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Efaroxan hydrochloride
🥰Excellent
Catalog No. T22760Cas No. 89197-00-2
Alias RX821037 hydrochloride, RX 821037 hydrochloride
Efaroxan hydrochloride is the salt form of Efaroxan, a selective, orally available α2-adrenoceptor antagonist that raises resting plasma insulin levels and significantly potentiates adrenaline-induced increases in insulin levels.
Efaroxan hydrochloride
🥰Excellent
Catalog No. T22760Alias RX821037 hydrochloride, RX 821037 hydrochlorideCas No. 89197-00-2
Efaroxan hydrochloride is the salt form of Efaroxan, a selective, orally available α2-adrenoceptor antagonist that raises resting plasma insulin levels and significantly potentiates adrenaline-induced increases in insulin levels.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 2 mg | $29 | In Stock |
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Product Introduction
Bioactivity
Chemical Properties
| Description | Efaroxan hydrochloride is the salt form of Efaroxan, a selective, orally available α2-adrenoceptor antagonist that raises resting plasma insulin levels and significantly potentiates adrenaline-induced increases in insulin levels. |
| In vitro | Efaroxan hydrochloride binds to 1-imidazoline and α2-adrenergic receptors in the ventrolateral medulla membrane of the cephalic bull with Ki values of 0.15 nM and 5.6 nM, respectively. [1] |
| Alias | RX821037 hydrochloride, RX 821037 hydrochloride |
| Molecular Weight | 252.74 |
| Formula | C13H17ClN2O |
| Cas No. | 89197-00-2 |
| Smiles | Cl.N1=C(NCC1)C2(OC=3C=CC=CC3C2)CC |
| Relative Density. | no data available |
Storage & Solubility Information
| Storage | keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
| Solubility Information | H2O: 40 mg/mL (158.27 mM), Sonication is recommended. | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
H2O
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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