tpa — TargetMol Chemicals

Cat No.	Product Name	Synonyms	Targets
T17144	TPA 023		GABA Receptor
	TPA 023 is a selective agonist of GABAA α2/α3 subtype (Kis = 0.19 - 0.41 nM).		GABA Receptor
T13192	TPA-023B		Others
	TPA-023B is an orally active and high-affinity agonist of the GABAA receptor α2/α3 subtype (Kis: 0.73 nM/2 nM) partial and an antagonist α1 subtype (Ki: 1.8 nM), has non-sedating anxiolytic-like properties.		Others
TN1025	3,29-O-Dibenzoyloxykarounidiol		Others
	3,29-O-Dibenzoyloxykarounidiol is a natural product with regulate blood sugar level, has potent inhibitory effects on Epstein-Barr virus early antigen (EBV-EA) induced by tumor promoter 12-O-tetradecanoylphorbol-13-aceta...		Others
TQ0198	Phorbol 12-myristate 13-acetate	PMA	NF-κB , S1P Receptor , PKC
	Phorbol 12-myristate 13-acetate (PMA) belongs to the phorbol ester group of natural products and is an activator of PKC, SphK, and NF-κB. Phorbol 12-myristate 13-acetate induces THP1 cell differentiation.		NF-κB , S1P Receptor , PKC
T9882	RUVBL1/2 ATPase-IN-1		Others
	RUVBL1/2 ATPase-IN-1 is an effective RUVBL1/2 ATPase inhibitor with IC50 values of 6.0 and 7.7 μM, respectively. RUVBL1/2 ATPase-IN-1 can be used in cancer disease studies.		Others
T12692	RAS GTPase inhibitor 1		Raf
	RAS GTPase inhibitor 1 is a RAS GTPase inhibitor with potential antitumor activity.		Raf
T83967	ATPase-IN-3		ATPase
	ATPase-IN-3 is an ATPase (ATPase) inhibitor that can be used in the study of metabolism-related diseases.		ATPase
T67967	EOB-DTPA	N-((2s)-2-(bis(carboxymethyl)amino)-3-(4-ethoxyphenyl)propyl)-n-(2-(bis(carboxymethyl)amino)ethyl)glycine	Others
	EOB-DTPA is a biochemical reagent that can be synthesized from other compounds and is commonly used in MRI.		Others
T82561	Di-DTPA TL
	Di-DTPA TL, a hydrophilic bivalent hapten derived from DTPA, is utilized in tumor research [1].
TP2287	Rac GTPase fragment		Others
	Rac GTPase fragment is a peptide with the sequence H2N-Val-Phe-Asp-Glu-Ala-Ile-Arg-Ala-Val-OH, MW= 1019.15. Rac is a subfamily of the Rho family of GTPases, small signaling G proteins (more specifically a GTPase).		Others
T61553	ATPase-IN-2
	ATPase-IN-2 is a compound that acts as an inhibitor of ATPase, with an IC50 value of 0.9 μM. It also inhibits the glycohydrolase activity of C. difficile toxin B (TcdB) with an AC50 value of 30.91 μM. ATPase-IN-2 is comm...
T27350	Fosmetpantotenate	RE-024,RE024,RE 024
	Fosmetpantotenate, a immunomodulator, is used for treatment of Pantothenate Kinase Associated Neurodegeneration (PKAN).
T81252	RTQLLWTPAAPTAMA TFA
	RTQLLWTPAAPTAMA TFA is a peptide-based antigen employed for enhancing drug delivery within the context of immunological responses [1].
T78239	Mergetpa		Carboxypeptidase
	Mergetpa, a carboxypeptidase inhibitor, impedes the conversion of kinins and B2 receptor antagonists into metabolites devoid of the C-terminal arginine [1].		Carboxypeptidase
T73237	GTPA2-OMe
	gTPA2-OMe is a potential hole transport layer candidate for perovskite solar cells (PSCs).
T19270	DTPA-DAB2		Others
	DAB2-DTPA is a conjugate of DTPA and two DABs used in the photooxidation experiment.		Others
TNU0612	S-2-(4-Aminobenzyl)-diethylenetriamine pentaacetic acid TFA salt, p-NH2-Bn-DTPA-TFA
	Super-chelating agent & MRI contrast agent
T10405	ATPA		Others
	ATPA is a selective glutamate receptor GluR5 activator (EC50s: 0.66, 1.4, 9.5, 23, 32, 18, and 14 μM for GluR5wt, GluR5(S721T), GluR5(S741M), GluR5(S721T, S741M), GluR5(S741A), GluR5(S741L), and GluR5(S741V)).		Others
T81433	P-NH2-CHX-A"-DTPA
	p-NH2-CHX-A"-DTPA is a bifunctional chelating agent [1].
T7604	Valrubicin	Valstar,AD-32	Antibiotic , PKC
	Valrubicin (AD-32) (AD 32) inhibits TPA- and PDBu-induced PKC activation (IC50s: 0.85 and 1.25 μM) and has antitumor and anti-inflammatory activity.		Antibiotic , PKC