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PD0176078

Name: PD0176078
Brand: TargetMol
SKU: T12385
Price: 57 USD
Availability: InStock
Rating: 5 (10 reviews)

🥰Excellent

Catalog No. T12385Cas No. 248922-46-5

Alias PD176078

PD0176078 () is a newly blocker of N-type Calcium channel.

PD0176078

🥰Excellent

Purity: 99.72%

Catalog No. T12385Alias PD176078Cas No. 248922-46-5

PD0176078 () is a newly blocker of N-type Calcium channel.

Pack Size	Price	Availability
1 mg	$57	In Stock
5 mg	$113	In Stock
10 mg	$190	In Stock
25 mg	$298	In Stock
50 mg	$416	In Stock
100 mg	$572	In Stock
200 mg	$773	In Stock
1 mL x 10 mM (in DMSO)	$141	In Stock

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Bulk & Custom

This molecule is a custom-made product. TargetMol has an excellent synthesis team with the experience and capability to provide you with cost-effective products. However, due to objective factors, there is a small probability that the synthesis may not be successful during the R&D process. We appreciate your understanding. If you have any questions, please feel free to contact us. We are committed to serving you wholeheartedly.

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Batch Information

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Purity:99.72%

Resource Download

COA LCMS HNMR

Product Introduction

Bioactivity

Description	PD0176078 () is a newly blocker of N-type Calcium channel.
Synonyms	PD176078

Chemical Properties

Molecular Weight	388.49
Formula	C₂₃H₃₀F₂N₂O
Cas No.	248922-46-5
Smiles	C(CCCNC([C@H](CC(C)C)NC)=O)(C1=CC=C(F)C=C1)C2=CC=C(F)C=C2
Relative Density.	1.083 g/cm3 (Predicted)

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 50 mg/mL (128.7 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.5741 mL	12.8703 mL	25.7407 mL	128.7034 mL
5 mM	0.5148 mL	2.5741 mL	5.1481 mL	25.7407 mL
10 mM	0.2574 mL	1.2870 mL	2.5741 mL	12.8703 mL
20 mM	0.1287 mL	0.6435 mL	1.2870 mL	6.4352 mL
50 mM	0.0515 mL	0.2574 mL	0.5148 mL	2.5741 mL
100 mM	0.0257 mL	0.1287 mL	0.2574 mL	1.2870 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc