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Remoxipride hydrochloride

Name: Remoxipride hydrochloride
Brand: TargetMol
SKU: T23232
Price: 39 USD
Availability: InStock
Rating: 5 (10 reviews)

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Catalog No. T23232Cas No. 73220-03-8

Alias Remoxipride Hydrochloride Anhydrous, (S)-Remoxipride Hydrochloride

Remoxipride hydrochloride (Roxiam) is a selective antagonist of D2 receptor with IC50s of 1.57 μM, ＞100 μM and 42 μM for D2 receptor, D1 receptor and α1-adrenoceptor.

Remoxipride hydrochloride

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Purity: 99.88%

Catalog No. T23232Alias Remoxipride Hydrochloride Anhydrous, (S)-Remoxipride HydrochlorideCas No. 73220-03-8

Remoxipride hydrochloride (Roxiam) is a selective antagonist of D2 receptor with IC50s of 1.57 μM, ＞100 μM and 42 μM for D2 receptor, D1 receptor and α1-adrenoceptor.

Pack Size	Price	USA Warehouse	Global Warehouse
1 mg	$39	In Stock	In Stock
5 mg	$89	In Stock	In Stock
10 mg	$139	In Stock	In Stock
25 mg	$278	In Stock	In Stock
50 mg	$419	In Stock	In Stock
100 mg	$619	In Stock	In Stock
500 mg	$1,280	-	In Stock

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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]

All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.

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Purity:99.88%

Appearance:Solid

Color:White

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COA HNMR LCMS

Product Introduction

Bioactivity

Description	Remoxipride hydrochloride (Roxiam) is a selective antagonist of D2 receptor with IC50s of 1.57 μM, ＞100 μM and 42 μM for D2 receptor, D1 receptor and α1-adrenoceptor.
In vivo	In male Sprague-Dawley rats, Remoxipride hydrochloride (0.1-100 μM/kg; i.p.) blockes apomorphine-induced hyperactivity and dose-dependent blockades apomorphine-induced behaviors. In beagle dogs, Remoxipride hydrochloride (0.25-5 μM/kg; gavage) blockes apomorphine-induced vomiting[1].
Synonyms	Remoxipride Hydrochloride Anhydrous, (S)-Remoxipride Hydrochloride

Chemical Properties

Molecular Weight	407.73
Formula	C₁₆H₂₄BrClN₂O₃
Cas No.	73220-03-8
Smiles	C(NC[C@H]1N(CC)CCC1)(=O)C2=C(OC)C(Br)=CC=C2OC.Cl
Relative Density.	no data available

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

H2O: 40.9 mg/mL (100.31 mM), Sonication is recommended.

Solution Preparation Table

H2O

	1mg	5mg	10mg	50mg
1 mM	2.4526 mL	12.2630 mL	24.5260 mL	122.6302 mL
5 mM	0.4905 mL	2.4526 mL	4.9052 mL	24.5260 mL
10 mM	0.2453 mL	1.2263 mL	2.4526 mL	12.2630 mL
20 mM	0.1226 mL	0.6132 mL	1.2263 mL	6.1315 mL
50 mM	0.0491 mL	0.2453 mL	0.4905 mL	2.4526 mL
100 mM	0.0245 mL	0.1226 mL	0.2453 mL	1.2263 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the stock solution preparation method and in vivo formula preparation method:

For example, if the intended dosage is 10 mg/kg for animals weighing 20 g , with a dosing volume of 100 μL per animal, TargetMol | Animal experiments

and a total of 10 animals are to be administered, using a formulation of TargetMol | reagent

10% DMSO+ 40% PEG300+ 5% Tween 80+ 45% Saline/PBS/ddH₂O , the resulting working solution concentration would be 2 mg/mL.

Stock Solution Preparation:

Dissolve 2 mg of the compound in 100 μL DMSO TargetMol | reagent to obtain a stock solution at a concentration of 20 mg/mL . If the required concentration exceeds the compound's known solubility, please contact us for technical support before proceeding.

Preparation of the In Vivo Formulation:

1) Add 100 μL of the DMSO TargetMol | reagent stock solution to 400 μL PEG300 and mix thoroughly until the solution becomes clear.

2) Add 50 μL Tween 80 and mix well until fully clarified.

3) Add 450 μL Saline,PBS or ddH₂O TargetMol | reagent and mix thoroughly until a homogeneous solution is obtained.

This example is provided solely to demonstrate the use of the In Vivo Formulation Calculator and does not constitute a recommended formulation for any specific compound. Please select an appropriate dissolution and formulation strategy based on your experimental model and route of administration.

All co-solvents required for this protocol, includingDMSO, PEG300/PEG400, Tween 80, SBE-β-CD, and Corn oil, are available for purchase on the TargetMol website.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc