T13463L2 |
Dihydrexidine hydrochloride
|
137417-08-4
|
98%
|
|
Dihydrexidine hydrochloride is a full efficacy D1-like dopamine receptor (D1/D5) agonist (IC50: 10 nM for D1 receptor). It also shows potent antiparkinsonian act...
|
TQ0175 |
Dexpramipexole
|
104632-28-2
|
98%
|
|
Dexpramipexole (KNS-760704, R-(+)-Pramipexole) is a neuroprotective agent and weak non-ergoline dopamine agonist.
|
T13570 |
Benzamide Derivative 1
|
108226-05-7
|
98%
|
|
Benzamide Derivative 1, extracted from patent EP0213775A1 (compound 18), may be useful in the treatment of gastrointestinal disorders.
|
T15744 |
Levophacetoperane hydrochloride
|
23257-56-9
|
98%
|
|
Levophacetoperane inhibits in vitro in a competitive manner. It also can norepinephrine uptake and dopamine uptake.
|
T6142 |
PD128907 HCl
|
112960-16-4
|
98%
|
|
PD 128907 HCl is a potent and selective dopamine D3 receptor agonist, with EC50 of 0.64 nM, exhibits 53-fold selectivity over dopamine D2 receptor.
|
T13898 |
SPD-473 citrate
|
161190-26-7
|
98%
|
|
SPD-473 citrate is an inhibitior of serotonin/dopamine/norepinephrine reuptake.
|
T3426 |
Bacoside A
|
11028-00-5
|
98%
|
|
Bacoside A has a possible anticancer activity that could be inducing cell cycle arrest and apoptosis through Notch pathway in GBM in vitro. It exerts cytoprotect...
|
T12252 |
NRA-0160
|
204718-47-8
|
98%
|
|
NRA-0160 is a selective antagonist of dopamine D4 receptor(Ki of 0.48 nM)
|
T0338 |
Minaprine
|
25905-77-5
|
98%
|
|
Minaprine is a reversible inhibitor of MAO-A, used in the treatment of various depressive states.
|
T12606 |
Quinpirole Hydrochloride
|
85798-08-9
|
98%
|
|
Quinpirole Hydrochloride is a high-affinity dopamine D2/D3 receptor agonist.
|
T15339 |
Foscarbidopa
|
1907685-81-7
|
98%
|
|
Foscarbidopa is a prodrug of Carbidopa. It acts as a dopamine receptor agonist.
|
T12861L |
SB-277011 dihydrochloride
|
1226917-67-4
|
98%
|
|
SB-277011 dihydrochloride is a potent, selective, orally bioavailable and brain penetrate antagonist of dopamine D3 receptor(pKis of 8.0, 6.0, <5.2 and 5.9 for D...
|
T12676 |
(Rac)-Rotigotine hydrochloride
|
102120-99-0
|
98%
|
|
(Rac)-Rotigotine hydrochloride is a racemate of Rotigotine. Rotigotine is a full agonist of dopamine receptor, a partial the 5-HT1A receptor agonist.
|
T13245 |
UCSF924
|
1434515-70-4
|
98%
|
|
UCSF924 is a potent and specific agonist of dopamine D4 receptor (DRD4) partial (EC50: 4.2 nM, Ki: 3 nM).
|
T14088 |
ABT-670
|
630119-43-6
|
98%
|
|
ABT-670 is a selective agonist of dopamine D4 receptor. For human D4, ferret D4, and rat D4, the EC50 values are 89 nM, 160 nM, and 93 nM , respectively.
|
T1769 |
Pardoprunox
|
269718-84-5
|
98%
|
|
Pardoprunox is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist properties. Pardoprunox has been used in trials studying the...
|
T10837L |
Clocapramine
|
47739-98-0
|
98%
|
|
Clocapramine is a D2 and 5-HT2A receptors antagonist.
|
T10681 |
Cariprazine D6
|
T10681
|
98%
|
|
Cariprazine D6 (RGH-188 D6) is a deuterium-labeled Cariprazine. Cariprazine is an antipsychotic agent (D3 receptors, Ki: 0.085 nM; D2 receptors, Ki: 0.49 nM).
|
T15100 |
Desmethyl cariprazine
|
839712-15-1
|
98%
|
|
Desmethyl cariprazine is a Cariprazine active metabolite. Cariprazine, an antipsychotic drug candidate, shows a high affinity for the D3 (Ki: 0.085 nM) and D2 (K...
|
T2S1397 |
L-Stepholidine
|
16562-13-3
|
98%
|
|
L-Stepholidine, which has dual actions on dopamine D1 and D2 receptors, attenuates heroin self-administration and cue-induced reinstatement. It also elicits anti...
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