Brexpiprazole S-oxide

Name: Brexpiprazole S-oxide
Brand: TargetMol
SKU: T10612
Rating: 4.5 (1 reviews)

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Catalog No. T10612Cas No. 1191900-51-2

Alias DM-3411

Brexpiprazole S-oxide (DM-3411), a primary metabolite of Brexpiprazole, acts as a partial agonist of human 5-HT1A and dopamine receptors with Ki values of 0.12 nM and 0.3 nM, respectively.

Brexpiprazole S-oxide

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Catalog No. T10612Alias DM-3411Cas No. 1191900-51-2

Brexpiprazole S-oxide (DM-3411), a primary metabolite of Brexpiprazole, acts as a partial agonist of human 5-HT1A and dopamine receptors with Ki values of 0.12 nM and 0.3 nM, respectively.

Pack Size	Price	USA Warehouse	Global Warehouse
25 mg	Inquiry	3-6 months	3-6 months
50 mg	Inquiry	3-6 months	3-6 months
100 mg	Inquiry	3-6 months	3-6 months

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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]

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Product Introduction

Bioactivity

Description	Brexpiprazole S-oxide (DM-3411), a primary metabolite of Brexpiprazole, acts as a partial agonist of human 5-HT1A and dopamine receptors with Ki values of 0.12 nM and 0.3 nM, respectively.
Targets&IC50	5-HT1A:ki： 0.12 nM , D2L:0.3 nM (ki), 5-HT2A:0.47 nM (ki)
Synonyms	DM-3411

Chemical Properties

Molecular Weight	449.57
Formula	C₂₅H₂₇N₃O₃S
Cas No.	1191900-51-2
Smiles	O=C1C=CC=2C=CC(OCCCCN3CCN(C4=CC=CC5=C4C=CS5=O)CC3)=CC2N1
Relative Density.	1.38 g/cm3 (Predicted)

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

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Stock solution preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

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Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

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