRX821037 hydrochloride, RX 821037 hydrochloride
Chemical Properties
Molecular Weight252.74
FormulaC13H17ClN2O
Cas No.89197-00-2
SmilesCl.N1=C(NCC1)C2(OC=3C=CC=CC3C2)CC
Relative Density.no data available
Storage & Solubility Information
Storagekeep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
Solubility Information
H2O: 40 mg/mL (158.27 mM), Sonication is recommended.
In Vivo Formulation
10% DMSO+40% PEG300+5% Tween 80+45% Saline: 2 mg/mL (7.91 mM), Sonication is recommended.
Please add the solvents sequentially, clarifying the solution as much as possible before adding the next one. Dissolve by heating and/or sonication if necessary. Working solution is recommended to be prepared and used immediately. The formulation provided above is for reference purposes only. In vivo formulations may vary and should be modified based on specific experimental conditions.
Solution Preparation Table
H2O
1mg5mg10mg50mg
1 mM3.9566 mL19.7832 mL39.5664 mL197.8318 mL
5 mM0.7913 mL3.9566 mL7.9133 mL39.5664 mL
10 mM0.3957 mL1.9783 mL3.9566 mL19.7832 mL
20 mM0.1978 mL0.9892 mL1.9783 mL9.8916 mL
50 mM0.0791 mL0.3957 mL0.7913 mL3.9566 mL
100 mM0.0396 mL0.1978 mL0.3957 mL1.9783 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
TargetMol | Animal experimentsFor example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH2O. So your working solution concentration is 2 mg/mL。
Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH2OTargetMol | reagent mix well and clarify
For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.
1 Enter information below:
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μL
2 Enter the in vivo formulation:
% DMSO
%
% Tween 80
% Saline/PBS/ddH2O

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Keywords

Efaroxan Hydrochloride
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