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Dopamine Receptor

Dopamine receptors are a class of G protein-coupled receptors that are prominent in the vertebrate central nervous system (CNS). Dopamine receptors activate different effectors through not only G-protein coupling, but also signaling through different protein (dopamine receptor-interacting proteins) interactions.
Cat. No. Product name CAS No. Purity Chemical Structure
T13463L2 Dihydrexidine hydrochloride 137417-08-4 98%
Dihydrexidine hydrochloride is a full efficacy D1-like dopamine receptor (D1/D5) agonist (IC50: 10 nM for D1 receptor). It also shows potent antiparkinsonian act...
TQ0175 Dexpramipexole 104632-28-2 98%
Dexpramipexole (KNS-760704, R-(+)-Pramipexole) is a neuroprotective agent and weak non-ergoline dopamine agonist.
T13570 Benzamide Derivative 1 108226-05-7 98%
Benzamide Derivative 1, extracted from patent EP0213775A1 (compound 18), may be useful in the treatment of gastrointestinal disorders.
T15744 Levophacetoperane hydrochloride 23257-56-9 98%
Levophacetoperane inhibits in vitro in a competitive manner. It also can norepinephrine uptake and dopamine uptake.
T6142 PD128907 HCl 112960-16-4 98%
PD 128907 HCl is a potent and selective dopamine D3 receptor agonist, with EC50 of 0.64 nM, exhibits 53-fold selectivity over dopamine D2 receptor.
T13898 SPD-473 citrate 161190-26-7 98%
SPD-473 citrate is an inhibitior of serotonin/dopamine/norepinephrine reuptake.
T3426 Bacoside A 11028-00-5 98%
Bacoside A has a possible anticancer activity that could be inducing cell cycle arrest and apoptosis through Notch pathway in GBM in vitro. It exerts cytoprotect...
T12252 NRA-0160 204718-47-8 98%
NRA-0160 is a selective antagonist of dopamine D4 receptor(Ki of 0.48 nM)
T0338 Minaprine 25905-77-5 98%
Minaprine is a reversible inhibitor of MAO-A, used in the treatment of various depressive states.
T12606 Quinpirole Hydrochloride 85798-08-9 98%
Quinpirole Hydrochloride is a high-affinity dopamine D2/D3 receptor agonist.
T15339 Foscarbidopa 1907685-81-7 98%
Foscarbidopa is a prodrug of Carbidopa. It acts as a dopamine receptor agonist.
T12861L SB-277011 dihydrochloride 1226917-67-4 98%
SB-277011 dihydrochloride is a potent, selective, orally bioavailable and brain penetrate antagonist of dopamine D3 receptor(pKis of 8.0, 6.0, <5.2 and 5.9 for D...
T12676 (Rac)-Rotigotine hydrochloride 102120-99-0 98%
(Rac)-Rotigotine hydrochloride is a racemate of Rotigotine. Rotigotine is a full agonist of dopamine receptor, a partial the 5-HT1A receptor agonist.
T13245 UCSF924 1434515-70-4 98%
UCSF924 is a potent and specific agonist of dopamine D4 receptor (DRD4) partial (EC50: 4.2 nM, Ki: 3 nM).
T14088 ABT-670 630119-43-6 98%
ABT-670 is a selective agonist of dopamine D4 receptor. For human D4, ferret D4, and rat D4, the EC50 values are 89 nM, 160 nM, and 93 nM , respectively.
T1769 Pardoprunox 269718-84-5 98%
Pardoprunox is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist properties. Pardoprunox has been used in trials studying the...
T10837L Clocapramine 47739-98-0 98%
Clocapramine is a D2 and 5-HT2A receptors antagonist.
T10681 Cariprazine D6 T10681 98%
Cariprazine D6 (RGH-188 D6) is a deuterium-labeled Cariprazine. Cariprazine is an antipsychotic agent (D3 receptors, Ki: 0.085 nM; D2 receptors, Ki: 0.49 nM).
T15100 Desmethyl cariprazine 839712-15-1 98%
Desmethyl cariprazine is a Cariprazine active metabolite. Cariprazine, an antipsychotic drug candidate, shows a high affinity for the D3 (Ki: 0.085 nM) and D2 (K...
T2S1397 L-Stepholidine 16562-13-3 98%
L-Stepholidine, which has dual actions on dopamine D1 and D2 receptors, attenuates heroin self-administration and cue-induced reinstatement. It also elicits anti...
Dihydrexidine hydrochloride
T13463L2
Dihydrexidine hydrochloride is a full efficacy D1-like dopamine receptor (D1/D5) agonist (IC50: 10 nM for D1 receptor). It also shows potent antiparkinsonian act...
Dexpramipexole
TQ0175
Dexpramipexole (KNS-760704, R-(+)-Pramipexole) is a neuroprotective agent and weak non-ergoline dopamine agonist.
Benzamide Derivative 1
T13570
Benzamide Derivative 1, extracted from patent EP0213775A1 (compound 18), may be useful in the treatment of gastrointestinal disorders.
Levophacetoperane hydrochloride
T15744
Levophacetoperane inhibits in vitro in a competitive manner. It also can norepinephrine uptake and dopamine uptake.
PD128907 HCl
T6142
PD 128907 HCl is a potent and selective dopamine D3 receptor agonist, with EC50 of 0.64 nM, exhibits 53-fold selectivity over dopamine D2 receptor.
SPD-473 citrate
T13898
SPD-473 citrate is an inhibitior of serotonin/dopamine/norepinephrine reuptake.
Bacoside A
T3426
Bacoside A has a possible anticancer activity that could be inducing cell cycle arrest and apoptosis through Notch pathway in GBM in vitro. It exerts cytoprotect...
NRA-0160
T12252
NRA-0160 is a selective antagonist of dopamine D4 receptor(Ki of 0.48 nM)
Minaprine
T0338
Minaprine is a reversible inhibitor of MAO-A, used in the treatment of various depressive states.
Quinpirole Hydrochloride
T12606
Quinpirole Hydrochloride is a high-affinity dopamine D2/D3 receptor agonist.
Foscarbidopa
T15339
Foscarbidopa is a prodrug of Carbidopa. It acts as a dopamine receptor agonist.
SB-277011 dihydrochloride
T12861L
SB-277011 dihydrochloride is a potent, selective, orally bioavailable and brain penetrate antagonist of dopamine D3 receptor(pKis of 8.0, 6.0, <5.2 and 5.9 for D...
(Rac)-Rotigotine hydrochloride
T12676
(Rac)-Rotigotine hydrochloride is a racemate of Rotigotine. Rotigotine is a full agonist of dopamine receptor, a partial the 5-HT1A receptor agonist.
UCSF924
T13245
UCSF924 is a potent and specific agonist of dopamine D4 receptor (DRD4) partial (EC50: 4.2 nM, Ki: 3 nM).
ABT-670
T14088
ABT-670 is a selective agonist of dopamine D4 receptor. For human D4, ferret D4, and rat D4, the EC50 values are 89 nM, 160 nM, and 93 nM , respectively.
Pardoprunox
T1769
Pardoprunox is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist properties. Pardoprunox has been used in trials studying the...
Clocapramine
T10837L
Clocapramine is a D2 and 5-HT2A receptors antagonist.
Cariprazine D6
T10681
Cariprazine D6 (RGH-188 D6) is a deuterium-labeled Cariprazine. Cariprazine is an antipsychotic agent (D3 receptors, Ki: 0.085 nM; D2 receptors, Ki: 0.49 nM).
Desmethyl cariprazine
T15100
Desmethyl cariprazine is a Cariprazine active metabolite. Cariprazine, an antipsychotic drug candidate, shows a high affinity for the D3 (Ki: 0.085 nM) and D2 (K...
L-Stepholidine
T2S1397
L-Stepholidine, which has dual actions on dopamine D1 and D2 receptors, attenuates heroin self-administration and cue-induced reinstatement. It also elicits anti...
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