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Asenapine hydrochloride
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Catalog No. T22589Cas No. 1261398-77-9
Alias Org 5222 hydrochloride
Asenapine hydrochloride (Org 5222 hydrochloride) is a 5-hydroxytryptamine receptor, adrenergic receptor, dopamine receptor and histamine receptor antagonist with antipsychotic effects used in neurological disorders such as schizophrenia and bipolar disorder.
Asenapine hydrochloride
😃Good
Catalog No. T22589Alias Org 5222 hydrochlorideCas No. 1261398-77-9
Asenapine hydrochloride (Org 5222 hydrochloride) is a 5-hydroxytryptamine receptor, adrenergic receptor, dopamine receptor and histamine receptor antagonist with antipsychotic effects used in neurological disorders such as schizophrenia and bipolar disorder.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $69 | 7-10 days |
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Product Introduction
Bioactivity
Chemical Properties
| Description | Asenapine hydrochloride (Org 5222 hydrochloride) is a 5-hydroxytryptamine receptor, adrenergic receptor, dopamine receptor and histamine receptor antagonist with antipsychotic effects used in neurological disorders such as schizophrenia and bipolar disorder. |
| Targets&IC50 | 5-HT2C receptor:0.03 nM (Ki), D2 receptor:1.3 nM (Ki), 5-HT2A receptor:0.06 nM (Ki), 5-HT7 receptor:0.13 nM (Ki), sPLA2:2.5 nM (Ki), D4 receptor:1.1 nM (Ki), D3 receptor:0.42 nM (Ki) |
| In vitro | Asenapine hydrochloride acts as an antagonist of 5-HT2A receptors and D2 receptors, commonly used in research related to neurological disorders[2]. |
| Synonyms | Org 5222 hydrochloride |
| Molecular Weight | 322.23 |
| Formula | C17H17Cl2NO |
| Cas No. | 1261398-77-9 |
| Smiles | Cl.[H][C@]12CN(C)C[C@]1([H])c1cc(Cl)ccc1Oc1ccccc21 |
| Relative Density. | no data available |
| Color | Green |
| Appearance | Solid |
Storage & Solubility Information
| Storage | store at low temperature | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature. | ||||||||||
| Solubility Information | DMSO: 1 mg/mL (3.10 mM), Sonication is recommended. | ||||||||||
Solution Preparation Table | |||||||||||
DMSO
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In Vivo Formulation Calculator (Clear solution)
Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . A total of 10 animals were administered, and the formula you used is 5% 
DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH2O. So your working solution concentration is 2 mg/mL。Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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