Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Compound 121, a D3R/MOR antagonist with K i values of 361 nM and 85.2 nM for D3R and MOR respectively, has the potential for analgesic effects through MOR partial agonism and may reduce opioid-misuse liability through D3R antagonism [1].
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Description | Compound 121, a D3R/MOR antagonist with K i values of 361 nM and 85.2 nM for D3R and MOR respectively, has the potential for analgesic effects through MOR partial agonism and may reduce opioid-misuse liability through D3R antagonism [1]. |
Molecular Weight | 410.98 |
Formula | C25H31ClN2O |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
You can also refer to dose conversion for different animals. More
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D3R/MOR antagonist 2 GPCR/G Protein Neuroscience Dopamine Receptor inhibitor inhibit