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Compounds

Cat No. Product Name
T10201 PDE IV-IN-1 PDE
PDE IV-IN-1 是一种有效的磷酸二酯酶4 (PDE4)抑制剂,具有抗炎活性,可用于治疗哮喘,慢性阻塞性肺病和其他炎症性疾病,是研究抑郁症的潜在化合物。
T68191 PDE-I2
PDE-I2 is a parasite schizogony inhibitor.
T12389 PDE-9 inhibitor Others
PDE-9 inhibitor is used for treatment neurodegenerative diseases.
T5411 PDE10-IN-1 SEP-0372814 PDE
SEP-0372814 是一种高效的 PDE10抑制剂,摘自专利 WO 2013192273 A1。
T12395 PDE9-IN-1 PDE
PDE9-IN-1 是一种选择性和口服生物可利用的 PDE9A 抑制剂(IC50 为 8.7 nM)。
T36832 PDE4B-IN-2 A 33 PDE
PDE4B-IN-2 是一种具有口服活性,选择性 PDE4B 抑制剂,IC50 为 15 nM。PDE4B-IN-2 抑制 PDE4D (IC50=1.7 µM)。PDE4B-IN-2 表现出有效的抗炎作用。
T8659 K-Ras-PDEδ-IN-1 PDE
K-Ras-PDEδ-IN-1 是新型的 K-Ras-PDEδ 抑制剂,它能够以低纳摩尔Kd8 nM 与 PDEδ 的法尼基结合袋竞争性结合。
T28352 PDE9-IN-(S)-C33 (S)-C33 PDE
PDE9-IN-(S)-C33 是一种有效的选择性 PDE9 抑制剂 (IC50 = 11 nM)。 PDE9-IN-(S)-C33 可用于中枢神经系统疾病和糖尿病的相关研究。
T18529 PDEC-NB 4-Nitrophenyl 2-(Pyridin-2-Yldisulfanyl)Ethyl Carbonate Others
PDEC-NB 是用于抗体-药物偶联物的二硫键可切割接头。
T12391 PDE1-IN-3 Others
PDE1-IN-3 is a selective inhibitor of human phosphodiesterase 1 (PDE1).
T12392 PDE12-IN-3 Others
PDE12-IN-3 is an inhibitor of phosphodiesterase 12 (PDE12) (pXC50 of 7.68),with antiviral activity.
T12390 PDE1-IN-2 Others
PDE1-IN-2 is an PDE1 inhibitor(PDE1C, PDE1B and PDE1A with IC50 values of 6, 140 and 164 nM, respectvely).
T12394 PDE5-IN-2 PDE
PDE5-IN-2 is a potent, highly selective, and orally active inhibitor of PDE5(IC50 of 0.31 nM)
T10028 PDE4 inhibitor intermediate 1 Others
PDE4 inhibitor intermediate 1 is a PDE4 inhibitor synthesis intermediate.
T12393 PDE2/PDE10-IN-1 Others
PDE2/PDE10-IN-1 is a inhibitor of phosphodiesterase 2 (PDE2) and PDE10(IC50s of 29 and 480 nM, respectively).
T39796 PDE12-IN-1 PDE12-IN-1
PDE12-IN-1 is a powerful and specific inhibitor of PDE12, exhibiting a pIC 50 value of 9.1 for enzyme inhibition. It eff...
T24605 PDE5-IN-6c PDE5IN6c,PDE5 inhibitor 6c
PDE5-IN-6c is a potent and selective inhibitor of PDE5A1.
T24606 PDE7 inhibitor S14 S14,PDE7 inhibitor-S14
PDE7 inhibitor S14 is a cell-permeable PDE7 inhibitor that acts by targeting the cyclic adenosine monophosphate (cAMP)/c...
T40356 PDE4-IN-3 PDE4-IN-3
PDE4-IN-3 is a newly developed oral compound that acts as a potent inhibitor of the enzyme phosphodiesterase 4 (PDE4), d...
T40278 PDE2A-IN-1 PDE2A-IN-1
PDE2A-IN-1 is a phosphodiesterase 2A (PDE2A) inhibitor with an IC 50 value of 1.3 nM.
PDE IV-IN-1
T10201
synonym:
Target:
PDE-I2
T68191
synonym:
Target:
PDE-9 inhibitor
T12389
synonym:
Target:
PDE10-IN-1
T5411
synonym: SEP-0372814
Target:
PDE9-IN-1
T12395
synonym:
Target:
PDE4B-IN-2
T36832
synonym: A 33
Target:
K-Ras-PDEδ-IN-1
T8659
synonym:
Target:
PDE9-IN-(S)-C33
T28352
synonym: (S)-C33
Target:
PDEC-NB
T18529
synonym: 4-Nitrophenyl 2-(Pyridin-2-Yldisulfanyl)Ethyl Carbonate
Target:
PDE1-IN-3
T12391
synonym:
Target:
PDE12-IN-3
T12392
synonym:
Target:
PDE1-IN-2
T12390
synonym:
Target:
PDE5-IN-2
T12394
synonym:
Target:
PDE4 inhibitor intermediate 1
T10028
synonym:
Target:
PDE2/PDE10-IN-1
T12393
synonym:
Target:
PDE12-IN-1
T39796
synonym: PDE12-IN-1
Target:
PDE5-IN-6c
T24605
synonym: PDE5IN6c,PDE5 inhibitor 6c
Target:
PDE7 inhibitor S14
T24606
synonym: S14,PDE7 inhibitor-S14
Target:
PDE4-IN-3
T40356
synonym: PDE4-IN-3
Target:
PDE2A-IN-1
T40278
synonym: PDE2A-IN-1
Target:
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