T12244 |
Norverapamil
|
67018-85-3
|
98%
|
|
Norverapamil is a blocker of L-type calcium channel and an inhibitor of P-glycoprotein (P-gp) function .
|
TN3042 |
4-Hydroxycinnamamide
|
194940-15-3
|
98%
|
|
4-Hydroxycinnamamide has antioxidant activity. 4-Hydroxycinnamamide derivatives are specific inhibitors of tyrosine-specific protein kinases.
|
T2S0118 |
Daurinoline
|
2831-75-6
|
98%
|
|
Daurinoline is a non-competitive antagonist, it exerts marked relaxation effect on basilar artery of rabbits through non-competitive antagonism, it would have a ...
|
T15301 |
Fluspirilene
|
1841-19-6
|
98%
|
|
Fluspirilene is a non-competitive L-type calcium channel antagonist (IC50: 0.03 μM). It is a long-acting injectable depot antipsychotic drug used for schizophren...
|
T12153 |
N-type calcium channel blocker-1
|
241499-17-2
|
98%
|
|
N-type calcium channel blocker-1 is an orally active analgesic agent,shows high affinity to functionally block N-type calcium channels.
|
T7009 |
Soyacerebroside II
|
115074-93-6
|
98%
|
|
Soyacerebroside II exhibits ionophoretic activity for Ca2+ ion. Soyacerebrosides I and II have modulating the cellular immune response effects, they show obvious...
|
T12625 |
(R)-Lercanidipine-d3 hydrochloride
|
1217724-52-1
|
98%
|
|
(R)-lercanidipine D3 hydrochloride is a deuterium labeled (R)-Lercanidipine hydrochloride. (R)-Lercanidipine D3 (hydrochloride) is a calcium channel blocker.
|
T12880 |
Semotiadil recemate fumarate
|
123388-25-0
|
98%
|
|
Semotiadil recemate fumarate is the recemate of Semotiadil fumarate. Semotiadil fumarate is a novel antagonist of vasoselective Ca2+ channel.
|
T4001 |
Euxanthone
|
529-61-3
|
98%
|
|
Euxanthone has vasorelaxation effect, may be through multiple pathways involved PKC-mediated signal pathway and calcium-independent pathway, it induces its vasod...
|
TN3319 |
9-Hydroxycanthin-6-one
|
138544-91-9
|
98%
|
|
9-Hydroxycanthin-6-one might be the active component that contributed to the aphrodisiac effect of E. longifolia by antagonizing the smooth muscle tone of CC as ...
|
T12108 |
MRS1845
|
544478-19-5
|
98%
|
|
MRS1845 is a selective inhibitor of store-operated calcium (SOC) channel (IC50 of 1.7 μM).
|
T16887 |
Sipatrigine
|
130800-90-7
|
98%
|
|
Sipatrigine is a glutamate release inhibitor and voltage-dependent sodium channel.
|
TN1367 |
Alismol
|
87827-55-2
|
98%
|
|
Alismol has antihypertensive action, it decreases cardiac output, heart rate and left ventricular pressure, but it increases coronary flow, it has been used for ...
|
T16357 |
NSC 663284
|
383907-43-5
|
98%
|
|
NSC 663284 is a cell-permeable and irreversible Cdc25 dual specificity phosphatase inhibitor (IC50 for Cdc25B2: 0.21 μM). NSC 663284 inhibits NSD2 (IC50 of 170 n...
|
TN2287 |
Turkesterone
|
41451-87-0
|
98%
|
|
Turkesterone is a phytoecdysteroid possessing an 11alpha-hydroxyl group, also is an analogue of the insect steroid hormone 20-hydroxyecdysone. It has immunomodul...
|
TN4303 |
Isokaempferide
|
1592-70-7
|
98%
|
|
Isokaempferide shows hepatoprotective, antiproliferative, and anti-inflammatory effects, the anti-inflammatory effects can be explained, at least in part, by red...
|
TN2116 |
Pteropodine
|
5629-60-7
|
98%
|
|
Pteropodine acts as a positive modulator of muscarinic M(1) and 5-HT(2) receptors. Pteropodine shows antigenotoxic, antioxidant and lymphocyte induction effects,...
|
TN5234 |
Vindorosine
|
5231-60-7
|
98%
|
|
Vindorosine has blood vessel relaxation effect, possible underlying mechanisms involving the inhibition of Ca(2+) entry via L-type Ca(2+) channels in vascular sm...
|
T12322 |
ORM-10962
|
763926-98-3
|
98%
|
|
ORM-10962 is a potent, highly selective inhibitor of sodium-calcium exchanger (NCX) (for the reverse and forward mode inhibition with IC50 values of 67 and 55 nM...
|
T12358 |
Palonidipine
|
96515-73-0
|
98%
|
|
Palonidipine is an antagonist of calcium, is potential for the therapy of angina-pectoris and hypertension.
|