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Remoxipride hydrochloride

🥰Excellent
Catalog No. T23232Cas No. 73220-03-8
Alias Remoxipride Hydrochloride Anhydrous, (S)-Remoxipride Hydrochloride

Remoxipride hydrochloride (Roxiam) is a selective antagonist of D2 receptor with IC50s of 1.57 μM, ＞100 μM and 42 μM for D2 receptor, D1 receptor and α1-adrenoceptor.

Remoxipride hydrochloride
Other Forms of Remoxipride hydrochloride:

Remoxipride hydrochloride

🥰Excellent
Purity: 99.88%
Catalog No. T23232Alias Remoxipride Hydrochloride Anhydrous, (S)-Remoxipride HydrochlorideCas No. 73220-03-8
Remoxipride hydrochloride (Roxiam) is a selective antagonist of D2 receptor with IC50s of 1.57 μM, ＞100 μM and 42 μM for D2 receptor, D1 receptor and α1-adrenoceptor.
Pack SizePriceUSA WarehouseGlobal WarehouseQuantity
1 mg$39In StockIn Stock
5 mg$89In StockIn Stock
10 mg$139In StockIn Stock
25 mg$278In StockIn Stock
50 mg$419In StockIn Stock
100 mg$619In StockIn Stock
500 mg$1,280-In Stock
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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]
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Purity:99.88%
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Product Introduction

Bioactivity
Description
Remoxipride hydrochloride (Roxiam) is a selective antagonist of D2 receptor with IC50s of 1.57 μM, ＞100 μM and 42 μM for D2 receptor, D1 receptor and α1-adrenoceptor.
In vivo
In male Sprague-Dawley rats, Remoxipride hydrochloride (0.1-100 μM/kg; i.p.) blockes apomorphine-induced hyperactivity and dose-dependent blockades apomorphine-induced behaviors. In beagle dogs, Remoxipride hydrochloride (0.25-5 μM/kg; gavage) blockes apomorphine-induced vomiting[1].
SynonymsRemoxipride Hydrochloride Anhydrous, (S)-Remoxipride Hydrochloride
Chemical Properties
Molecular Weight407.73
FormulaC16H24BrClN2O3
Cas No.73220-03-8
SmilesC(NC[C@H]1N(CC)CCC1)(=O)C2=C(OC)C(Br)=CC=C2OC.Cl
Relative Density.no data available
ColorWhite
AppearanceSolid
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
Solubility Information
H2O: 40.9 mg/mL (100.31 mM), Sonication is recommended.
Solution Preparation Table
H2O
1mg5mg10mg50mg
1 mM2.4526 mL12.2630 mL24.5260 mL122.6302 mL
5 mM0.4905 mL2.4526 mL4.9052 mL24.5260 mL
10 mM0.2453 mL1.2263 mL2.4526 mL12.2630 mL
20 mM0.1226 mL0.6132 mL1.2263 mL6.1315 mL
50 mM0.0491 mL0.2453 mL0.4905 mL2.4526 mL
100 mM0.0245 mL0.1226 mL0.2453 mL1.2263 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
TargetMol | Animal experimentsFor example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH2O. So your working solution concentration is 2 mg/mL。
Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH2OTargetMol | reagent mix well and clarify
For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.
1 Enter information below:
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2 Enter the in vivo formulation:
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Keywords

Remoxipride HydrochlorideDopamineReceptorDopamine ReceptorD2 receptor
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