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TD-5471
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Catalog No. T207120Cas No. 530084-87-8
TD-5471 is a potent and selective full agonist of the human β2 adrenergic receptor.
TD-5471
😃Good
Catalog No. T207120Cas No. 530084-87-8
TD-5471 is a potent and selective full agonist of the human β2 adrenergic receptor.
| Pack Size | Price | USA Warehouse | Global Warehouse | Quantity |
|---|---|---|---|---|
| 10 mg | Inquiry | 10-14 weeks | 10-14 weeks | |
| 50 mg | Inquiry | 10-14 weeks | 10-14 weeks |
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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]
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Product Introduction
Bioactivity
Chemical Properties
| Description | TD-5471 is a potent and selective full agonist of the human β2 adrenergic receptor. |
| In vitro | TD-5471 acts slowly in an in vitro guinea pig trachea model but exhibits strong efficacy. In the guinea pig tracheal ring test, TD-5471 has a pEC50 of 8.7. Structurally distinct from Milveterol, TD-5471's prolonged action duration aligns with the hydrophobicity observed in other long-acting β2-agonist research projects. |
| In vivo | TD-5471 demonstrates a dose-dependent and prolonged pharmacological effect in a bronchoprotection model in guinea pigs. It exhibits excellent efficacy in this model, specifically observed 1.5 hours after aerosol administration. The bronchoprotective effect mediated by TD-5471 persists for up to 72 hours, exhibiting a clear dose-dependence. |
| Molecular Weight | 521.61 |
| Formula | C32H31N3O4 |
| Cas No. | 530084-87-8 |
| Smiles | [C@@H](CNCCC1=CC=C(NC2=CC(=C(OC)C=C2)C3=CC=CC=C3)C=C1)(O)C4=C5C(=C(O)C=C4)NC(=O)C=C5 |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature. |
Calculator
In Vivo Formulation Calculator (Clear solution)
Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . A total of 10 animals were administered, and the formula you used is 5% 
DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH2O. So your working solution concentration is 2 mg/mL。Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
Dose Conversion
You can also refer to dose conversion for different animals. More Dose Conversion
Tech Support
Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc
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